Crystal structures of the A(2A) adenosine receptor and their use in medicinal chemistry

por Jacobson, Kenneth A
Publicado 2013

Editorial: Purinergic pharmacology, Volume II

por Ciruela, Francisco, Jacobson, Kenneth A.
Publicado 2023

Structural Probing and Molecular Modeling of the A(3) Adenosine Receptor: A Focus on Agonist Binding

por Ciancetta, Antonella, Jacobson, Kenneth A.
Publicado 2017

Editorial: Purinergic Pharmacology

por Ciruela, Francisco, Jacobson, Kenneth A.
Publicado 2019

In Silico Drug Design for Purinergic GPCRs: Overview on Molecular Dynamics Applied to Adenosine and P2Y Receptors

por Salmaso, Veronica, Jacobson, Kenneth A.
Publicado 2020

Purinergic Signaling in Liver Pathophysiology

por Jain, Shanu, Jacobson, Kenneth A.
Publicado 2021

Optical Control of Adenosine A(3) Receptor Signaling: Towards a Multimodal Phototherapy in Psoriasis?

por Ciruela, Francisco, Jacobson, Kenneth A.
Publicado 2022

Purinergic Signaling in Mast Cell Degranulation and Asthma

por Gao, Zhan-Guo, Jacobson, Kenneth A.
Publicado 2017

A(2B) Adenosine Receptor and Cancer

por Gao, Zhan-Guo, Jacobson, Kenneth A.
Publicado 2019

Adenosine-Related Mechanisms in Non-Adenosine Receptor Drugs

por Jacobson, Kenneth A., Reitman, Marc L.
Publicado 2020

Preface: special issue on medicinal chemistry of purines

por Jacobson, Kenneth A., Zablocki, Jeff, Bhagwat, Shripad
Publicado 2008

Portraying G Protein-Coupled Receptors with Fluorescent Ligands

por Ciruela, Francisco, Jacobson, Kenneth A., Fernández-Dueñas, Víctor
Publicado 2014

Species dependence of A(3) adenosine receptor pharmacology and function

por Gao, Zhan-Guo, Auchampach, John A., Jacobson, Kenneth A.
Publicado 2022

Evidence for the possible involvement of the P2Y(6) receptor in Ca(2+) mobilization and insulin secretion in mouse pancreatic islets

por Ohtani, Masahiro, Suzuki, Jun-ichiro, Jacobson, Kenneth A., Oka, Takami
Publicado 2008

Structural Probing of Off-Target G Protein-Coupled Receptor Activities within a Series of Adenosine/Adenine Congeners

por Paoletta, Silvia, Tosh, Dilip K., Salvemini, Daniela, Jacobson, Kenneth A.
Publicado 2014

Enhancement of Glucose Uptake in Mouse Skeletal Muscle Cells and Adipocytes by P2Y(6) Receptor Agonists

por Balasubramanian, Ramachandran, Robaye, Bernard, Boeynaems, Jean-Marie, Jacobson, Kenneth A.
Publicado 2014

Thermostabilization and purification of the human dopamine transporter (hDAT) in an inhibitor and allosteric ligand bound conformation

por Navratna, Vikas, Tosh, Dilip K., Jacobson, Kenneth A., Gouaux, Eric
Publicado 2018

Design and Synthesis of 2,6-Disubstituted-4′-Selenoadenosine-5′-N,N-Dimethyluronamide Derivatives as Human A(3) Adenosine Receptor Antagonists

por Choi, Hongseok, Jacobson, Kenneth A., Yu, Jinha, Jeong, Lak Shin
Publicado 2021

Stereospecific antiseizure activity in mouse and rat epilepsy models by a pyridinium inhibitor of TNFα/NFκB signaling

por Pollard, Bette S., Wen, Zhiwei, Jacobson, Kenneth A., Pollard, John R.
Publicado 2022

Historical and Current Adenosine Receptor Agonists in Preclinical and Clinical Development

por Jacobson, Kenneth A., Tosh, Dilip K., Jain, Shanu, Gao, Zhan-Guo
Publicado 2019