Steroidal Antagonists of Progesterone- and Prostaglandin E(1)-Induced Activation of the Cation Channel of Sperm

por Carlson, Erick J., Georg, Gunda I., Hawkinson, Jon E.
Publicado 2022

Design, Synthesis, and in Vitro and in Vivo Evaluation of Ouabain Analogues as Potent and Selective Na,K-ATPase α4 Isoform Inhibitors for Male Contraception

por Syeda, Shameem Sultana, Sánchez, Gladis, Hong, Kwon Ho, Hawkinson, Jon E., Georg, Gunda I., Blanco, Gustavo
Publicado 2018

Development of WEE2 kinase inhibitors as novel non-hormonal female contraceptives that target meiosis

por Hanna, Carol B, Mudaliar, Deepti, John, Kristen, Allen, C Leigh, Sun, Luxin, Hawkinson, Jon E, Schönbrunn, Ernst, Georg, Gunda I, Jensen, Jeffrey T
Publicado 2020

Structure–Activity Studies of N‐Butyl‐1‐deoxynojirimycin (NB‐DNJ) Analogues: Discovery of Potent and Selective Aminocyclopentitol Inhibitors of GBA1 and GBA2

por Gu, Xingxian, Gupta, Vijayalaxmi, Yang, Yan, Zhu, Jin‐Yi, Carlson, Erick J., Kingsley, Carolyn, Tash, Joseph S., Schönbrunn, Ernst, Hawkinson, Jon, Georg, Gunda I.
Publicado 2017

Discovery and Characterization of Multiple Classes of Human CatSper Blockers

por Carlson, Erick J., Francis, Rawle, Liu, Yutong, Li, Ping, Lyon, Maximilian, Santi, Celia M., Hook, Derek J., Hawkinson, Jon E., Georg, Gunda I.
Publicado 2022

The Fungal Sexual Pheromone Sirenin Activates the Human CatSper Channel Complex

por Syeda, Shameem Sultana, Carlson, Erick J., Miller, Melissa R., Francis, Rawle, Clapham, David E., Lishko, Polina V., Hawkinson, Jon E., Hook, Derek, Georg, Gunda I.
Publicado 2015

The anti-parasitic agent suramin and several of its analogues are inhibitors of the DNA binding protein Mcm10

por Paulson, Carolyn N., John, Kristen, Baxley, Ryan M., Kurniawan, Fredy, Orellana, Kayo, Francis, Rawle, Sobeck, Alexandra, Eichman, Brandt F., Chazin, Walter J., Aihara, Hideki, Georg, Gunda I., Hawkinson, Jon E., Bielinsky, Anja-Katrin
Publicado 2019

Automated Live-Cell Imaging of Synapses in Rat and Human Neuronal Cultures

por Green, Matthew V., Pengo, Thomas, Raybuck, Jonathan D., Naqvi, Tahmina, McMullan, Hannah M., Hawkinson, Jon E., Marron Fernandez de Velasco, Ezequiel, Muntean, Brian S., Martemyanov, Kirill A., Satterfield, Rachel, Young, Samuel M., Thayer, Stanley A.
Publicado 2019

Development of allosteric and selective CDK2 inhibitors for contraception with negative cooperativity to cyclin binding

por Faber, Erik B., Sun, Luxin, Tang, Jian, Roberts, Emily, Ganeshkumar, Sornakala, Wang, Nan, Rasmussen, Damien, Majumdar, Abir, Hirsch, Laura E., John, Kristen, Yang, An, Khalid, Hira, Hawkinson, Jon E., Levinson, Nicholas M., Chennathukuzhi, Vargheese, Harki, Daniel A., Schönbrunn, Ernst, Georg, Gunda I.
Publicado 2023

Amyloid precursor protein selective gamma-secretase inhibitors for treatment of Alzheimer's disease

por Basi, Guriqbal S, Hemphill, Susanna, Brigham, Elizabeth F, Liao, Anna, Aubele, Danielle L, Baker, Jeanne, Barbour, Robin, Bova, Michael, Chen, Xiao-Hua, Dappen, Michael S, Eichenbaum, Tovah, Goldbach, Erich, Hawkinson, Jon, Lawler-Herbold, Rose, Hu, Kang, Hui, Terence, Jagodzinski, Jacek J, Keim, Pamela S, Kholodenko, Dora, Latimer, Lee H, Lee, Mike, Marugg, Jennifer, Mattson, Matthew N, McCauley, Scott, Miller, James L, Motter, Ruth, Mutter, Linda, Neitzel, Martin L, Ni, Huifang, Nguyen, Lan, Quinn, Kevin, Ruslim, Lany, Semko, Christopher M, Shapiro, Paul, Smith, Jenifer, Soriano, Ferdie, Szoke, Balazs, Tanaka, Kevin, Tang, Pearl, Tucker, John A, Ye, Xiacong Michael, Yu, Mei, Wu, Jing, Xu, Ying-zi, Garofalo, Albert W, Sauer, John Michael, Konradi, Andrei W, Ness, Daniel, Shopp, George, Pleiss, Michael A, Freedman, Stephen B, Schenk, Dale
Publicado 2010