Inhibition studies of the protozoan α-carbonic anhydrase from Trypanosoma cruzi with phenols

por Bonardi, Alessandro, Parkkila, Seppo, Supuran, Claudiu T.
Publicado 2022

4-Cyanamidobenzenesulfonamide derivatives: a novel class of human and bacterial carbonic anhydrase inhibitors

por Abdoli, Morteza, Bonardi, Alessandro, Supuran, Claudiu T., Žalubovskis, Raivis
Publicado 2022

Investigation of novel alkyl/benzyl (4-sulphamoylphenyl)carbamimidothioates as carbonic anhydrase inhibitors

por Abdoli, Morteza, Bonardi, Alessandro, Supuran, Claudiu T., Žalubovskis, Raivis
Publicado 2023

Discovery of the first-in-class potent and isoform-selective human carbonic anhydrase III inhibitors

por Giovannuzzi, Simone, Bonardi, Alessandro, Gratteri, Paola, Nocentini, Alessio, Supuran, Claudiu T.
Publicado 2023

Isocoumarins: a new class of selective carbonic anhydrase IX and XII inhibitors

por Onyılmaz, Mehmet, Koca, Murat, Bonardi, Alessandro, Degirmenci, Mustafa, Supuran, Claudiu T.
Publicado 2022

Diversely N-substituted benzenesulfonamides dissimilarly bind to human carbonic anhydrases: crystallographic investigations of N-nitrosulfonamides

por Angeli, Andrea, Ferraroni, Marta, Bonardi, Alessandro, Supuran, Claudiu T., Nocentini, Alessio
Publicado 2023

Steroids interfere with human carbonic anhydrase activity by using alternative binding mechanisms

por Nocentini, Alessio, Bonardi, Alessandro, Gratteri, Paola, Cerra, Bruno, Gioiello, Antimo, Supuran, Claudiu T.
Publicado 2018

Pharmaceutical strategies for preventing toxicity and promoting antioxidant and anti-inflammatory actions of bilirubin

por Nocentini, Alessio, Bonardi, Alessandro, Pratesi, Simone, Gratteri, Paola, Dani, Carlo, Supuran, Claudiu T.
Publicado 2022

The antibiotic furagin and its derivatives are isoform-selective human carbonic anhydrase inhibitors

por Pustenko, Aleksandrs, Nocentini, Alessio, Gratteri, Paola, Bonardi, Alessandro, Vozny, Igor, Žalubovskis, Raivis, Supuran, Claudiu T.
Publicado 2020

Evaluation of docking procedures reliability in affitins-partners interactions

por Ranaudo, Anna, Cosentino, Ugo, Greco, Claudio, Moro, Giorgio, Bonardi, Alessandro, Maiocchi, Alessandro, Moroni, Elisabetta
Publicado 2022

Discovery of Novel Hydroxyimine-Tethered Benzenesulfonamides as Potential Human Carbonic Anhydrase IX/XII Inhibitors

por Peerzada, Mudasir Nabi, Vullo, Daniela, Paoletti, Niccolò, Bonardi, Alessandro, Gratteri, Paola, Supuran, Claudiu T., Azam, Amir
Publicado 2023

Inhibition Studies on Human and Mycobacterial Carbonic Anhydrases with N-((4-Sulfamoylphenyl)carbamothioyl) Amides

por Abdoli, Morteza, Bonardi, Alessandro, Paoletti, Niccolò, Aspatwar, Ashok, Parkkila, Seppo, Gratteri, Paola, Supuran, Claudiu T., Žalubovskis, Raivis
Publicado 2023

Development of Hydrogen Sulfide-Releasing Carbonic Anhydrases IX- and XII-Selective Inhibitors with Enhanced Antihyperalgesic Action in a Rat Model of Arthritis

por Bonardi, Alessandro, Micheli, Laura, Di Cesare Mannelli, Lorenzo, Ghelardini, Carla, Gratteri, Paola, Nocentini, Alessio, Supuran, Claudiu T.
Publicado 2022

Probing the Efficiency of 13-Pyridylalkyl Berberine Derivatives to Human Telomeric G-Quadruplexes Binding: Spectroscopic, Solid State and In Silico Analysis

por Bazzicalupi, Carla, Bonardi, Alessandro, Biver, Tarita, Ferraroni, Marta, Papi, Francesco, Savastano, Matteo, Lombardi, Paolo, Gratteri, Paola
Publicado 2022

Selenium-analogs based on natural sources as cancer-associated carbonic anhydrase isoforms IX and XII inhibitors

por Astrain-Redin, Nora, Paoletti, Niccolò, Plano, Daniel, Bonardi, Alessandro, Gratteri, Paola, Angeli, Andrea, Sanmartin, Carmen, Supuran, Claudiu T.
Publicado 2023

Sulphonamide inhibition studies of the β-carbonic anhydrase GsaCAβ present in the salmon platyhelminth parasite Gyrodactylus salaris

por Aspatwar, Ashok, Bonardi, Alessandro, Aisala, Heidi, Zueva, Ksenia, Primmer, Craig R, Lumme, Jaakko, Parkkila, Seppo, Supuran, Claudiu T.
Publicado 2023

Dependence on linkers’ flexibility designed for benzenesulfonamides targeting discovery of novel hCA IX inhibitors as potent anticancer agents

por Tawfik, Haytham O., Belal, Amany, Abourehab, Mohammed A. S., Angeli, Andrea, Bonardi, Alessandro, Supuran, Claudiu T., El-Hamamsy, Mervat H.
Publicado 2022

Novel insights on saccharin- and acesulfame-based carbonic anhydrase inhibitors: design, synthesis, modelling investigations and biological activity evaluation

por Guglielmi, Paolo, Rotondi, Giulia, Secci, Daniela, Angeli, Andrea, Chimenti, Paola, Nocentini, Alessio, Bonardi, Alessandro, Gratteri, Paola, Carradori, Simone, Supuran, Claudiu T.
Publicado 2020

Inhibition of α-, β- and γ-carbonic anhydrases from the pathogenic bacterium Vibrio cholerae with aromatic sulphonamides and clinically licenced drugs – a joint docking/molecular d...

por Bonardi, Alessandro, Nocentini, Alessio, Osman, Sameh Mohamed, Alasmary, Fatmah Ali, Almutairi, Tahani Mazyad, Abdullah, Dalal Saied, Gratteri, Paola, Supuran, Claudiu T.
Publicado 2021

Synthesis, biological evaluation and theoretical studies of (E)-1-(4-sulfamoyl-phenylethyl)-3-arylidene-5-aryl-1H-pyrrol-2(3H)-ones as human carbonic anhydrase inhibitors

por Ramzan, Farhat, Nabi, Syed Ayaz, Lone, Mehak Saba, Bonardi, Alessandro, Hamid, Aabid, Bano, Sameena, Sharma, Kalicharan, Shafi, Syed, Samim, Mohammed, Javed, Kalim, Supran, Claudiu T.
Publicado 2023