Structure-Based Virtual Screening of Ultra-Large Library Yields Potent Antagonists for a Lipid GPCR

por Sadybekov, Arman A., Brouillette, Rebecca L., Marin, Egor, Sadybekov, Anastasiia V., Luginina, Aleksandra, Gusach, Anastasiia, Mishin, Alexey, Besserer-Offroy, Élie, Longpré, Jean-Michel, Borshchevskiy, Valentin, Cherezov, Vadim, Sarret, Philippe, Katritch, Vsevolod
Publicado 2020

Data set describing the in vitro biological activity of JMV2009, a novel silylated neurotensin(8–13) analog

por Besserer-Offroy, Élie, Tétreault, Pascal, Brouillette, Rebecca L, René, Adeline, Murza, Alexandre, Fanelli, Roberto, Kirby, Karyn, Parent, Alexandre, Dubuc, Isabelle, Beaudet, Nicolas, Côté, Jérôme, Longpré, Jean-Michel, Martinez, Jean, Cavelier, Florine, Sarret, Philippe
Publicado 2020

Structural basis of ligand selectivity and disease mutations in cysteinyl leukotriene receptors

por Gusach, Anastasiia, Luginina, Aleksandra, Marin, Egor, Brouillette, Rebecca L., Besserer-Offroy, Élie, Longpré, Jean-Michel, Ishchenko, Andrii, Popov, Petr, Patel, Nilkanth, Fujimoto, Taku, Maruyama, Toru, Stauch, Benjamin, Ergasheva, Margarita, Romanovskaia, Daria, Stepko, Anastasiia, Kovalev, Kirill, Shevtsov, Mikhail, Gordeliy, Valentin, Han, Gye Won, Katritch, Vsevolod, Borshchevskiy, Valentin, Sarret, Philippe, Mishin, Alexey, Cherezov, Vadim
Publicado 2019

Structure-based mechanism of cysteinyl leukotriene receptor inhibition by antiasthmatic drugs

por Luginina, Aleksandra, Gusach, Anastasiia, Marin, Egor, Mishin, Alexey, Brouillette, Rebecca, Popov, Petr, Shiriaeva, Anna, Besserer-Offroy, Élie, Longpré, Jean-Michel, Lyapina, Elizaveta, Ishchenko, Andrii, Patel, Nilkanth, Polovinkin, Vitaly, Safronova, Nadezhda, Bogorodskiy, Andrey, Edelweiss, Evelina, Hu, Hao, Weierstall, Uwe, Liu, Wei, Batyuk, Alexander, Gordeliy, Valentin, Han, Gye Won, Sarret, Philippe, Katritch, Vsevolod, Borshchevskiy, Valentin, Cherezov, Vadim
Publicado 2019