Novel 1,2,4-Oxadiazole Derivatives in Drug Discovery

por Biernacki, Karol, Daśko, Mateusz, Ciupak, Olga, Kubiński, Konrad, Rachon, Janusz, Demkowicz, Sebastian
Publicado 2020

Recent progress in the development of steroid sulphatase inhibitors – examples of the novel and most promising compounds from the last decade

por Daśko, Mateusz, Demkowicz, Sebastian, Biernacki, Karol, Ciupak, Olga, Kozak, Witold, Masłyk, Maciej, Rachon, Janusz
Publicado 2020

Novel 1,2,3-Triazole Derivatives as Mimics of Steroidal System—Synthesis, Crystal Structures Determination, Hirshfeld Surfaces Analysis and Molecular Docking

por Daśko, Mateusz, Dołęga, Anna, Siedzielnik, Magdalena, Biernacki, Karol, Ciupak, Olga, Rachon, Janusz, Demkowicz, Sebastian
Publicado 2021

New potent steroid sulphatase inhibitors based on 6-(1-phenyl-1H-1,2,3-triazol-4-yl)naphthalen-2-yl sulphamate derivatives

por Ciupak, Olga, Daśko, Mateusz, Biernacki, Karol, Rachon, Janusz, Masłyk, Maciej, Kubiński, Konrad, Martyna, Aleksandra, Demkowicz, Sebastian
Publicado 2020

Hydration of Simple Model Peptides in Aqueous Osmolyte Solutions

por Panuszko, Aneta, Pieloszczyk, Maciej, Kuffel, Anna, Jacek, Karol, Biernacki, Karol A., Demkowicz, Sebastian, Stangret, Janusz, Bruździak, Piotr
Publicado 2021

Electron-Induced Decomposition of Uracil-5-yl O-(N,N-dimethylsulfamate): Role of Methylation in Molecular Stability

por Arthur-Baidoo, Eugene, Falkiewicz, Karina, Chomicz-Mańka, Lidia, Czaja, Anna, Demkowicz, Sebastian, Biernacki, Karol, Kozak, Witold, Rak, Janusz, Denifl, Stephan
Publicado 2021

Development of Sulfamoylated 4-(1-Phenyl-1H-1,2,3-triazol-4-yl)phenol Derivatives as Potent Steroid Sulfatase Inhibitors for Efficient Treatment of Breast Cancer

por Biernacki, Karol, Ciupak, Olga, Daśko, Mateusz, Rachon, Janusz, Kozak, Witold, Rak, Janusz, Kubiński, Konrad, Masłyk, Maciej, Martyna, Aleksandra, Śliwka-Kaszyńska, Magdalena, Wietrzyk, Joanna, Świtalska, Marta, Nocentini, Alessio, Supuran, Claudiu T., Demkowicz, Sebastian
Publicado 2022

Intramolecular Proton Transfer in the Radical Anion of Cytidine Monophosphate Sheds Light on the Sensitivities of Dry vs Wet DNA to Electron Attachment-Induced Damage

por Chomicz-Mańka, Lidia, Czaja, Anna, Falkiewicz, Karina, Zdrowowicz, Magdalena, Biernacki, Karol, Demkowicz, Sebastian, Izadi, Farhad, Arthur-Baidoo, Eugene, Denifl, Stephan, Zhu, Zhaoguo, Tufekci, Burak Ahmet, Harris, Rachel, Bowen, Kit H., Rak, Janusz
Publicado 2023