Computational Tool for Fast in silico Evaluation of hERG K(+) Channel Affinity

por Chemi, Giulia, Gemma, Sandra, Campiani, Giuseppe, Brogi, Simone, Butini, Stefania, Brindisi, Margherita
Publicado 2017

A Therapeutic Perspective of HDAC8 in Different Diseases: An Overview of Selective Inhibitors

por Fontana, Anna, Cursaro, Ilaria, Carullo, Gabriele, Gemma, Sandra, Butini, Stefania, Campiani, Giuseppe
Publicado 2022

Multiple Targeting Approaches on Histamine H(3) Receptor Antagonists

por Khanfar, Mohammad A., Affini, Anna, Lutsenko, Kiril, Nikolic, Katarina, Butini, Stefania, Stark, Holger
Publicado 2016

The FAAH inhibitor URB597 suppresses hippocampal maximal dentate afterdischarges and restores seizure-induced impairment of short and long-term synaptic plasticity

por Colangeli, Roberto, Pierucci, Massimo, Benigno, Arcangelo, Campiani, Giuseppe, Butini, Stefania, Di Giovanni, Giuseppe
Publicado 2017

Author Correction: The FAAH inhibitor URB597 suppresses hippocampal maximal dentate afterdischarges and restores seizure-induced impairment of short and long-term synaptic plastici...

por Colangeli, Roberto, Pierucci, Massimo, Benigno, Arcangelo, Campiani, Giuseppe, Butini, Stefania, Di Giovanni, Giuseppe
Publicado 2018

Author Correction: The FAAH inhibitor URB597 suppresses hippocampal maximal dentate afterdischarges and restores seizure-induced impairment of short and long-term synaptic plastici...

por Colangeli, Roberto, Pierucci, Massimo, Benigno, Arcangelo, Campiani, Giuseppe, Butini, Stefania, Di Giovanni, Giuseppe
Publicado 2018

Dopamine D3 Receptor Antagonists as Potential Therapeutics for the Treatment of Neurological Diseases

por Maramai, Samuele, Gemma, Sandra, Brogi, Simone, Campiani, Giuseppe, Butini, Stefania, Stark, Holger, Brindisi, Margherita
Publicado 2016

A Repurposing Approach for Uncovering the Anti-Tubercular Activity of FDA-Approved Drugs with Potential Multi-Targeting Profiles

por Battah, Basem, Chemi, Giulia, Butini, Stefania, Campiani, Giuseppe, Brogi, Simone, Delogu, Giovanni, Gemma, Sandra
Publicado 2019

Covalent Reversible Inhibitors of Cysteine Proteases Containing the Nitrile Warhead: Recent Advancement in the Field of Viral and Parasitic Diseases

por Brogi, Simone, Ibba, Roberta, Rossi, Sara, Butini, Stefania, Calderone, Vincenzo, Gemma, Sandra, Campiani, Giuseppe
Publicado 2022

Polypharmacological Approaches for CNS Diseases: Focus on Endocannabinoid Degradation Inhibition

por Papa, Alessandro, Pasquini, Silvia, Contri, Chiara, Gemma, Sandra, Campiani, Giuseppe, Butini, Stefania, Varani, Katia, Vincenzi, Fabrizio
Publicado 2022

The green chemistry of chalcones: Valuable sources of privileged core structures for drug discovery

por Marotta, Ludovica, Rossi, Sara, Ibba, Roberta, Brogi, Simone, Calderone, Vincenzo, Butini, Stefania, Campiani, Giuseppe, Gemma, Sandra
Publicado 2022

In silico study of subtilisin-like protease 1 (SUB1) from different Plasmodium species in complex with peptidyl-difluorostatones and characterization of potent pan-SUB1 inhibitors

por Brogi, Simone, Giovani, Simone, Brindisi, Margherita, Gemma, Sandra, Novellino, Ettore, Campiani, Giuseppe, Blackman, Michael J., Butini, Stefania
Publicado 2016

A non-toxic, reversibly released imaging probe for oral cancer that is derived from natural compounds

por Ghanim, Magda, Relitti, Nicola, McManus, Gavin, Butini, Stefania, Cappelli, Andrea, Campiani, Giuseppe, Mok, K. H., Kelly, Vincent P.
Publicado 2021

The pyrrolo-1,5-benzoxazepine, PBOX-15, enhances TRAIL-induced apoptosis by upregulation of DR5 and downregulation of core cell survival proteins in acute lymphoblastic leukaemia c...

por NATHWANI, SEEMA-MARIA, GREENE, LISA M., BUTINI, STEFANIA, CAMPIANI, GIUSEPPE, WILLIAMS, D. CLIVE, SAMALI, AFSHIN, SZEGEZDI, EVA, ZISTERER, DANIELA M.
Publicado 2016

Development of Quinazolinone Derivatives as Modulators of Virulence Factors of Pseudomonas aeruginosa Cystic Fibrosis Strains

por Carullo, Gabriele, Di Bonaventura, Giovanni, Rossi, Sara, Lupetti, Veronica, Tudino, Valeria, Brogi, Simone, Butini, Stefania, Campiani, Giuseppe, Gemma, Sandra, Pompilio, Arianna
Publicado 2023

Bronchoalveolar-Lavage-Derived Fibroblast Cell Line (B-LSDM7) as a New Protocol for Investigating the Mechanisms of Idiopathic Pulmonary Fibrosis

por Bergantini, Laura, d’Alessandro, Miriana, Gangi, Sara, Cavallaro, Dalila, Campiani, Giuseppe, Butini, Stefania, Landi, Claudia, Bini, Luca, Cameli, Paolo, Bargagli, Elena
Publicado 2022

Identification of Novel 3-Hydroxy-pyran-4-One Derivatives as Potent HIV-1 Integrase Inhibitors Using in silico Structure-Based Combinatorial Library Design Approach

por Sirous, Hajar, Chemi, Giulia, Gemma, Sandra, Butini, Stefania, Debyser, Zeger, Christ, Frauke, Saghaie, Lotfollah, Brogi, Simone, Fassihi, Afshin, Campiani, Giuseppe, Brindisi, Margherita
Publicado 2019

Development of a Multiplexed Activity-Based Protein Profiling Assay to Evaluate Activity of Endocannabinoid Hydrolase Inhibitors

por Janssen, Antonius P. A., van der Vliet, Daan, Bakker, Alexander T., Jiang, Ming, Grimm, Sebastian H., Campiani, Giuseppe, Butini, Stefania, van der Stelt, Mario
Publicado 2018

Total Synthesis of the Natural Chalcone Lophirone E, Synthetic Studies toward Benzofuran and Indole-Based Analogues, and Investigation of Anti-Leishmanial Activity

por Pozzetti, Luca, Ibba, Roberta, Rossi, Sara, Taglialatela-Scafati, Orazio, Taramelli, Donatella, Basilico, Nicoletta, D’Alessandro, Sarah, Parapini, Silvia, Butini, Stefania, Campiani, Giuseppe, Gemma, Sandra
Publicado 2022

Crystal structures of Schistosoma mansoni histone deacetylase 8 reveal a novel binding site for allosteric inhibitors

por Saccoccia, Fulvio, Pozzetti, Luca, Gimmelli, Roberto, Butini, Stefania, Guidi, Alessandra, Papoff, Giuliana, Giannaccari, Marialaura, Brogi, Simone, Scognamiglio, Viviana, Gemma, Sandra, Ruberti, Giovina, Campiani, Giuseppe
Publicado 2022