Natural Products as Cathepsin Inhibitors

por Vidal-Albalat, Andreu, González, Florenci V.
Publicado 2016

Three-Step Telescoped Synthesis of Monosubstituted Vicinal Diamines from Aldehydes

por Bou-Iserte, Lledó, Latorre, Antonio, Rodríguez, Santiago, González, Florenci V.
Publicado 2019

Formal [3+2] Cycloaddition Reactions of Electron-Rich Aryl Epoxides with Alkenes under Lewis Acid Catalysis Affording Tetrasubstituted Tetrahydrofurans

por Macías-Villamizar, Víctor E., Cuca-Suárez, Luís, Rodríguez, Santiago, González, Florenci V.
Publicado 2020

Impact of the Recognition Part of Dipeptidyl Nitroalkene Compounds on the Inhibition Mechanism of Cysteine Proteases Cruzain and Cathepsin L

por Arafet, Kemel, Royo, Santiago, Schirmeister, Tanja, Barthels, Fabian, González, Florenci V., Moliner, Vicent
Publicado 2023

Mechanism of inhibition of SARS-CoV-2 M(pro) by N3 peptidyl Michael acceptor explained by QM/MM simulations and design of new derivatives with tunable chemical reactivity

por Arafet, Kemel, Serrano-Aparicio, Natalia, Lodola, Alessio, Mulholland, Adrian J., González, Florenci V., Świderek, Katarzyna, Moliner, Vicent
Publicado 2020

Impact of the Warhead of Dipeptidyl Keto Michael Acceptors on the Inhibition Mechanism of Cysteine Protease Cathepsin L

por Fernández-de-la-Pradilla, Adrián, Royo, Santiago, Schirmeister, Tanja, Barthels, Fabian, Świderek, Katarzyna, González, Florenci V., Moliner, Vicent
Publicado 2023

Advances in the Development of SARS-CoV-2 Mpro Inhibitors

por Agost-Beltrán, Laura, de la Hoz-Rodríguez, Sergio, Bou-Iserte, Lledó, Rodríguez, Santiago, Fernández-de-la-Pradilla, Adrián, González, Florenci V.
Publicado 2022

Investigation of the Compatibility between Warheads and Peptidomimetic Sequences of Protease Inhibitors—A Comprehensive Reactivity and Selectivity Study

por Müller, Patrick, Meta, Mergim, Meidner, Jan Laurenz, Schwickert, Marvin, Meyr, Jessica, Schwickert, Kevin, Kersten, Christian, Zimmer, Collin, Hammerschmidt, Stefan Josef, Frey, Ariane, Lahu, Albin, de la Hoz-Rodríguez, Sergio, Agost-Beltrán, Laura, Rodríguez, Santiago, Diemer, Kira, Neumann, Wilhelm, Gonzàlez, Florenci V., Engels, Bernd, Schirmeister, Tanja
Publicado 2023

Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes–7

por Gütschow, Michael, Vanden Eynde, Jean Jacques, Jampilek, Josef, Kang, CongBao, Mangoni, Arduino A., Fossa, Paola, Karaman, Rafik, Trabocchi, Andrea, Scott, Peter J. H., Reynisson, Jóhannes, Rapposelli, Simona, Galdiero, Stefania, Winum, Jean-Yves, Brullo, Chiara, Prokai-Tatrai, Katalin, Sharma, Arun K., Schapira, Matthieu, Azuma, Yasu-Taka, Cerchia, Laura, Spetea, Mariana, Torri, Giangiacomo, Collina, Simona, Geronikaki, Athina, García-Sosa, Alfonso T., Vasconcelos, M. Helena, Sousa, Maria Emília, Kosalec, Ivan, Tuccinardi, Tiziano, Duarte, Iola F., Salvador, Jorge A. R., Bertinaria, Massimo, Pellecchia, Maurizio, Amato, Jussara, Rastelli, Giulio, Gomes, Paula A. C., Guedes, Rita C., Sabatier, Jean-Marc, Estévez-Braun, Ana, Pagano, Bruno, Mangani, Stefano, Ragno, Rino, Kokotos, George, Brindisi, Margherita, González, Florenci V., Borges, Fernanda, Miloso, Mariarosaria, Rautio, Jarkko, Muñoz-Torrero, Diego
Publicado 2020