4-Aminobenzoic Acid Derivatives: Converting Folate Precursor to Antimicrobial and Cytotoxic Agents

por Krátký, Martin, Konečná, Klára, Janoušek, Jiří, Brablíková, Michaela, Janďourek, Ondřej, Trejtnar, František, Stolaříková, Jiřina, Vinšová, Jarmila
Publicado 2019

Synthesis, Biological Evaluation, and In Silico Modeling of N-Substituted Quinoxaline-2-Carboxamides

por Bouz, Ghada, Bouz, Sarah, Janďourek, Ondřej, Konečná, Klára, Bárta, Pavel, Vinšová, Jarmila, Doležal, Martin, Zitko, Jan
Publicado 2021

Insight into the Antibacterial Action of Iodinated Imine, an Analogue of Rafoxanide: a Comprehensive Study of Its Antistaphylococcal Activity

por Krátký, Martin, Konečná, Klára, Janďourek, Ondřej, Diepoltová, Adéla, Vávrová, Pavlína, Voxová, Barbora, Vejsová, Marcela, Bárta, Pavel, Bősze, Szilvia
Publicado 2023

Synthesis of Novel Pyrazinamide Derivatives Based on 3-Chloropyrazine-2-carboxamide and Their Antimicrobial Evaluation

por Jandourek, Ondrej, Tauchman, Marek, Paterova, Pavla, Konecna, Klara, Navratilova, Lucie, Kubicek, Vladimir, Holas, Ondrej, Zitko, Jan, Dolezal, Martin
Publicado 2017

N-Substituted 5-Amino-6-methylpyrazine-2,3-dicarbonitriles: Microwave-Assisted Synthesis and Biological Properties

por Jandourek, Ondrej, Dolezal, Martin, Paterova, Pavla, Kubicek, Vladimir, Pesko, Matus, Kunes, Jiri, Coffey, Aidan, Guo, Jiahui, Kralova, Katarina
Publicado 2014

New Potentially Active Pyrazinamide Derivatives Synthesized Under Microwave Conditions

por Jandourek, Ondrej, Dolezal, Martin, Kunes, Jiri, Kubicek, Vladimir, Paterova, Pavla, Pesko, Matus, Buchta, Vladimir, Kralova, Katarina, Zitko, Jan
Publicado 2014

Novel Aminoguanidine Hydrazone Analogues: From Potential Antimicrobial Agents to Potent Cholinesterase Inhibitors

por Krátký, Martin, Štěpánková, Šárka, Konečná, Klára, Svrčková, Katarína, Maixnerová, Jana, Švarcová, Markéta, Janďourek, Ondřej, Trejtnar, František, Vinšová, Jarmila
Publicado 2021

Adenosine-Mimicking Derivatives of 3-Aminopyrazine-2-Carboxamide: Towards Inhibitors of Prolyl-tRNA Synthetase with Antimycobacterial Activity

por Pallabothula, Vinod Sukanth Kumar, Kerda, Marek, Juhás, Martin, Janďourek, Ondřej, Konečná, Klára, Bárta, Pavel, Paterová, Pavla, Zitko, Jan
Publicado 2022

5-Alkylamino-N-phenylpyrazine-2-carboxamides: Design, Preparation, and Antimycobacterial Evaluation

por Ambrożkiewicz, Weronika, Kučerová-Chlupáčová, Marta, Janďourek, Ondřej, Konečná, Klára, Paterová, Pavla, Bárta, Pavel, Vinšová, Jarmila, Doležal, Martin, Zitko, Jan
Publicado 2020

3-Substituted N-Benzylpyrazine-2-carboxamide Derivatives: Synthesis, Antimycobacterial and Antibacterial Evaluation

por Semelková, Lucia, Janďourek, Ondřej, Konečná, Klára, Paterová, Pavla, Navrátilová, Lucie, Trejtnar, František, Kubíček, Vladimír, Kuneš, Jiří, Doležal, Martin, Zitko, Jan
Publicado 2017

Derivatives of 3-Aminopyrazine-2-carboxamides: Synthesis, Antimicrobial Evaluation, and in Vitro Cytotoxicity

por Bouz, Ghada, Semelková, Lucia, Janďourek, Ondřej, Konečná, Klára, Paterová, Pavla, Navrátilová, Lucie, Kubíček, Vladimír, Kuneš, Jiří, Doležal, Martin, Zitko, Jan
Publicado 2019

Ureidopyrazine Derivatives: Synthesis and Biological Evaluation as Anti-Infectives and Abiotic Elicitors

por Bouz, Ghada, Juhás, Martin, Niklová, Pavlína, Janďourek, Ondřej, Paterová, Pavla, Janoušek, Jiří, Tůmová, Lenka, Kovalíková, Zuzana, Kastner, Petr, Doležal, Martin, Zitko, Jan
Publicado 2017

Design, Synthesis, Antimycobacterial Evaluation, and In Silico Studies of 3-(Phenylcarbamoyl)-pyrazine-2-carboxylic Acids

por Semelková, Lucia, Janošcová, Petra, Fernandes, Carlos, Bouz, Ghada, Janďourek, Ondřej, Konečná, Klára, Paterová, Pavla, Navrátilová, Lucie, Kuneš, Jiří, Doležal, Martin, Zitko, Jan
Publicado 2017

Novel Halogenated Pyrazine-Based Chalcones as Potential Antimicrobial Drugs †

por Kucerova-Chlupacova, Marta, Vyskovska-Tyllova, Veronika, Richterova-Finkova, Lenka, Kunes, Jiri, Buchta, Vladimir, Vejsova, Marcela, Paterova, Pavla, Semelkova, Lucia, Jandourek, Ondrej, Opletalova, Veronika
Publicado 2016

Substituted N-(Pyrazin-2-yl)benzenesulfonamides; Synthesis, Anti-Infective Evaluation, Cytotoxicity, and In Silico Studies

por Bouz, Ghada, Juhás, Martin, Pausas Otero, Lluis, Paredes de la Red, Cristina, Janďourek, Ondřej, Konečná, Klára, Paterová, Pavla, Kubíček, Vladimír, Janoušek, Jiří, Doležal, Martin, Zitko, Jan
Publicado 2019

N-Pyrazinoyl Substituted Amino Acids as Potential Antimycobacterial Agents—the Synthesis and Biological Evaluation of Enantiomers

por Juhás, Martin, Kučerová, Lucie, Horáček, Ondřej, Janďourek, Ondřej, Kubíček, Vladimír, Konečná, Klára, Kučera, Radim, Bárta, Pavel, Janoušek, Jiří, Paterová, Pavla, Kuneš, Jiří, Doležal, Martin, Zitko, Jan
Publicado 2020

Correction: Juhás et al. Improving Antimicrobial Activity and Physico-Chemical Properties by Isosteric Replacement of 2-Aminothiazole with 2-Aminooxazole. Pharmaceuticals 2022, 15,...

por Juhás, Martin, Bachtíková, Andrea, Nawrot, Daria Elżbieta, Hatoková, Paulína, Pallabothula, Vinod Sukanth Kumar, Diepoltová, Adéla, Janďourek, Ondřej, Bárta, Pavel, Konečná, Klára, Paterová, Pavla, Šesták, Vít, Zitko, Jan
Publicado 2023

Improving Antimicrobial Activity and Physico-Chemical Properties by Isosteric Replacement of 2-Aminothiazole with 2-Aminooxazole

por Juhás, Martin, Bachtíková, Andrea, Nawrot, Daria Elżbieta, Hatoková, Paulína, Pallabothula, Vinod Sukanth Kumar, Diepoltová, Adéla, Janďourek, Ondřej, Bárta, Pavel, Konečná, Klára, Paterová, Pavla, Šesták, Vít, Zitko, Jan
Publicado 2022

Semisynthetic Derivatives of Selected Amaryllidaceae Alkaloids as a New Class of Antimycobacterial Agents

por Maafi, Negar, Mamun, Abdullah Al, Janďourek, Ondřej, Maříková, Jana, Breiterová, Kateřina, Diepoltová, Adéla, Konečná, Klára, Hošťálková, Anna, Hulcová, Daniela, Kuneš, Jiří, Kohelová, Eliška, Koutová, Darja, Šafratová, Marcela, Nováková, Lucie, Cahlíková, Lucie
Publicado 2021

Alkaloids of Dicranostigma franchetianum (Papaveraceae) and Berberine Derivatives as a New Class of Antimycobacterial Agents

por Wijaya, Viriyanata, Janďourek, Ondřej, Křoustková, Jana, Hradiská-Breiterová, Kateřina, Korábečný, Jan, Sobolová, Kateřina, Kohelová, Eliška, Hošťálková, Anna, Konečná, Klára, Šafratová, Marcela, Vrabec, Rudolf, Kuneš, Jiří, Opletal, Lubomír, Chlebek, Jakub, Cahlíková, Lucie
Publicado 2022