Anticancer Inhibitors

por Ammazzalorso, Alessandra, Fantacuzzi, Marialuigia
Publicado 2022

PPAR Ligands Induce Antiviral Effects Targeting Perturbed Lipid Metabolism during SARS-CoV-2, HCV, and HCMV Infection

por Fantacuzzi, Marialuigia, Amoroso, Rosa, Ammazzalorso, Alessandra
Publicado 2022

Anticancer Activity of Natural Products and Related Compounds

por De Filippis, Barbara, Fantacuzzi, Marialuigia, Ammazzalorso, Alessandra
Publicado 2023

Development of CDK4/6 Inhibitors: A Five Years Update

por Ammazzalorso, Alessandra, Agamennone, Mariangela, De Filippis, Barbara, Fantacuzzi, Marialuigia
Publicado 2021

HDAC Inhibitors for the Therapy of Triple Negative Breast Cancer

por Maccallini, Cristina, Ammazzalorso, Alessandra, De Filippis, Barbara, Fantacuzzi, Marialuigia, Giampietro, Letizia, Amoroso, Rosa
Publicado 2022

Antiviral Peptides as Anti-Influenza Agents

por Agamennone, Mariangela, Fantacuzzi, Marialuigia, Vivenzio, Giovanni, Scala, Maria Carmina, Campiglia, Pietro, Superti, Fabiana, Sala, Marina
Publicado 2022

A Novel Prodrug of a nNOS Inhibitor with Improved Pharmacokinetic Potential

por Maccallini, Cristina, Marinelli, Lisa, Indorf, Patrick, Cacciatore, Ivana, Fantacuzzi, Marialuigia, Clement, Bernd, Di Stefano, Antonio, Amoroso, Rosa
Publicado 2020

Coumarin-Based Dual Inhibitors of Human Carbonic Anhydrases and Monoamine Oxidases Featuring Amino Acyl and (Pseudo)-Dipeptidyl Appendages: In Vitro and Computational Studies

por Agamennone, Mariangela, Fantacuzzi, Marialuigia, Carradori, Simone, Petzer, Anél, Petzer, Jacobus P., Angeli, Andrea, Supuran, Claudiu T., Luisi, Grazia
Publicado 2022

The Selective Acetamidine-Based iNOS Inhibitor CM544 Reduces Glioma Cell Proliferation by Enhancing PARP-1 Cleavage In Vitro

por Gallorini, Marialucia, Maccallini, Cristina, Ammazzalorso, Alessandra, Amoia, Pasquale, De Filippis, Barbara, Fantacuzzi, Marialuigia, Giampietro, Letizia, Cataldi, Amelia, Amoroso, Rosa
Publicado 2019

Fibrate-based N-acylsulphonamides targeting carbonic anhydrases: synthesis, biochemical evaluation, and docking studies

por Ammazzalorso, Alessandra, Carradori, Simone, Angeli, Andrea, Akdemir, Atilla, De Filippis, Barbara, Fantacuzzi, Marialuigia, Giampietro, Letizia, Maccallini, Cristina, Amoroso, Rosa, Supuran, Claudiu T.
Publicado 2019

New azolyl-derivatives as multitargeting agents against breast cancer and fungal infections: synthesis, biological evaluation and docking study

por Maccallini, Cristina, Gallorini, Marialucia, Sisto, Francesca, Akdemir, Atilla, Ammazzalorso, Alessandra, De Filippis, Barbara, Fantacuzzi, Marialuigia, Giampietro, Letizia, Carradori, Simone, Cataldi, Amelia, Amoroso, Rosa
Publicado 2021

Benzenesulfonamide derivatives as Vibrio cholerae carbonic anhydrases inhibitors: a computational-aided insight in the structural rigidity-activity relationships

por Fantacuzzi, Marialuigia, D’Agostino, Ilaria, Carradori, Simone, Liguori, Francesco, Carta, Fabrizio, Agamennone, Mariangela, Angeli, Andrea, Sannio, Filomena, Docquier, Jean-Denis, Capasso, Clemente, Supuran, Claudiu T.
Publicado 2023

Resveratrol Analogues as Dual Inhibitors of Monoamine Oxidase B and Carbonic Anhydrase VII: A New Multi-Target Combination for Neurodegenerative Diseases?

por Carradori, Simone, Fantacuzzi, Marialuigia, Ammazzalorso, Alessandra, Angeli, Andrea, De Filippis, Barbara, Galati, Salvatore, Petzer, Anél, Petzer, Jacobus P., Poli, Giulio, Tuccinardi, Tiziano, Agamennone, Mariangela, Supuran, Claudiu T.
Publicado 2022

Design, Synthesis and Biological Evaluation of Aromatase Inhibitors Based on Sulfonates and Sulfonamides of Resveratrol

por Fantacuzzi, Marialuigia, Gallorini, Marialucia, Gambacorta, Nicola, Ammazzalorso, Alessandra, Aturki, Zeineb, Balaha, Marwa, Carradori, Simone, Giampietro, Letizia, Maccallini, Cristina, Cataldi, Amelia, Nicolotti, Orazio, Amoroso, Rosa, De Filippis, Barbara
Publicado 2021

Benzothiazole Derivatives Endowed with Antiproliferative Activity in Paraganglioma and Pancreatic Cancer Cells: Structure–Activity Relationship Studies and Target Prediction Analys...

por Amoroso, Rosa, De Lellis, Laura, Florio, Rosalba, Moreno, Nazaret, Agamennone, Mariangela, De Filippis, Barbara, Giampietro, Letizia, Maccallini, Cristina, Fernández, Inmaculada, Recio, Rocío, Cama, Alessandro, Fantacuzzi, Marialuigia, Ammazzalorso, Alessandra
Publicado 2022

Sulfonimide and Amide Derivatives as Novel PPARα Antagonists: Synthesis, Antiproliferative Activity, and Docking Studies

por Ammazzalorso, Alessandra, Bruno, Isabella, Florio, Rosalba, De Lellis, Laura, Laghezza, Antonio, Cerchia, Carmen, De Filippis, Barbara, Fantacuzzi, Marialuigia, Giampietro, Letizia, Maccallini, Cristina, Tortorella, Paolo, Veschi, Serena, Loiodice, Fulvio, Lavecchia, Antonio, Cama, Alessandro, Amoroso, Rosa
Publicado 2020