Identifying hotspots in land use land cover change and the drivers in a semi-arid region of India

por Duraisamy, Vijayasekaran, Bendapudi, Ramkumar, Jadhav, Ajit
Publicado 2018

A Grid Algorithm for High Throughput Fitting of Dose-Response Curve Data

por Wang, Yuhong, Jadhav, Ajit, Southal, Noel, Huang, Ruili, Nguyen, Dac-Trung
Publicado 2010

High-Throughput 1,536-Well Fluorescence Polarization Assays for α(1)-Acid Glycoprotein and Human Serum Albumin Binding

por Yasgar, Adam, Furdas, Silviya D., Maloney, David J., Jadhav, Ajit, Jung, Manfred, Simeonov, Anton
Publicado 2012

A High-Throughput Approach for Identification of Novel General Anesthetics

por Lea, Wendy A., Xi, Jin, Jadhav, Ajit, Lu, Louis, Austin, Christopher P., Simeonov, Anton, Eckenhoff, Roderic G.
Publicado 2009

Diverse Small Molecule Inhibitors of Human Apurinic/Apyrimidinic Endonuclease APE1 Identified from a Screen of a Large Public Collection

por Dorjsuren, Dorjbal, Kim, Daemyung, Vyjayanti, Vaddadi N., Maloney, David J., Jadhav, Ajit, Wilson, David M., Simeonov, Anton
Publicado 2012

A Comprehensive Strategy to Discover Inhibitors of the Translesion Synthesis DNA Polymerase κ

por Yamanaka, Kinrin, Dorjsuren, Dorjbal, Eoff, Robert L., Egli, Martin, Maloney, David J., Jadhav, Ajit, Simeonov, Anton, Lloyd, R. Stephen
Publicado 2012

Identification and Characterization of Inhibitors of Human Apurinic/apyrimidinic Endonuclease APE1

por Simeonov, Anton, Kulkarni, Avanti, Dorjsuren, Dorjbal, Jadhav, Ajit, Shen, Min, McNeill, Daniel R., Austin, Christopher P., Wilson, David M.
Publicado 2009

A High-Throughput Assay for Small Molecule Destabilizers of the KRAS Oncoprotein

por Carver, Joseph, Dexheimer, Thomas S., Hsu, Dennis, Weng, Meng-Tzu, Smith, Jordan L., Guha, Rajarshi, Jadhav, Ajit, Simeonov, Anton, Luo, Ji
Publicado 2014

A High Throughput Screen Identifies Potent and Selective Inhibitors to Human Epithelial 15-Lipoxygenase-2

por Jameson, J. Brian, Kantz, Auric, Schultz, Lena, Kalyanaraman, Chakrapani, Jacobson, Matthew P., Maloney, David J., Jadhav, Ajit, Simeonov, Anton, Holman, Theodore R.
Publicado 2014

Quantitative High-Throughput Screen Identifies Inhibitors of the Schistosoma mansoni Redox Cascade

por Simeonov, Anton, Jadhav, Ajit, Sayed, Ahmed A., Wang, Yuhong, Nelson, Michael E., Thomas, Craig J., Inglese, James, Williams, David L., Austin, Christopher P.
Publicado 2008

A novel P300 inhibitor reverses DUX4-mediated global histone H3 hyperacetylation, target gene expression, and cell death

por Bosnakovski, Darko, da Silva, Meiricris T., Sunny, Sithara T., Ener, Elizabeth T., Toso, Erik A., Yuan, Ce, Cui, Ziyou, Walters, Michael A., Jadhav, Ajit, Kyba, Michael
Publicado 2019

A High-Content Assay Enables the Automated Screening and Identification of Small Molecules with Specific ALDH1A1-Inhibitory Activity

por Yasgar, Adam, Titus, Steven A., Wang, Yuhong, Danchik, Carina, Yang, Shyh-Ming, Vasiliou, Vasilis, Jadhav, Ajit, Maloney, David J., Simeonov, Anton, Martinez, Natalia J.
Publicado 2017

Correction: A High-Content Assay Enables the Automated Screening and Identification of Small Molecules with Specific ALDH1A1-Inhibitory Activity

por Yasgar, Adam, Titus, Steven A., Wang, Yuhong, Danchik, Carina, Yang, Shyh-Ming, Vasiliou, Vasilis, Jadhav, Ajit, Maloney, David J., Simeonov, Anton, Martinez, Natalia J.
Publicado 2018

High-Affinity Inhibitors of Human NAD(+)-Dependent 15-Hydroxyprostaglandin Dehydrogenase: Mechanisms of Inhibition and Structure-Activity Relationships

por Niesen, Frank H., Schultz, Lena, Jadhav, Ajit, Bhatia, Chitra, Guo, Kunde, Maloney, David J., Pilka, Ewa S., Wang, Minghua, Oppermann, Udo, Heightman, Tom D., Simeonov, Anton
Publicado 2010

Inhibition of DNA Glycosylases via Small Molecule Purine Analogs

por Jacobs, Aaron C., Calkins, Marcus J., Jadhav, Ajit, Dorjsuren, Dorjbal, Maloney, David, Simeonov, Anton, Jaruga, Pawel, Dizdaroglu, Miral, McCullough, Amanda K., Lloyd, R. Stephen
Publicado 2013

A high-throughput screen to identify novel small molecule inhibitors of the Werner Syndrome Helicase-Nuclease (WRN)

por Sommers, Joshua A., Kulikowicz, Tomasz, Croteau, Deborah L., Dexheimer, Thomas, Dorjsuren, Dorjbal, Jadhav, Ajit, Maloney, David J., Simeonov, Anton, Bohr, Vilhelm A., Brosh, Robert M.
Publicado 2019

A platform of assays for the discovery of anti-Zika small-molecules with activity in a 3D-bioprinted outer-blood-retina model

por Dorjsuren, Dorjbal, Eastman, Richard T., Song, Min Jae, Yasgar, Adam, Chen, Yuchi, Bharti, Kapil, Zakharov, Alexey V., Jadhav, Ajit, Ferrer, Marc, Shi, Pei-Yong, Simeonov, Anton
Publicado 2022

Complementarity Between a Docking and a High-Throughput Screen in Discovering New Cruzain Inhibitors

por Ferreira, Rafaela S., Simeonov, Anton, Jadhav, Ajit, Eidam, Oliv, Mott, Bryan T., Keiser, Michael J., McKerrow, James H., Maloney, David J., Irwin, John J., Shoichet, Brian K.
Publicado 2010

A high-throughput screening platform for Polycystic Kidney Disease (PKD) drug repurposing utilizing murine and human ADPKD cells

por Asawa, Rosita R., Danchik, Carina, Zakharov, Alexey, Chen, Yuchi, Voss, Ty, Jadhav, Ajit, Wallace, Darren P., Trott, Josephine F., Weiss, Robert H., Simeonov, Anton, Martinez, Natalia J.
Publicado 2020

Author Correction: A high-throughput screening platform for Polycystic Kidney Disease (PKD) drug repurposing utilizing murine and human ADPKD cells

por Asawa, Rosita R., Danchik, Carina, Zakharov, Alexey, Chen, Yuchi, Voss, Ty, Jadhav, Ajit, Wallace, Darren P., Trott, Josephine F., Weiss, Robert H., Simeonov, Anton, Martinez, Natalia J.
Publicado 2022