Facile access to 3-sulfonylquinolines via Knoevenagel condensation/aza-Wittig reaction cascade involving ortho-azidobenzaldehydes and β-ketosulfonamides and sulfones

por Malkova, Ksenia, Bubyrev, Andrey, Kalinin, Stanislav, Dar’in, Dmitry
Publicado 2023

Inhibitory activity against carbonic anhydrase IX and XII as a candidate selection criterion in the development of new anticancer agents

por Krasavin, Mikhail, Kalinin, Stanislav, Sharonova, Tatiana, Supuran, Claudiu T.
Publicado 2020

Filtered FCS: Species Auto- and Cross-Correlation Functions Highlight Binding and Dynamics in Biomolecules**

por Felekyan, Suren, Kalinin, Stanislav, Sanabria, Hugo, Valeri, Alessandro, Seidel, Claus A M
Publicado 2012

Biochemical profiling of anti-HIV prodrug Elsulfavirine (Elpida(®)) and its active form VM1500A against a panel of twelve human carbonic anhydrase isoforms

por Supuran, Claudiu T., Nocentini, Alessio, Yakubova, Elena, Savchuk, Nikolay, Kalinin, Stanislav, Krasavin, Mikhail
Publicado 2021

Primary mono- and bis-sulfonamides obtained via regiospecific sulfochlorination of N-arylpyrazoles: inhibition profile against a panel of human carbonic anhydrases

por Krasavin, Mikhail, Korsakov, Mikhail, Ronzhina, Oksana, Tuccinardi, Tiziano, Kalinin, Stanislav, Tanç, Muhammet, Supuran, Claudiu T.
Publicado 2017

Further validation of strecker-type α-aminonitriles as a new class of potent human carbonic anhydrase II inhibitors: hit expansion within the public domain using differential scann...

por Krasavin, Mikhail, Kalinin, Stanislav, Zozulya, Sergey, Griniukova, Anastasia, Borysko, Petro, Angeli, Andrea, Supuran, Claudiu T.
Publicado 2019

Screening of benzenesulfonamide in combination with chemically diverse fragments against carbonic anhydrase by differential scanning fluorimetry

por Krasavin, Mikhail, Kalinin, Stanislav, Zozulya, Sergey, Gryniukova, Anastasiia, Borysko, Petro, Angeli, Andrea, Supuran, Claudiu T.
Publicado 2019

Carbonic Anhydrase IX Inhibitors as Candidates for Combination Therapy of Solid Tumors

por Kalinin, Stanislav, Malkova, Anna, Sharonova, Tatiana, Sharoyko, Vladimir, Bunev, Alexander, Supuran, Claudiu T., Krasavin, Mikhail
Publicado 2021

Combining carbonic anhydrase and thioredoxin reductase inhibitory motifs within a single molecule dramatically increases its cytotoxicity

por Krasavin, Mikhail, Sharonova, Tatiana, Sharoyko, Vladimir, Zhukovsky, Daniil, Kalinin, Stanislav, Žalubovskis, Raivis, Tennikova, Tatiana, Supuran, Claudiu T.
Publicado 2020

Unraveling multi-state molecular dynamics in single-molecule FRET experiments. I. Theory of FRET-lines

por Barth, Anders, Opanasyuk, Oleg, Peulen, Thomas-Otavio, Felekyan, Suren, Kalinin, Stanislav, Sanabria, Hugo, Seidel, Claus A. M.
Publicado 2022

Diversely substituted sulfamides for fragment-based drug discovery of carbonic anhydrase inhibitors: synthesis and inhibitory profile

por Sharonova, Tatiana, Zhmurov, Petr, Kalinin, Stanislav, Nocentini, Alessio, Angeli, Andrea, Ferraroni, Marta, Korsakov, Mikhail, Supuran, Claudiu T., Krasavin, Mikhail
Publicado 2022

5-(Sulfamoyl)thien-2-yl 1,3-oxazole inhibitors of carbonic anhydrase II with hydrophilic periphery

por Kalinin, Stanislav, Kovalenko, Alexander, Valtari, Annika, Nocentini, Alessio, Gureev, Maxim, Urtti, Arto, Korsakov, Mikhail, Supuran, Claudiu T., Krasavin, Mikhail
Publicado 2022

1,2,4-Oxadiazole/2-Imidazoline Hybrids: Multi-target-directed Compounds for the Treatment of Infectious Diseases and Cancer

por Shetnev, Anton, Baykov, Sergey, Kalinin, Stanislav, Belova, Alexandra, Sharoyko, Vladimir, Rozhkov, Anton, Zelenkov, Lev, Tarasenko, Marina, Sadykov, Evgeny, Korsakov, Mikhail, Krasavin, Mikhail
Publicado 2019

Carbonic Anhydrase Inhibitors Induce Ferroptosis through Inhibition of AKT/FTH1 Signaling in Ewing Sarcoma Tumor Cells

por Fayzullina, Darya, Yakushov, Semyon, Kantserova, Kamilla, Belyaeva, Elizaveta, Aniskin, Denis, Tsibulnikov, Sergey, Fayzullina, Nafisa, Kalinin, Stanislav, Romantsova, Olga, Timashev, Peter S., Schroeder, Brett A., Ulasov, Ilya V.
Publicado 2023

Synthesis, Structure, and Antiproliferative Action of 2-Pyridyl Urea-Based Cu(II) Complexes

por Geyl, Kirill K., Baykov, Sergey V., Kalinin, Stanislav A., Bunev, Alexandr S., Troshina, Marina A., Sharonova, Tatiana V., Skripkin, Mikhail Yu., Kasatkina, Svetlana O., Presnukhina, Sofia I., Shetnev, Anton A., Krasavin, Mikhail Yu., Boyarskiy, Vadim P.
Publicado 2022