Enantioselective Synthesis of 3,4-Dihydro-1,2-oxazepin-5(2H)-ones and 2,3-Dihydropyridin-4(1H)-ones from β-Substituted β-Hydroxyaminoaldehydes

por Ranade, Adwait R., Georg, Gunda I.
Publicado 2014

Boron–Heck Reaction of Cyclic Enaminones: Regioselective Direct Arylation via Oxidative Palladium(II) Catalysis

por Kim, Yong Wook, Georg, Gunda I.
Publicado 2014

Synthesis and Cytotoxicity Evaluation of C4‐ and C5‐Modified Analogues of the α,β‐Unsaturated Lactone of Pironetin

por Huang, David S., Wong, Henry L., Georg, Gunda I.
Publicado 2017

Synthesis and Spectral Properties of 8-Anilinonaphthalene-1-sulfonic Acid (ANS) Derivatives Prepared by Microwave-Assisted Copper(0)-Catalyzed Ullmann Reaction

por Wang, Nan, Faber, Erik B., Georg, Gunda I.
Publicado 2019

A special issue on contraceptive development: past, present, and future

por Matzuk, Martin M, Georg, Gunda I, Yan, Wei
Publicado 2020

Review of rationale and progress toward targeting cyclin-dependent kinase 2 (CDK2) for male contraception(†)

por Faber, Erik B, Wang, Nan, Georg, Gunda I
Publicado 2020

Absolute Quantitative (1)H NMR Spectroscopy for Compound Purity Determination

por Cushman, Mark, Georg, Gunda I., Holzgrabe, Ulrike, Wang, Shaomeng
Publicado 2014

Steroidal Antagonists of Progesterone- and Prostaglandin E(1)-Induced Activation of the Cation Channel of Sperm

por Carlson, Erick J., Georg, Gunda I., Hawkinson, Jon E.
Publicado 2022

Enantiospecific Synthesis and Cytotoxicity Evaluation of Oximidine II Analogues

por Schneider, Christopher M., Li, Wei, Khownium, Kriangsak, Lushington, Gerald H., Georg, Gunda I.
Publicado 2016

Synthesis of Arylazide‐ and Diazirine‐Containing CrAsH‐EDT(2) Photoaffinity Probes

por Syeda, Shameem S., Rice, Daren, Hook, Derek J., Heckert, Leslie L., Georg, Gunda I.
Publicado 2016

Design, Synthesis, and in Vitro and in Vivo Evaluation of Ouabain Analogues as Potent and Selective Na,K-ATPase α4 Isoform Inhibitors for Male Contraception

por Syeda, Shameem Sultana, Sánchez, Gladis, Hong, Kwon Ho, Hawkinson, Jon E., Georg, Gunda I., Blanco, Gustavo
Publicado 2018

Retinoic acid receptor antagonists for male contraception: current status(†)

por Noman, Md Abdullah Al, Kyzer, Jillian L, Chung, Sanny S W, Wolgemuth, Debra J, Georg, Gunda I
Publicado 2020

The Na(+) and K(+) transport system of sperm (ATP1A4) is essential for male fertility and an attractive target for male contraception

por Syeda, Shameem Sultana, Sánchez, Gladis, McDermott, Jeffrey P, Hong, Kwon Ho, Blanco, Gustavo, Georg, Gunda I
Publicado 2020

Reformulating Tylocrebrine in Epidermal Growth Factor Receptor Targeted Polymeric Nanoparticles Improves Its Therapeutic Index

por Kirtane, Ameya R., Wong, Henry L., Guru, Bharath Raja, Lis, Lev G., Georg, Gunda I., Gurvich, Vadim J., Panyam, Jayanth
Publicado 2015

The Ecstasy and Agony of Assay Interference Compounds

por Aldrich, Courtney, Bertozzi, Carolyn, Georg, Gunda I., Kiessling, Laura, Lindsley, Craig, Liotta, Dennis, Merz, Kenneth M., Schepartz, Alanna, Wang, Shaomeng
Publicado 2017

Stability of the Human Hsp90-p50(Cdc37) Chaperone Complex against Nucleotides and Hsp90 Inhibitors, and the Influence of Phosphorylation by Casein Kinase 2

por Olesen, Sanne H., Ingles, Donna J., Zhu, Jin-Yi, Martin, Mathew P., Betzi, Stephane, Georg, Gunda I., Tash, Joseph S., Schönbrunn, Ernst
Publicado 2015

Acetyl-lysine Binding Site of Bromodomain-Containing Protein 4 (BRD4) Interacts with Diverse Kinase Inhibitors

por Ember, Stuart W. J., Zhu, Jin-Yi, Olesen, Sanne H., Martin, Mathew P., Becker, Andreas, Berndt, Norbert, Georg, Gunda I., Schönbrunn, Ernst
Publicado 2014

N-Butyldeoxygalactonojirimycin Induces Reversible Infertility in Male CD Rats

por Gupta, Vijayalaxmi, Hild, Sheri A., Jakkaraj, Sudhakar R., Carlson, Erick J., Wong, Henry L., Allen, C. Leigh, Georg, Gunda I., Tash, Joseph S.
Publicado 2019

Development of WEE2 kinase inhibitors as novel non-hormonal female contraceptives that target meiosis

por Hanna, Carol B, Mudaliar, Deepti, John, Kristen, Allen, C Leigh, Sun, Luxin, Hawkinson, Jon E, Schönbrunn, Ernst, Georg, Gunda I, Jensen, Jeffrey T
Publicado 2020

Structure–Activity Studies of N‐Butyl‐1‐deoxynojirimycin (NB‐DNJ) Analogues: Discovery of Potent and Selective Aminocyclopentitol Inhibitors of GBA1 and GBA2

por Gu, Xingxian, Gupta, Vijayalaxmi, Yang, Yan, Zhu, Jin‐Yi, Carlson, Erick J., Kingsley, Carolyn, Tash, Joseph S., Schönbrunn, Ernst, Hawkinson, Jon, Georg, Gunda I.
Publicado 2017