The Selectivity of Fosfosal for STAT5b over STAT5a is Mediated by Arg566 in the Linker Domain

por Gräb, Julian, Berg, Thorsten
Publicado 2020

Asymmetrically Substituted m‐Terphenyl Phosphates Inhibit the Transcription Factor STAT5a

por Müller‐Klieser, Daniel, Berg, Thorsten
Publicado 2021

Polymer Nanocomposite Ultrafiltration Membranes: The Influence of Polymeric Additive, Dispersion Quality and Particle Modification on the Integration of Zinc Oxide Nanoparticles in...

por van den Berg, Thorsten, Ulbricht, Mathias
Publicado 2020

Stafiba: A STAT5‐Selective Small‐Molecule Inhibitor

por Eckhardt, Katrin S., Münzel, Theresa, Gräb, Julian, Berg, Thorsten
Publicado 2022

Stafia‐1: a STAT5a‐Selective Inhibitor Developed via Docking‐Based Screening of in Silico O‐Phosphorylated Fragments

por Natarajan, Kalaiselvi, Müller‐Klieser, Daniel, Rubner, Stefan, Berg, Thorsten
Publicado 2019

Nanomolar Inhibitors of the Transcription Factor STAT5b with High Selectivity over STAT5a**

por Elumalai, Nagarajan, Berg, Angela, Natarajan, Kalaiselvi, Scharow, Andrej, Berg, Thorsten
Publicado 2015

Effect of Amino Acid Substitutions on 70S Ribosomal Binding, Cellular Uptake, and Antimicrobial Activity of Oncocin Onc112

por Kolano, Lisa, Knappe, Daniel, Berg, Angela, Berg, Thorsten, Hoffmann, Ralf
Publicado 2022

A High-Throughput Fluorescence Polarization-Based Assay for the SH2 Domain of STAT4

por Berg, Angela, Gräber, Martin, Schmutzler, Sebastian, Hoffmann, Ralf, Berg, Thorsten
Publicado 2022

Templated Generation of a Bcl‐x(L) Inhibitor by Isomer‐Free SPAAC Based on Azacyclonon‐5‐yne

por Brauer, Juliane, Mötzing, Marina, Gröst, Corinna, Hoffmann, Ralf, Berg, Thorsten
Publicado 2022

Rational development of Stafib-2: a selective, nanomolar inhibitor of the transcription factor STAT5b

por Elumalai, Nagarajan, Berg, Angela, Rubner, Stefan, Blechschmidt, Linda, Song, Chen, Natarajan, Kalaiselvi, Matysik, Jörg, Berg, Thorsten
Publicado 2017

Serendipitous alkylation of a Plk1 ligand uncovers a new binding channel

por Liu, Fa, Park, Jung-Eun, Qian, Wen-Jian, Lim, Dan, Gräber, Martin, Berg, Thorsten, Yaffe, Michael B., Lee, Kyung S., Burke, Terrence R.
Publicado 2011

Development of Erasin: a chromone-based STAT3 inhibitor which induces apoptosis in Erlotinib-resistant lung cancer cells

por Lis, Christian, Rubner, Stefan, Roatsch, Martin, Berg, Angela, Gilcrest, Tyler, Fu, Darwin, Nguyen, Elizabeth, Schmidt, Anne-Marie, Krautscheid, Harald, Meiler, Jens, Berg, Thorsten
Publicado 2017

MCC1019, a selective inhibitor of the Polo-box domain of Polo-like kinase 1 as novel, potent anticancer candidate

por Abdelfatah, Sara, Berg, Angela, Huang, Qi, Yang, Li Jun, Hamdoun, Sami, Klinger, Anette, Greten, Henry J., Fleischer, Edmond, Berg, Thorsten, Wong, Vincent K.W., Efferth, Thomas
Publicado 2019

GM-CSF-activated STAT5A regulates macrophage functions and inflammation in atherosclerosis

por Nagenborg, Jan, Jin, Han, Ruder, Adele V., Temmerman, Lieve, Mees, Barend, Schalkwijk, Casper, Müller-Klieser, Daniel, Berg, Thorsten, Goossens, Pieter, Donners, Marjo M. P. C., Biessen, Erik A. L.
Publicado 2023