Discovery of the first-in-class potent and isoform-selective human carbonic anhydrase III inhibitors

por Giovannuzzi, Simone, Bonardi, Alessandro, Gratteri, Paola, Nocentini, Alessio, Supuran, Claudiu T.
Publicado 2023

Cation, Anion and Ion-Pair Complexes with a G-3 Poly(ethylene imine) Dendrimer in Aqueous Solution

por Savastano, Matteo, Bazzicalupi, Carla, Giorgi, Claudia, Gratteri, Paola, Bianchi, Antonio
Publicado 2017

The crystal structure of human telomeric DNA complexed with berberine: an interesting case of stacked ligand to G-tetrad ratio higher than 1:1

por Bazzicalupi, Carla, Ferraroni, Marta, Bilia, Anna Rita, Scheggi, Francesca, Gratteri, Paola
Publicado 2013

Tales of the Unexpected: The Case of Zirconium(IV) Complexes with Desferrioxamine

por Savastano, Matteo, Bazzicalupi, Carla, Ferraro, Giovanni, Fratini, Emiliano, Gratteri, Paola, Bianchi, Antonio
Publicado 2019

Steroids interfere with human carbonic anhydrase activity by using alternative binding mechanisms

por Nocentini, Alessio, Bonardi, Alessandro, Gratteri, Paola, Cerra, Bruno, Gioiello, Antimo, Supuran, Claudiu T.
Publicado 2018

Pharmaceutical strategies for preventing toxicity and promoting antioxidant and anti-inflammatory actions of bilirubin

por Nocentini, Alessio, Bonardi, Alessandro, Pratesi, Simone, Gratteri, Paola, Dani, Carlo, Supuran, Claudiu T.
Publicado 2022

Sensing Zn(2+) in Aqueous Solution with a Fluorescent Scorpiand Macrocyclic Ligand Decorated with an Anthracene Bearing Tail

por Savastano, Matteo, Fiaschi, Matteo, Ferraro, Giovanni, Gratteri, Paola, Mariani, Palma, Bianchi, Antonio, Bazzicalupi, Carla
Publicado 2020

The antibiotic furagin and its derivatives are isoform-selective human carbonic anhydrase inhibitors

por Pustenko, Aleksandrs, Nocentini, Alessio, Gratteri, Paola, Bonardi, Alessandro, Vozny, Igor, Žalubovskis, Raivis, Supuran, Claudiu T.
Publicado 2020

Discovery of Novel Hydroxyimine-Tethered Benzenesulfonamides as Potential Human Carbonic Anhydrase IX/XII Inhibitors

por Peerzada, Mudasir Nabi, Vullo, Daniela, Paoletti, Niccolò, Bonardi, Alessandro, Gratteri, Paola, Supuran, Claudiu T., Azam, Amir
Publicado 2023

Inhibition Studies on Human and Mycobacterial Carbonic Anhydrases with N-((4-Sulfamoylphenyl)carbamothioyl) Amides

por Abdoli, Morteza, Bonardi, Alessandro, Paoletti, Niccolò, Aspatwar, Ashok, Parkkila, Seppo, Gratteri, Paola, Supuran, Claudiu T., Žalubovskis, Raivis
Publicado 2023

Development of Hydrogen Sulfide-Releasing Carbonic Anhydrases IX- and XII-Selective Inhibitors with Enhanced Antihyperalgesic Action in a Rat Model of Arthritis

por Bonardi, Alessandro, Micheli, Laura, Di Cesare Mannelli, Lorenzo, Ghelardini, Carla, Gratteri, Paola, Nocentini, Alessio, Supuran, Claudiu T.
Publicado 2022

Probing the Efficiency of 13-Pyridylalkyl Berberine Derivatives to Human Telomeric G-Quadruplexes Binding: Spectroscopic, Solid State and In Silico Analysis

por Bazzicalupi, Carla, Bonardi, Alessandro, Biver, Tarita, Ferraroni, Marta, Papi, Francesco, Savastano, Matteo, Lombardi, Paolo, Gratteri, Paola
Publicado 2022

Selenium-analogs based on natural sources as cancer-associated carbonic anhydrase isoforms IX and XII inhibitors

por Astrain-Redin, Nora, Paoletti, Niccolò, Plano, Daniel, Bonardi, Alessandro, Gratteri, Paola, Angeli, Andrea, Sanmartin, Carmen, Supuran, Claudiu T.
Publicado 2023

Novel insights on saccharin- and acesulfame-based carbonic anhydrase inhibitors: design, synthesis, modelling investigations and biological activity evaluation

por Guglielmi, Paolo, Rotondi, Giulia, Secci, Daniela, Angeli, Andrea, Chimenti, Paola, Nocentini, Alessio, Bonardi, Alessandro, Gratteri, Paola, Carradori, Simone, Supuran, Claudiu T.
Publicado 2020

Inhibition of α-, β- and γ-carbonic anhydrases from the pathogenic bacterium Vibrio cholerae with aromatic sulphonamides and clinically licenced drugs – a joint docking/molecular d...

por Bonardi, Alessandro, Nocentini, Alessio, Osman, Sameh Mohamed, Alasmary, Fatmah Ali, Almutairi, Tahani Mazyad, Abdullah, Dalal Saied, Gratteri, Paola, Supuran, Claudiu T.
Publicado 2021

Solid State and Solution Study on the Formation of Inorganic Anion Complexes with a Series of Tetrazine-Based Ligands

por Savastano, Matteo, García-Gallarín, Celeste, Giorgi, Claudia, Gratteri, Paola, López de la Torre, Maria Dolores, Bazzicalupi, Carla, Bianchi, Antonio, Melguizo, Manuel
Publicado 2019

Aryl-4,5-dihydro-1H-pyrazole-1-carboxamide Derivatives Bearing a Sulfonamide Moiety Show Single-digit Nanomolar-to-Subnanomolar Inhibition Constants against the Tumor-associated Hu...

por Hargunani, Priya, Tadge, Nikhil, Ceruso, Mariangela, Leitans, Janis, Kazaks, Andris, Tars, Kaspars, Gratteri, Paola, Supuran, Claudiu T., Nocentini, Alessio, Toraskar, Mrunmayee P.
Publicado 2020

Appraisal of anti-protozoan activity of nitroaromatic benzenesulfonamides inhibiting carbonic anhydrases from Trypanosoma cruzi and Leishmania donovani

por Nocentini, Alessio, Osman, Sameh M., Rodrigues, Igor A., Cardoso, Veronica S., Alasmary, Fatmah Ali S., AlOthman, Zeid, Vermelho, Alane B., Gratteri, Paola, Supuran, Claudiu T.
Publicado 2019

Inhibition of the β-carbonic anhydrase from the dandruff-producing fungus Malassezia globosa with monothiocarbamates

por Nocentini, Alessio, Vullo, Daniela, Del Prete, Sonia, Osman, Sameh M., Alasmary, Fatmah A.S., AlOthman, Zeid, Capasso, Clemente, Carta, Fabrizio, Gratteri, Paola, Supuran, Claudiu T.
Publicado 2017

β3-Adrenoreceptor Activity Limits Apigenin Efficacy in Ewing Sarcoma Cells: A Dual Approach to Prevent Cell Survival

por Pasha, Amada, Vignoli, Marina, Subbiani, Angela, Nocentini, Alessio, Selleri, Silvia, Gratteri, Paola, Dabraio, Annalisa, Casini, Tommaso, Filippi, Luca, Fotzi, Ilaria, Favre, Claudio, Calvani, Maura
Publicado 2019