Kinetic Study on the Base-Catalyzed Imine-Enamine Tautomerism of a Chiral Biologically Active Isoxazoline Derivative by HPLC on Amylose Tris(3,5-dimethylphenylcarbamate) Chiral Sta...

por Sadutto, Daniele, Guglielmi, Paolo, Carradori, Simone, Secci, Daniela, Cirilli, Roberto
Publicado 2023

The Up-Regulation of Oxidative Stress as a Potential Mechanism of Novel MAO-B Inhibitors for Glioblastoma Treatment

por Marconi, Guya Diletta, Gallorini, Marialucia, Carradori, Simone, Guglielmi, Paolo, Cataldi, Amelia, Zara, Susi
Publicado 2019

Kinesin Eg5 Targeting Inhibitors as a New Strategy for Gastric Adenocarcinoma Treatment

por Marconi, Guya Diletta, Carradori, Simone, Ricci, Alessia, Guglielmi, Paolo, Cataldi, Amelia, Zara, Susi
Publicado 2019

Design, Synthesis, Docking Studies and Monoamine Oxidase Inhibition of a Small Library of 1-acetyl- and 1-thiocarbamoyl-3,5-diphenyl-4,5-dihydro-(1H)-pyrazoles

por Guglielmi, Paolo, Carradori, Simone, Poli, Giulio, Secci, Daniela, Cirilli, Roberto, Rotondi, Giulia, Chimenti, Paola, Petzer, Anél, Petzer, Jacobus P.
Publicado 2019

Novel insights on saccharin- and acesulfame-based carbonic anhydrase inhibitors: design, synthesis, modelling investigations and biological activity evaluation

por Guglielmi, Paolo, Rotondi, Giulia, Secci, Daniela, Angeli, Andrea, Chimenti, Paola, Nocentini, Alessio, Bonardi, Alessandro, Gratteri, Paola, Carradori, Simone, Supuran, Claudiu T.
Publicado 2020

Open saccharin-based secondary sulfonamides as potent and selective inhibitors of cancer-related carbonic anhydrase IX and XII isoforms

por D’Ascenzio, Melissa, Guglielmi, Paolo, Carradori, Simone, Secci, Daniela, Florio, Rosalba, Mollica, Adriano, Ceruso, Mariangela, Akdemir, Atilla, Sobolev, Anatoly P., Supuran, Claudiu T.
Publicado 2016

Analysis of imidazoles and triazoles in biological samples after MicroExtraction by packed sorbent

por Campestre, Cristina, Locatelli, Marcello, Guglielmi, Paolo, De Luca, Elisa, Bellagamba, Giuseppe, Menta, Sergio, Zengin, Gokhan, Celia, Christian, Di Marzio, Luisa, Carradori, Simone
Publicado 2017

Synthesis and biological evaluation of anti-Toxoplasma gondii activity of a novel scaffold of thiazolidinone derivatives

por Carradori, Simone, Secci, Daniela, Bizzarri, Bruna, Chimenti, Paola, De Monte, Celeste, Guglielmi, Paolo, Campestre, Cristina, Rivanera, Daniela, Bordón, Claudia, Jones-Brando, Lorraine
Publicado 2017

Synthesis and evaluation of a large library of nitroxoline derivatives as pancreatic cancer antiproliferative agents

por Veschi, Serena, Carradori, Simone, De Lellis, Laura, Florio, Rosalba, Brocco, Davide, Secci, Daniela, Guglielmi, Paolo, Spano, Mattia, Sobolev, Anatoly P., Cama, Alessandro
Publicado 2020

4-(3-Nitrophenyl)thiazol-2-ylhydrazone derivatives as antioxidants and selective hMAO-B inhibitors: synthesis, biological activity and computational analysis

por Secci, Daniela, Carradori, Simone, Petzer, Anél, Guglielmi, Paolo, D’Ascenzio, Melissa, Chimenti, Paola, Bagetta, Donatella, Alcaro, Stefano, Zengin, Gokhan, Petzer, Jacobus P., Ortuso, Francesco
Publicado 2019

Dual Carbonic Anhydrase IX/XII Inhibitors and Carbon Monoxide Releasing Molecules Modulate LPS-Mediated Inflammation in Mouse Macrophages

por Berrino, Emanuela, Carradori, Simone, Angeli, Andrea, Carta, Fabrizio, Supuran, Claudiu T., Guglielmi, Paolo, Coletti, Cecilia, Paciotti, Roberto, Schweikl, Helmut, Maestrelli, Francesca, Cerbai, Elisabetta, Gallorini, Marialucia
Publicado 2021

Synthesis and Evaluation of Thymol-Based Synthetic Derivatives as Dual-Action Inhibitors against Different Strains of H. pylori and AGS Cell Line

por Sisto, Francesca, Carradori, Simone, Guglielmi, Paolo, Spano, Mattia, Secci, Daniela, Granese, Arianna, Sobolev, Anatoly P., Grande, Rossella, Campestre, Cristina, Di Marcantonio, Maria Carmela, Mincione, Gabriella
Publicado 2021

Design, synthesis and biological activity of selective hCAs inhibitors based on 2-(benzylsulfinyl)benzoic acid scaffold

por Rotondi, Giulia, Guglielmi, Paolo, Carradori, Simone, Secci, Daniela, De Monte, Celeste, De Filippis, Barbara, Maccallini, Cristina, Amoroso, Rosa, Cirilli, Roberto, Akdemir, Atilla, Angeli, Andrea, Supuran, Claudiu T.
Publicado 2019

Synthesis and Biological Evaluation of Carvacrol-Based Derivatives as Dual Inhibitors of H. pylori Strains and AGS Cell Proliferation

por Sisto, Francesca, Carradori, Simone, Guglielmi, Paolo, Traversi, Carmen Beatrice, Spano, Mattia, Sobolev, Anatoly P., Secci, Daniela, Di Marcantonio, Maria Carmela, Haloci, Entela, Grande, Rossella, Mincione, Gabriella
Publicado 2020

Novel Insights on Human Carbonic Anhydrase Inhibitors Based on Coumalic Acid: Design, Synthesis, Molecular Modeling Investigation, and Biological Studies

por Pontecorvi, Virginia, Mori, Mattia, Picarazzi, Francesca, Zara, Susi, Carradori, Simone, Cataldi, Amelia, Angeli, Andrea, Berrino, Emanuela, Chimenti, Paola, Ciogli, Alessia, Secci, Daniela, Guglielmi, Paolo, Supuran, Claudiu T.
Publicado 2022

Benzo[b]tiophen-3-ol derivatives as effective inhibitors of human monoamine oxidase: design, synthesis, and biological activity

por Guglielmi, Paolo, Secci, Daniela, Petzer, Anél, Bagetta, Donatella, Chimenti, Paola, Rotondi, Giulia, Ferrante, Claudio, Recinella, Lucia, Leone, Sheila, Alcaro, Stefano, Zengin, Gokhan, Petzer, Jacobus P., Ortuso, Francesco, Carradori, Simone
Publicado 2019