Pyrazole-Based Thrombin Inhibitors with a Serine-Trapping Mechanism of Action: Synthesis and Biological Activity

por Dunker, Calvin, Imberg, Lukas, Siutkina, Alena I., Erbacher, Catharina, Daniliuc, Constantin G., Karst, Uwe, Kalinin, Dmitrii V.
Publicado 2022

Semisynthetic Approach toward Biologically Active Derivatives of Phenylspirodrimanes from S. chartarum

por Steinert, Katharina, Berg, Nina, Kalinin, Dmitrii V., Jagels, Annika, Würthwein, Ernst-Ulrich, Humpf, Hans-Ulrich, Kalinina, Svetlana
Publicado 2022

Microwave-Assisted Synthesis, Structure, and Preliminary Biological Evaluation of Novel 6-Methoxy-5,6-dihydro-5-azapurines

por Siutkina, Alena I., Kalinina, Svetlana, Liu, Rongfang, Heitman, Laura H., Junker, Anna, Daniliuc, Constantin G., Kalinin, Dmitrii V.
Publicado 2023

Microscale Parallel Synthesis of Acylated Aminotriazoles Enabling the Development of Factor XIIa and Thrombin Inhibitors

por Platte, Simon, Korff, Marvin, Imberg, Lukas, Balicioglu, Ilker, Erbacher, Catharina, Will, Jonas M., Daniliuc, Constantin G., Karst, Uwe, Kalinin, Dmitrii V.
Publicado 2021

Structure‐Based Design, Synthesis, and Biological Evaluation of Triazole‐Based smHDAC8 Inhibitors

por Kalinin, Dmitrii V., Jana, Sunit K., Pfafenrot, Maxim, Chakrabarti, Alokta, Melesina, Jelena, Shaik, Tajith B., Lancelot, Julien, Pierce, Raymond J., Sippl, Wolfgang, Romier, Christophe, Jung, Manfred, Holl, Ralph
Publicado 2020

Platelet functional abnormalities in pediatric patients with kaposiform hemangioendothelioma/Kasabach-Merritt phenomenon

por Martyanov, Alexey A., Tesakov, Ivan P., Khachatryan, Lili A., An, Olga I., Boldova, Anna E., Ignatova, Anastasia A., Koltsova, Ekaterina M., Korobkin, Julia-Jessica D., Podoplelova, Nadezhda A., Svidelskaya, Galina S., Yushkova, Eugenia, Novichkova, Galina A., Eble, Johannes A., Panteleev, Mikhail A., Kalinin, Dmitrii V., Sveshnikova, Anastasia N.
Publicado 2023