Rapid and Efficient Access to Novel Bio-Inspired 3-Dimensional Tricyclic SpiroLactams as Privileged Structures via Meyers’ Lactamization

por Tangara, Salia, Faïon, Léo, Piveteau, Catherine, Capet, Frédéric, Godelier, Romain, Michel, Marion, Flipo, Marion, Deprez, Benoit, Willand, Nicolas, Villemagne, Baptiste
Publicado 2023

On the Hunt for Next-Generation Antimicrobial Agents: An Online Symposium Organized Jointly by the French Society for Medicinal Chemistry (Société de Chimie Thérapeutique) and the...

por Antraygues, Kevin, Compagne, Nina, Ruggieri, Francesca, Djaout, Kamel, Edoo, Zainab, Eveque, Maxime, Faïon, Léo, Gioia, Bruna, Tangara, Salia, Vieira Da Cruz, Anais, Villemagne, Baptiste, Flipo, Marion, Baulard, Alain, Willand, Nicolas
Publicado 2022

Exploring the Antitubercular Activity of Anthranilic Acid Derivatives: From MabA (FabG1) Inhibition to Intrabacterial Acidification

por Faïon, Léo, Djaout, Kamel, Pintiala, Catalin, Piveteau, Catherine, Leroux, Florence, Biela, Alexandre, Slupek, Stéphanie, Antoine, Rudy, Záhorszká, Monika, Cantrelle, Francois-Xavier, Hanoulle, Xavier, Korduláková, Jana, Deprez, Benoit, Willand, Nicolas, Baulard, Alain R., Flipo, Marion
Publicado 2023

Tricyclic SpiroLactams Kill Mycobacteria In Vitro and In Vivo by Inhibiting Type II NADH Dehydrogenases

por Dam, Sushovan, Tangara, Salia, Hamela, Claire, Hattabi, Theo, Faïon, Léo, Carre, Paul, Antoine, Rudy, Herledan, Adrien, Leroux, Florence, Piveteau, Catherine, Eveque, Maxime, Flipo, Marion, Deprez, Benoit, Kremer, Laurent, Willand, Nicolas, Villemagne, Baptiste, Hartkoorn, Ruben C.
Publicado 2022