Click chemistry approaches for developing carbonic anhydrase inhibitors and their applications

por Angeli, Andrea, Supuran, Claudiu T.
Publicado 2023

Five-Membered Heterocyclic Sulfonamides as Carbonic Anhydrase Inhibitors

por Angeli, Andrea, Paoletti, Niccolò, Supuran, Claudiu T.
Publicado 2023

Benzamide-4-Sulfonamides Are Effective Human Carbonic Anhydrase I, II, VII, and IX Inhibitors

por Abdoli, Morteza, Bozdag, Murat, Angeli, Andrea, Supuran, Claudiu T.
Publicado 2018

Inhibition of Schistosoma mansoni carbonic anhydrase by the antiparasitic drug clorsulon: X-ray crystallographic and in vitro studies

por Ferraroni, Marta, Angeli, Andrea, Carradori, Simone, Supuran, Claudiu T.
Publicado 2022

Psychoactive substances belonging to the amphetamine class potently activate brain carbonic anhydrase isoforms VA, VB, VII, and XII

por Angeli, Andrea, Vaiano, Fabio, Mari, Francesco, Bertol, Elisabetta, Supuran, Claudiu T.
Publicado 2017

Synthesis and biological evaluation of novel 8-substituted quinoline-2-carboxamides as carbonic anhydrase inhibitors

por Thacker, Pavitra S., Shaikh, Pirpasha, Angeli, Andrea, Arifuddin, Mohammed, Supuran, Claudiu T.
Publicado 2019

Pharmacological Inhibition of CA-IX Impairs Tumor Cell Proliferation, Migration and Invasiveness

por Ciccone, Valerio, Filippelli, Arianna, Angeli, Andrea, Supuran, Claudiu T., Morbidelli, Lucia
Publicado 2020

Diversely N-substituted benzenesulfonamides dissimilarly bind to human carbonic anhydrases: crystallographic investigations of N-nitrosulfonamides

por Angeli, Andrea, Ferraroni, Marta, Bonardi, Alessandro, Supuran, Claudiu T., Nocentini, Alessio
Publicado 2023

Investigation of piperazines as human carbonic anhydrase I, II, IV and VII activators

por Angeli, Andrea, Chiaramonte, Niccolò, Manetti, Dina, Romanelli, Maria Novella, Supuran, Claudiu T.
Publicado 2017

Novel thiazolidinone-containing compounds, without the well-known sulphonamide zinc-binding group acting as human carbonic anhydrase IX inhibitors

por Güzel-Akdemir, Özlen, Angeli, Andrea, Demir, Kübra, Supuran, Claudiu T., Akdemir, Atilla
Publicado 2018

Activation studies with amino acids and amines of a β-carbonic anhydrase from Mammaliicoccus (Staphylococcus) sciuri previously annotated as Staphylococcus aureus (SauBCA) carbonic...

por Angeli, Andrea, Urbański, Linda J, Capasso, Clemente, Parkkila, Seppo, Supuran, Claudiu T.
Publicado 2022

Synthesis carbonic anhydrase enzyme inhibition and antioxidant activity of novel benzothiazole derivatives incorporating glycine, methionine, alanine, and phenylalanine moieties

por Payaz, Deniz Üzeroğlu, Küçükbay, F. Zehra, Küçükbay, Hasan, Angeli, Andrea, Supuran, Claudiu T.
Publicado 2018

Activation Effects of Carnosine- and Histidine-Containing Dipeptides on Human Carbonic Anhydrases: A Comprehensive Study

por Vistoli, Giulio, Aldini, Giancarlo, Fumagalli, Laura, Dallanoce, Clelia, Angeli, Andrea, Supuran, Claudiu T.
Publicado 2020

Novel Indole-Based Hydrazones as Potent Inhibitors of the α-class Carbonic Anhydrase from Pathogenic Bacterium Vibrio cholerae

por Demir-Yazıcı, Kübra, Güzel-Akdemir, Özlen, Angeli, Andrea, Supuran, Claudiu T., Akdemir, Atilla
Publicado 2020

Activation of the β-carbonic anhydrase from the protozoan pathogen Trichomonas vaginalis with amines and amino acids

por Angeli, Andrea, Urbański, Linda J., Hytönen, Vesa P., Parkkila, Seppo, Supuran, Claudiu T.
Publicado 2021

Selenocarbamates As a Prodrug‐Based Approach to Carbonic Anhydrase Inhibition

por Angeli, Andrea, Ferraroni, Marta, Capperucci, Antonella, Tanini, Damiano, Costantino, Gabriele, Supuran, Claudiu T.
Publicado 2022

Synthesis of Sulfonamides Incorporating Piperidinyl-Hydrazidoureido and Piperidinyl-Hydrazidothioureido Moieties and Their Carbonic Anhydrase I, II, IX and XII Inhibitory Activity

por Moi, Davide, Deplano, Alessandro, Angeli, Andrea, Balboni, Gianfranco, Supuran, Claudiu T., Onnis, Valentina
Publicado 2022

Investigation on Hydrazonobenzenesulfonamides as Human Carbonic Anhydrase I, II, IX and XII Inhibitors

por Moi, Davide, Vittorio, Serena, Angeli, Andrea, Balboni, Gianfranco, Supuran, Claudiu T., Onnis, Valentina
Publicado 2022

Novel 2-indolinones containing a sulfonamide moiety as selective inhibitors of candida β-carbonic anhydrase enzyme

por Akdemir, Atilla, Angeli, Andrea, Göktaş, Füsun, Eraslan Elma, Pınar, Karalı, Nilgün, Supuran, Claudiu T.
Publicado 2019

Crystal structure and chemical inhibition of essential schistosome host-interactive virulence factor carbonic anhydrase SmCA

por Da’dara, Akram A., Angeli, Andrea, Ferraroni, Marta, Supuran, Claudiu T., Skelly, Patrick J.
Publicado 2019