The Parallel Structure–Activity Relationship Screening of Three Compounds Identifies the Common Agonist Pharmacophore of Pyrrolidine Bis-Cyclic Guanidine Melanocortin-3 Receptor (M...

por Ericson, Mark D., Freeman, Katie T., LaVoi, Travis M., Donow, Haley M., Santos, Radleigh G., Giulianotti, Marc A., Pinilla, Clemencia, Houghten, Richard A., Haskell-Luevano, Carrie
Publicado 2023

Identification of SARS-CoV-2 Spike Palmitoylation Inhibitors That Results in Release of Attenuated Virus with Reduced Infectivity

por Ramadan, Ahmed A., Mayilsamy, Karthick, McGill, Andrew R., Ghosh, Anandita, Giulianotti, Marc A., Donow, Haley M., Mohapatra, Shyam S., Mohapatra, Subhra, Chandran, Bala, Deschenes, Robert J., Roy, Arunava
Publicado 2022

Inhibition of Aminoglycoside 6′-N-acetyltransferase Type Ib (AAC(6′)-Ib): Structure–Activity Relationship of Substituted Pyrrolidine Pentamine Derivatives as Inhibitors

por Rocha, Kenneth, Magallon, Jesus, Reeves, Craig, Phan, Kimberly, Vu, Peter, Oakley-Havens, Crista L., Kwan, Stella, Ramirez, Maria Soledad, LaVoi, Travis, Donow, Haley, Chapagain, Prem, Santos, Radleigh, Pinilla, Clemencia, Giulianotti, Marc A., Tolmasky, Marcelo E.
Publicado 2021