Bioorganometallic derivatives of 4-hydrazino-benzenesulphonamide as carbonic anhydrase inhibitors: synthesis, characterisation and biological evaluation

por Brichet, Jeremie, Arancibia, Rodrigo, Berrino, Emanuela, Supuran, Claudiu T.
Publicado 2020

New sulfonamides containing organometallic-acylhydrazones: synthesis, characterisation and biological evaluation as inhibitors of human carbonic anhydrases

por Huentupil, Yosselin, Peña, Luis, Novoa, Néstor, Berrino, Emanuela, Arancibia, Rodrigo, Supuran, Claudiu T.
Publicado 2019

A class of carbonic anhydrase IX/XII – selective carboxylate inhibitors

por Alhameed, Rakia Abd, Berrino, Emanuela, Almarhoon, Zainab, El-Faham, Ayman, Supuran, Claudiu T.
Publicado 2020

Toxicity evaluation of sulfamides and coumarins that efficiently inhibit human carbonic anhydrases

por Aspatwar, Ashok, Berrino, Emanuela, Bua, Silvia, Carta, Fabrizio, Capasso, Clemente, Parkkila, Seppo, Supuran, Claudiu T.
Publicado 2020

Amine- and Amino Acid-Based Compounds as Carbonic Anhydrase Activators

por Angeli, Andrea, Berrino, Emanuela, Carradori, Simone, Supuran, Claudiu T., Cirri, Marzia, Carta, Fabrizio, Costantino, Gabriele
Publicado 2021

Carbonic Anhydrase Inhibitors of Different Structures Dilate Pre-Contracted Porcine Retinal Arteries

por Eysteinsson, Thor, Gudmundsdottir, Hrönn, Hardarson, Arnar Oessur, Berrino, Emanuela, Selleri, Silvia, Supuran, Claudiu T., Carta, Fabrizio
Publicado 2019

A Novel Class of Dual-Acting DCH-CORMs Counteracts Oxidative Stress-Induced Inflammation in Human Primary Tenocytes

por Appetecchia, Federico, Consalvi, Sara, Berrino, Emanuela, Gallorini, Marialucia, Granese, Arianna, Campestre, Cristina, Carradori, Simone, Biava, Mariangela, Poce, Giovanna
Publicado 2021

Inhibition of α-, β-, γ-, and δ-carbonic anhydrases from bacteria and diatoms with N′-aryl-N-hydroxy-ureas

por Berrino, Emanuela, Bozdag, Murat, Del Prete, Sonia, Alasmary, Fatmah A. S., Alqahtani, Linah S., AlOthman, Zeid, Capasso, Clemente, Supuran, Claudiu T.
Publicado 2018

Synthesis of novel benzenesulfamide derivatives with inhibitory activity against human cytosolic carbonic anhydrase I and II and Vibrio cholerae α- and β-class enzymes

por Bua, Silvia, Berrino, Emanuela, Del Prete, Sonia, Murthy, Vallabhaneni S., Vijayakumar, Vijayaparthasarathi, Tamboli, Yasinalli, Capasso, Clemente, Cerbai, Elisabetta, Mugelli, Alessandro, Carta, Fabrizio, Supuran, Claudiu T.
Publicado 2018

Novel Sulfamide-Containing Compounds as Selective Carbonic Anhydrase I Inhibitors

por Berrino, Emanuela, Bua, Silvia, Mori, Mattia, Botta, Maurizio, Murthy, Vallabhaneni S., Vijayakumar, Vijayaparthasarathi, Tamboli, Yasinalli, Bartolucci, Gianluca, Mugelli, Alessandro, Cerbai, Elisabetta, Supuran, Claudiu T., Carta, Fabrizio
Publicado 2017

Dual Carbonic Anhydrase IX/XII Inhibitors and Carbon Monoxide Releasing Molecules Modulate LPS-Mediated Inflammation in Mouse Macrophages

por Berrino, Emanuela, Carradori, Simone, Angeli, Andrea, Carta, Fabrizio, Supuran, Claudiu T., Guglielmi, Paolo, Coletti, Cecilia, Paciotti, Roberto, Schweikl, Helmut, Maestrelli, Francesca, Cerbai, Elisabetta, Gallorini, Marialucia
Publicado 2021

Zeta-carbonic anhydrases show CS(2) hydrolase activity: A new metabolic carbon acquisition pathway in diatoms?

por Alterio, Vincenzo, Langella, Emma, Buonanno, Martina, Esposito, Davide, Nocentini, Alessio, Berrino, Emanuela, Bua, Silvia, Polentarutti, Maurizio, Supuran, Claudiu T., Monti, Simona Maria, De Simone, Giuseppina
Publicado 2021

Uncovering Novel Capsaicin Inhibitory Activity towards Human Carbonic Anhydrase Isoforms IX and XII by Combining In Silico and In Vitro Studies

por Gualtieri, Gianmarco, Maruca, Annalisa, Rocca, Roberta, Carta, Fabrizio, Berrino, Emanuela, Salatino, Alessandro, Brescia, Carolina, Torcasio, Roberta, Crispo, Manuel, Trapasso, Francesco, Alcaro, Stefano, Supuran, Claudiu T., Costa, Giosuè
Publicado 2023

Tetrahydroquinazole-based secondary sulphonamides as carbonic anhydrase inhibitors: synthesis, biological evaluation against isoforms I, II, IV, and IX, and computational studies

por Baglini, Emma, Ravichandran, Rahul, Berrino, Emanuela, Salerno, Silvia, Barresi, Elisabetta, Marini, Anna Maria, Viviano, Monica, Castellano, Sabrina, Da Settimo, Federico, Supuran, Claudiu T., Cosconati, Sandro, Taliani, Sabrina
Publicado 2021

Novel Insights on Human Carbonic Anhydrase Inhibitors Based on Coumalic Acid: Design, Synthesis, Molecular Modeling Investigation, and Biological Studies

por Pontecorvi, Virginia, Mori, Mattia, Picarazzi, Francesca, Zara, Susi, Carradori, Simone, Cataldi, Amelia, Angeli, Andrea, Berrino, Emanuela, Chimenti, Paola, Ciogli, Alessia, Secci, Daniela, Guglielmi, Paolo, Supuran, Claudiu T.
Publicado 2022

In Silico Identification and Biological Evaluation of Antioxidant Food Components Endowed with Human Carbonic Anhydrase IX and XII Inhibition

por Costa, Giosuè, Maruca, Annalisa, Rocca, Roberta, Ambrosio, Francesca Alessandra, Berrino, Emanuela, Carta, Fabrizio, Mesiti, Francesco, Salatino, Alessandro, Lanzillotta, Delia, Trapasso, Francesco, Artese, Anna, Alcaro, Stefano, Supuran, Claudiu T.
Publicado 2020

Azidothymidine “Clicked” into 1,2,3-Triazoles: First Report on Carbonic Anhydrase–Telomerase Dual-Hybrid Inhibitors

por Berrino, Emanuela, Angeli, Andrea, Zhdanov, Dmitry D., Kiryukhina, Anna P., Milaneschi, Andrea, De Luca, Alessandro, Bozdag, Murat, Carradori, Simone, Selleri, Silvia, Bartolucci, Gianluca, Peat, Thomas S., Ferraroni, Marta, Supuran, Claudiu T., Carta, Fabrizio
Publicado 2020