The 2′-Trifluoromethyl Analogue of Indomethacin Is a Potent and Selective COX-2 Inhibitor

por Blobaum, Anna L., Uddin, Md. Jashim, Felts, Andrew S., Crews, Brenda C., Rouzer, Carol A., Marnett, Lawrence J.
Publicado 2013

Cyclooxygenase-1-Selective Inhibitors Based on the (E)-2′-Des-methyl-sulindac Sulfide Scaffold

por Liedtke, Andy J., Crews, Brenda C., Daniel, Cristina M., Blobaum, Anna L., Kingsley, Philip J., Ghebreselasie, Kebreab, Marnett, Lawrence J.
Publicado 2012

Conservative Secondary Shell Substitution In Cyclooxygenase-2 Reduces Inhibition by Indomethacin Amides and Esters via Altered Enzyme Dynamics

por Konkle, Mary E., Blobaum, Anna L., Moth, Christopher W., Prusakiewicz, Jeffery J., Xu, Shu, Ghebreselasie, Kebreab, Akingbade, Dapo, Jacobs, Aaron T., Rouzer, Carol A., Lybrand, Terry P., Marnett, Lawrence J.
Publicado 2015

Discovery of N-(5-Fluoropyridin-2-yl)-6-methyl-4-(pyrimidin-5-yloxy)picolinamide (VU0424238): A Novel Negative Allosteric Modulator of Metabotropic Glutamate Receptor Subtype 5 Sel...

por Felts, Andrew S., Rodriguez, Alice L., Blobaum, Anna L., Morrison, Ryan D., Bates, Brittney S., Thompson Gray, Analisa, Rook, Jerri M., Tantawy, Mohammed N., Byers, Frank W., Chang, Sichen, Venable, Daryl F., Luscombe, Vincent B., Tamagnan, Gilles D., Niswender, Colleen M., Daniels, J. Scott, Jones, Carrie K., Conn, P. Jeffrey, Lindsley, Craig W., Emmitte, Kyle A.
Publicado 2017