Discovery of a new class of orthosteric antagonists with nanomolar potency at extrasynaptic GABA(A) receptors

por Falk-Petersen, Christina Birkedahl, Tsonkov, Tsonko M., Nielsen, Malene Sofie, Harpsøe, Kasper, Bundgaard, Christoffer, Frølund, Bente, Kristiansen, Uffe, Gloriam, David E., Wellendorph, Petrine
Publicado 2020

Molecular Determinants and Pharmacological Analysis for a Class of Competitive Non-transported Bicyclic Inhibitors of the Betaine/GABA Transporter BGT1

por Kickinger, Stefanie, Lie, Maria E. K., Suemasa, Akihiro, Al-Khawaja, Anas, Fujiwara, Koichi, Watanabe, Mizuki, Wilhelmsen, Kristine S., Falk-Petersen, Christina B., Frølund, Bente, Shuto, Satoshi, Ecker, Gerhard F., Wellendorph, Petrine
Publicado 2021

Synthesis and Pharmacological Evaluation of [(11)C]4-Methoxy-N-[2-(thiophen-2-yl)imidazo[1,2-a]pyridin-3-yl]benzamide as a Brain Penetrant PET Ligand Selective for the δ-Subunit-Co...

por L’Estrade, Elina T., Hansen, Hanne D., Falk-Petersen, Christina, Haugaard, Anne, Griem-Krey, Nane, Jung, Sascha, Lüddens, Hartmut, Schirmeister, Tanja, Erlandsson, Maria, Ohlsson, Tomas, Knudsen, Gitte M., Herth, Matthias M., Wellendorph, Petrine, Frølund, Bente
Publicado 2019