Exploring the molecular determinants for subtype-selectivity of 2-amino-1,4,5,6-tetrahydropyrimidine-5-carboxylic acid analogs as betaine/GABA transporter 1 (BGT1) substrate-inhibi...

por Kickinger, Stefanie, Al-Khawaja, Anas, Haugaard, Anne Stæhr, Lie, Maria E. K., Bavo, Francesco, Löffler, Rebekka, Damgaard, Maria, Ecker, Gerhard F., Frølund, Bente, Wellendorph, Petrine
Publicado 2020

Molecular Determinants and Pharmacological Analysis for a Class of Competitive Non-transported Bicyclic Inhibitors of the Betaine/GABA Transporter BGT1

por Kickinger, Stefanie, Lie, Maria E. K., Suemasa, Akihiro, Al-Khawaja, Anas, Fujiwara, Koichi, Watanabe, Mizuki, Wilhelmsen, Kristine S., Falk-Petersen, Christina B., Frølund, Bente, Shuto, Satoshi, Ecker, Gerhard F., Wellendorph, Petrine
Publicado 2021