Insertion of an Amphipathic Linker in a Tetrapodal Tryptophan Derivative Leads to a Novel and Highly Potent Entry Inhibitor of Enterovirus A71 Clinical Isolates

por Martí-Marí, Olaia, Abdelnabi, Rana, Schols, Dominique, Neyts, Johan, Camarasa, María-José, Gago, Federico, San-Félix, Ana
Publicado 2023

(F)uridylylated Peptides Linked to VPg1 of Foot-and- Mouth Disease Virus (FMDV): Design, Synthesis and X-Ray Crystallography of the Complexes with FMDV RNA-Dependent RNA Polymerase

por de Castro, Sonia, Ferrer-Orta, Cristina, Mills, Alberto, Fernández-Cureses, Gloria, Gago, Federico, Verdaguer, Nuria, Camarasa, María-José
Publicado 2019

Inhibition of XPO-1 Mediated Nuclear Export through the Michael-Acceptor Character of Chalcones

por Gargantilla, Marta, López-Fernández, José, Camarasa, Maria-Jose, Persoons, Leentje, Daelemans, Dirk, Priego, Eva-Maria, Pérez-Pérez, María-Jesús
Publicado 2021

Design and Synthesis of New 6-Nitro and 6-Amino-3,3a,4,5-Tetrahydro-2H-Benzo[g]indazole Derivatives: Antiproliferative and Antibacterial Activity

por Cuartas, Viviana, Crespo, María del Pilar, Priego, Eva-María, Persoons, Leentje, Daelemans, Dirk, Camarasa, María-José, Insuasty, Braulio, Pérez-Pérez, María-Jesús
Publicado 2019

Modifications in the branched arms of a class of dual inhibitors of HIV and EV71 replication expand their antiviral spectrum

por Martínez-Gualda, Belén, Sun, Liang, Martí-Marí, Olaia, Mirabelli, Carmen, Delang, Leen, Neyts, Johan, Schols, Dominique, Camarasa, María-José, San-Félix, Ana
Publicado 2019

Efficient Dimerization Disruption of Leishmania infantum Trypanothione Reductase by Triazole-phenyl-thiazoles

por Revuelto, Alejandro, de Lucio, Héctor, García-Soriano, Juan Carlos, Sánchez-Murcia, Pedro A., Gago, Federico, Jiménez-Ruiz, Antonio, Camarasa, María-José, Velázquez, Sonsoles
Publicado 2021

Interrogation of Essentiality in the Reconstructed Haemophilus influenzae Metabolic Network Identifies Lipid Metabolism Antimicrobial Targets: Preclinical Evaluation of a FabH β-Ke...

por López-López, Nahikari, León, David San, de Castro, Sonia, Díez-Martínez, Roberto, Iglesias-Bexiga, Manuel, Camarasa, María José, Menéndez, Margarita, Nogales, Juan, Garmendia, Junkal
Publicado 2022

A Novel Class of Cationic and Non-Peptidic Small Molecules as Hits for the Development of Antimicrobial Agents

por Jiménez, Aranza, García, Pablo, de la Puente, Sofia, Madrona, Andrés, Camarasa, María José, Pérez-Pérez, María-Jesús, Quintela, José-Carlos, García-del Portillo, Francisco, San-Félix, Ana
Publicado 2018

Small Molecule–Peptide Conjugates as Dimerization Inhibitors of Leishmania infantum Trypanothione Disulfide Reductase

por Revuelto, Alejandro, López-Martín, Isabel, de Lucio, Héctor, García-Soriano, Juan Carlos, Zanda, Nicola, de Castro, Sonia, Gago, Federico, Jiménez-Ruiz, Antonio, Velázquez, Sonsoles, Camarasa, María-José
Publicado 2021

Multivalent Tryptophan‐ and Tyrosine‐Containing [60]Fullerene Hexa‐Adducts as Dual HIV and Enterovirus A71 Entry Inhibitors

por Ruiz‐Santaquiteria, Marta, Illescas, Beatriz M., Abdelnabi, Rana, Boonen, Arnaud, Mills, Alberto, Martí‐Marí, Olaia, Noppen, Sam, Neyts, Johan, Schols, Dominique, Gago, Federico, San‐Félix, Ana, Camarasa, María‐José, Martín, Nazario
Publicado 2021

A Versatile Class of 1,4,4-Trisubstituted Piperidines Block Coronavirus Replication In Vitro

por De Castro, Sonia, Stevaert, Annelies, Maldonado, Miguel, Delpal, Adrien, Vandeput, Julie, Van Loy, Benjamin, Eydoux, Cecilia, Guillemot, Jean-Claude, Decroly, Etienne, Gago, Federico, Canard, Bruno, Camarasa, Maria-Jose, Velázquez, Sonsoles, Naesens, Lieve
Publicado 2022

Leishmania infantum EndoG Is an Endo/Exo-Nuclease Essential for Parasite Survival

por Rico, Eva, Oliva, Cristina, Gutierrez, Kilian Jesús, Alzate, Juan Fernando, Genes, Carlos Mario, Moreno, David, Casanova, Elena, Gigante, Alba, Pérez-Pérez, María-Jesús, Camarasa, María-José, Clos, Joachim, Gago, Federico, Jiménez-Ruiz, Antonio
Publicado 2014

Double Arylation of the Indole Side Chain of Tri- and Tetrapodal Tryptophan Derivatives Renders Highly Potent HIV-1 and EV-A71 Entry Inhibitors†

por Martí-Marí, Olaia, Martínez-Gualda, Belén, de la Puente-Secades, Sofía, Mills, Alberto, Quesada, Ernesto, Abdelnabi, Rana, Sun, Liang, Boonen, Arnaud, Noppen, Sam, Neyts, Johan, Schols, Dominique, Camarasa, María-José, Gago, Federico, San-Félix, Ana
Publicado 2021

High-affinity ligands of the colchicine domain in tubulin based on a structure-guided design

por Bueno, Oskía, Estévez Gallego, Juan, Martins, Solange, Prota, Andrea E., Gago, Federico, Gómez-SanJuan, Asier, Camarasa, María-José, Barasoain, Isabel, Steinmetz, Michel O., Díaz, J. Fernando, Pérez-Pérez, María-Jesús, Liekens, Sandra, Priego, Eva-María
Publicado 2018

Antivascular and antitumor properties of the tubulin-binding chalcone TUB091

por Canela, María-Dolores, Noppen, Sam, Bueno, Oskía, Prota, Andrea E., Bargsten, Katja, Sáez-Calvo, Gonzalo, Jimeno, María-Luisa, Benkheil, Mohammed, Ribatti, Domenico, Velázquez, Sonsoles, Camarasa, María-José, Fernando Díaz, J., Steinmetz, Michel O., Priego, Eva-María, Pérez-Pérez, María-Jesús, Liekens, Sandra
Publicado 2016