Approval of oliceridine (TRV130) for intravenous use in moderate to severe pain in adults

por Lambert, David, Calo, Girolamo
Publicado 2020

The Insect Type 1 Tyramine Receptors: From Structure to Behavior

por Finetti, Luca, Roeder, Thomas, Calò, Girolamo, Bernacchia, Giovanni
Publicado 2021

NOP receptor pharmacological profile – A dynamic mass redistribution study

por Malfacini, Davide, Simon, Katharina, Trapella, Claudio, Guerrini, Remo, Zaveri, Nurulain T., Kostenis, Evi, Calo’, Girolamo
Publicado 2018

Pharmacological Investigations of N-Substituent Variation in Morphine and Oxymorphone: Opioid Receptor Binding, Signaling and Antinociceptive Activity

por Ben Haddou, Tanila, Béni, Szabolcs, Hosztafi, Sándor, Malfacini, Davide, Calo, Girolamo, Schmidhammer, Helmut, Spetea, Mariana
Publicado 2014

Pharmacological profile of the neuropeptide S receptor: Dynamic mass redistribution studies

por Ruzza, Chiara, Ferrari, Federica, Guerrini, Remo, Marzola, Erika, Preti, Delia, Reinscheid, Rainer K., Calo, Girolamo
Publicado 2018

Biased versus Partial Agonism in the Search for Safer Opioid Analgesics

por Azevedo Neto, Joaquim, Costanzini, Anna, De Giorgio, Roberto, Lambert, David G., Ruzza, Chiara, Calò, Girolamo
Publicado 2020

Functional Selectivity Does Not Predict Antinociceptive/Locomotor Impairing Potencies of NOP Receptor Agonists

por Azevedo Neto, Joaquim, Ruzza, Chiara, Sturaro, Chiara, Malfacini, Davide, Pacifico, Salvatore, Zaveri, Nurulain T., Calò, Girolamo
Publicado 2021

Hyaluronic Acid Induces Activation of the κ-Opioid Receptor

por Zavan, Barbara, Ferroni, Letizia, Giorgi, Carlotta, Calò, Girolamo, Brun, Paola, Cortivo, Roberta, Abatangelo, Giovanni, Pinton, Paolo
Publicado 2013

Functional selectivity of EM-2 analogs at the mu-opioid receptor

por Piekielna-Ciesielska, Justyna, Malfacini, Davide, Djeujo, Francine Medjiofack, Marconato, Chantal, Wtorek, Karol, Calo’, Girolamo, Janecka, Anna
Publicado 2023

A diastereoselective synthesis of Cebranopadol, a novel analgesic showing NOP/mu mixed agonism

por Fantinati, Anna, Bianco, Sara, Guerrini, Remo, Salvadori, Severo, Pacifico, Salvatore, Cerlesi, Maria Camilla, Calo, Girolamo, Trapella, Claudio
Publicado 2017

Blockade of nociceptin/orphanin FQ signaling facilitates an active copying strategy due to acute and repeated stressful stimuli in mice

por Holanda, Victor A.D., Oliveira, Matheus C., Da Silva Junior, Edilson D., Calo', Girolamo, Ruzza, Chiara, Gavioli, Elaine C.
Publicado 2020

Biased Agonism at Nociceptin/Orphanin FQ Receptors: A Structure Activity Study on N/OFQ(1–13)-NH(2)

por Pacifico, Salvatore, Ferrari, Federica, Albanese, Valentina, Marzola, Erika, Neto, Joaquim Azevedo, Ruzza, Chiara, Calò, Girolamo, Preti, Delia, Guerrini, Remo
Publicado 2020

Synthesis and Structure-Activity Relationships of (−)-cis-N-Normetazocine-Based LP1 Derivatives

por Pasquinucci, Lorella, Parenti, Carmela, Amata, Emanuele, Georgoussi, Zafiroula, Pallaki, Paschalina, Camarda, Valeria, Calò, Girolamo, Arena, Emanuela, Montenegro, Lucia, Turnaturi, Rita
Publicado 2018

The Nociceptin/Orphanin FQ Receptor Antagonist UFP-101 Reduces Microvascular Inflammation to Lipopolysaccharide In Vivo

por Brookes, Zoë L. S., Stedman, Emily N., Brown, Nicola J., Hebbes, Christopher P., Guerrini, Remo, Calo, Girolamo, Reilly, Charles S., Lambert, David G.
Publicado 2013

Exploring pharmacological activities and signaling of morphinans substituted in position 6 as potent agonists interacting with the μ opioid receptor

por Ben Haddou, Tanila, Malfacini, Davide, Calo, Girolamo, Aceto, Mario D, Harris, Louis S, Traynor, John R, Coop, Andrew, Schmidhammer, Helmut, Spetea, Mariana
Publicado 2014

In vitro and in vivo pharmacological characterization of a neuropeptide S tetrabranched derivative

por Ruzza, Chiara, Rizzi, Anna, Malfacini, Davide, Pulga, Alice, Pacifico, Salvatore, Salvadori, Severo, Trapella, Claudio, Reinscheid, Rainer K, Calo, Girolamo, Guerrini, Remo
Publicado 2015

Pharmacological characterization of cebranopadol a novel analgesic acting as mixed nociceptin/orphanin FQ and opioid receptor agonist

por Rizzi, Anna, Cerlesi, Maria Camilla, Ruzza, Chiara, Malfacini, Davide, Ferrari, Federica, Bianco, Sara, Costa, Tommaso, Guerrini, Remo, Trapella, Claudio, Calo', Girolamo
Publicado 2016

In vitro pharmacological characterization of a novel unbiased NOP receptor‐selective nonpeptide agonist AT‐403

por Ferrari, Federica, Malfacini, Davide, Journigan, Blair V., Bird, Mark F., Trapella, Claudio, Guerrini, Remo, Lambert, David G., Calo', Girolamo, Zaveri, Nurulain T.
Publicado 2017

Pyridostigmine in Pediatric Intestinal Pseudo-obstruction: Case Report of a 2-year Old Girl and Literature Review

por Di Nardo, Giovanni, Viscogliosi, Federica, Esposito, Francesco, Stanghellini, Vincenzo, Villa, Maria Pia, Parisi, Pasquale, Morlando, Alessia, Calò, Girolamo, De Giorgio, Roberto
Publicado 2019

Synthesis and Pharmacological Evaluation of Hybrids Targeting Opioid and Neurokinin Receptors

por Wtorek, Karol, Adamska-Bartłomiejczyk, Anna, Piekielna-Ciesielska, Justyna, Ferrari, Federica, Ruzza, Chiara, Kluczyk, Alicja, Piasecka-Zelga, Joanna, Calo’, Girolamo, Janecka, Anna
Publicado 2019