Small Molecule Inhibitors of CXCR4

por Debnath, Bikash, Xu, Shili, Grande, Fedora, Garofalo, Antonio, Neamati, Nouri
Publicado 2013

A New Generation of Dihydropyridine Calcium Channel Blockers: Photostabilization of Liquid Formulations Using Nonionic Surfactants

por Ioele, Giuseppina, Gündüz, Miyase Gözde, Spatari, Claudia, De Luca, Michele, Grande, Fedora, Ragno, Gaetano
Publicado 2019

Photodegradation of Anti-Inflammatory Drugs: Stability Tests and Lipid Nanocarriers for Their Photoprotection

por Ioele, Giuseppina, Grande, Fedora, De Luca, Michele, Occhiuzzi, Maria Antonietta, Garofalo, Antonio, Ragno, Gaetano
Publicado 2021

Promising Perspectives of the Antiproliferative GPER Inverse Agonist ERα17p in Breast Cancer

por Kampa, Marilena, Lappano, Rosamaria, Grande, Fedora, Rizzuti, Bruno, Maggiolini, Marcello, Castanas, Elias, Jacquot, Yves
Publicado 2023

Lavandula angustifolia mill. (Lamiaceae) ethanol extract and its main constituents as promising agents for the treatment of metabolic disorders: chemical profile, in vitro biologic...

por Tundis, Rosa, Grande, Fedora, Occhiuzzi, Maria A., Sicari, Vincenzo, Loizzo, Monica R., Cappello, Anna R.
Publicado 2023

Multivariate Curve Resolution Methodology Applied to the ATR-FTIR Data for Adulteration Assessment of Virgin Coconut Oil

por De Luca, Michele, Ioele, Giuseppina, Grande, Fedora, Occhiuzzi, Maria Antonietta, Chieffallo, Martina, Garofalo, Antonio, Ragno, Gaetano
Publicado 2023

Polyphenols from Citrus Tacle(®) Extract Endowed with HMGCR Inhibitory Activity: An Antihypercholesterolemia Natural Remedy

por Grande, Fedora, Occhiuzzi, Maria Antonietta, Perri, Maria Rosaria, Ioele, Giuseppina, Rizzuti, Bruno, Statti, Giancarlo, Garofalo, Antonio
Publicado 2021

Interaction of letrozole and its degradation products with aromatase: chemometric assessment of kinetics and structure-based binding validation

por De Luca, Michele, Occhiuzzi, Maria Antonietta, Rizzuti, Bruno, Ioele, Giuseppina, Ragno, Gaetano, Garofalo, Antonio, Grande, Fedora
Publicado 2022

Anticancer Drugs: Recent Strategies to Improve Stability Profile, Pharmacokinetic and Pharmacodynamic Properties

por Ioele, Giuseppina, Chieffallo, Martina, Occhiuzzi, Maria Antonietta, De Luca, Michele, Garofalo, Antonio, Ragno, Gaetano, Grande, Fedora
Publicado 2022

Reverse Transcriptase Inhibitors Nanosystems Designed for Drug Stability and Controlled Delivery

por Grande, Fedora, Ioele, Giuseppina, Occhiuzzi, Maria Antonietta, De Luca, Michele, Mazzotta, Elisabetta, Ragno, Gaetano, Garofalo, Antonio, Muzzalupo, Rita
Publicado 2019

Gel Formulation of Nabumetone and a Newly Synthesized Analog: Microemulsion as a Photoprotective Topical Delivery System

por Grande, Fedora, Ragno, Gaetano, Muzzalupo, Rita, Occhiuzzi, Maria Antonietta, Mazzotta, Elisabetta, De Luca, Michele, Garofalo, Antonio, Ioele, Giuseppina
Publicado 2020

Identification by Molecular Docking of Homoisoflavones from Leopoldia comosa as Ligands of Estrogen Receptors

por Grande, Fedora, Rizzuti, Bruno, Occhiuzzi, Maria A., Ioele, Giuseppina, Casacchia, Teresa, Gelmini, Fabrizio, Guzzi, Rita, Garofalo, Antonio, Statti, Giancarlo
Publicado 2018

Computational Approaches for the Discovery of GPER Targeting Compounds

por Grande, Fedora, Occhiuzzi, Maria A., Lappano, Rosamaria, Cirillo, Francesca, Guzzi, Rita, Garofalo, Antonio, Jacquot, Yves, Maggiolini, Marcello, Rizzuti, Bruno
Publicado 2020

Chloro-1,4-dimethyl-9H-carbazole Derivatives Displaying Anti-HIV Activity

por Saturnino, Carmela, Grande, Fedora, Aquaro, Stefano, Caruso, Anna, Iacopetta, Domenico, Bonomo, Maria Grazia, Longo, Pasquale, Schols, Dominique, Sinicropi, Maria Stefania
Publicado 2018

CCR5/CXCR4 Dual Antagonism for the Improvement of HIV Infection Therapy

por Grande, Fedora, Occhiuzzi, Maria Antonietta, Rizzuti, Bruno, Ioele, Giuseppina, De Luca, Michele, Tucci, Paola, Svicher, Valentina, Aquaro, Stefano, Garofalo, Antonio
Publicado 2019

Ligand-activated PPARγ downregulates CXCR4 gene expression through a novel identified PPAR response element and inhibits breast cancer progression

por Rovito, Daniela, Gionfriddo, Giulia, Barone, Ines, Giordano, Cinzia, Grande, Fedora, De Amicis, Francesca, Lanzino, Marilena, Catalano, Stefania, Andò, Sebastiano, Bonofiglio, Daniela
Publicado 2016

Use of Pluronic Surfactants in Gel Formulations of Photosensitive 1,4-Dihydropyridine Derivatives: A Potential Approach in the Treatment of Neuropathic Pain

por Ioele, Giuseppina, Muzzalupo, Rita, Gündüz, Miyase Gözde, De Luca, Michele, Mazzotta, Elisabetta, Grande, Fedora, Occhiuzzi, Maria Antonietta, Garofalo, Antonio, Ragno, Gaetano
Publicado 2021

Sub-Micromolar Inhibition of SARS-CoV-2 3CLpro by Natural Compounds

por Rizzuti, Bruno, Ceballos-Laita, Laura, Ortega-Alarcon, David, Jimenez-Alesanco, Ana, Vega, Sonia, Grande, Fedora, Conforti, Filomena, Abian, Olga, Velazquez-Campoy, Adrian
Publicado 2021

The Peptide ERα17p Is a GPER Inverse Agonist that Exerts Antiproliferative Effects in Breast Cancer Cells

por Lappano, Rosamaria, Mallet, Christophe, Rizzuti, Bruno, Grande, Fedora, Galli, Giulia Raffaella, Byrne, Cillian, Broutin, Isabelle, Boudieu, Ludivine, Eschalier, Alain, Jacquot, Yves, Maggiolini, Marcello
Publicado 2019

Toward Multitasking Pharmacological COX-Targeting Agents: Non-Steroidal Anti-Inflammatory Prodrugs with Antiproliferative Effects

por Grande, Fedora, Giordano, Francesca, Occhiuzzi, Maria Antonietta, Rocca, Carmine, Ioele, Giuseppina, De Luca, Michele, Ragno, Gaetano, Panno, Maria Luisa, Rizzuti, Bruno, Garofalo, Antonio
Publicado 2021