Special Issue “Adenosine Receptors as Attractive Targets in Human Diseases”

por Catarzi, Daniela, Varano, Flavia, Colotta, Vittoria
Publicado 2021

Piperazine- and Piperidine-Containing Thiazolo[5,4-d]pyrimidine Derivatives as New Potent and Selective Adenosine A(2A) Receptor Inverse Agonists

por Varano, Flavia, Catarzi, Daniela, Vigiani, Erica, Vincenzi, Fabrizio, Pasquini, Silvia, Varani, Katia, Colotta, Vittoria
Publicado 2020

Amino-3,5-Dicyanopyridines Targeting the Adenosine Receptors. Ranging from Pan Ligands to Combined A1/A2B Partial Agonists

por Catarzi, Daniela, Varano, Flavia, Varani, Katia, Vincenzi, Fabrizio, Pasquini, Silvia, Dal Ben, Diego, Volpini, Rosaria, Colotta, Vittoria
Publicado 2019

Inhibition of A(2A) Adenosine Receptor Signaling in Cancer Cells Proliferation by the Novel Antagonist TP455

por Gessi, Stefania, Bencivenni, Serena, Battistello, Enrica, Vincenzi, Fabrizio, Colotta, Vittoria, Catarzi, Daniela, Varano, Flavia, Merighi, Stefania, Borea, Pier Andrea, Varani, Katia
Publicado 2017

Pharmacological Characterization of P626, a Novel Dual Adenosine A(2A)/A(2B) Receptor Antagonist, on Synaptic Plasticity and during an Ischemic-like Insult in CA1 Rat Hippocampus

por Venturini, Martina, Cherchi, Federica, Santalmasi, Clara, Frulloni, Lucia, Dettori, Ilaria, Catarzi, Daniela, Pedata, Felicita, Colotta, Vittoria, Varano, Flavia, Coppi, Elisabetta, Pugliese, Anna Maria
Publicado 2023

Design and Synthesis of Novel Thiazolo[5,4-d]pyrimidine Derivatives with High Affinity for Both the Adenosine A(1) and A(2A) Receptors, and Efficacy in Animal Models of Depression

por Varano, Flavia, Catarzi, Daniela, Vigiani, Erica, Dal Ben, Diego, Buccioni, Michela, Marucci, Gabriella, Di Cesare Mannelli, Lorenzo, Lucarini, Elena, Ghelardini, Carla, Volpini, Rosaria, Colotta, Vittoria
Publicado 2021

The role of 5-arylalkylamino- and 5-piperazino- moieties on the 7-aminopyrazolo[4,3-d]pyrimidine core in affecting adenosine A(1) and A(2A) receptor affinity and selectivity profil...

por Squarcialupi, Lucia, Betti, Marco, Catarzi, Daniela, Varano, Flavia, Falsini, Matteo, Ravani, Annalisa, Pasquini, Silvia, Vincenzi, Fabrizio, Salmaso, Veronica, Sturlese, Mattia, Varani, Katia, Moro, Stefano, Colotta, Vittoria
Publicado 2017

4-Heteroaryl Substituted Amino-3,5-Dicyanopyridines as New Adenosine Receptor Ligands: Novel Insights on Structure-Activity Relationships and Perspectives

por Catarzi, Daniela, Varano, Flavia, Vigiani, Erica, Calenda, Sara, Melani, Fabrizio, Varani, Katia, Vincenzi, Fabrizio, Pasquini, Silvia, Mennini, Natascia, Nerli, Giulia, Dal Ben, Diego, Volpini, Rosaria, Colotta, Vittoria
Publicado 2022

“Dual Anta-Inhibitors” of the A(2A) Adenosine Receptor and Casein Kinase CK1delta: Synthesis, Biological Evaluation, and Molecular Modeling Studies

por Spinaci, Andrea, Buccioni, Michela, Catarzi, Daniela, Cui, Chang, Colotta, Vittoria, Dal Ben, Diego, Cescon, Eleonora, Francucci, Beatrice, Grieco, Ilenia, Lambertucci, Catia, Marucci, Gabriella, Bassani, Davide, Pavan, Matteo, Varano, Flavia, Federico, Stephanie, Spalluto, Giampiero, Moro, Stefano, Volpini, Rosaria
Publicado 2023