Trace amine-associated receptors at the cross-road between innate olfaction of amines, emotions, and adult neurogenesis

por Efimova, Evgeniya V., Katolikova, Nataliia V., Kanov, Evgeny V., Gainetdinov, Raul R.
Publicado 2021

The Expression of Trace Amine-Associated Receptors (TAARs) in Breast Cancer Is Coincident with the Expression of Neuroactive Ligand–Receptor Systems and Depends on Tumor Intrinsic...

por Vaganova, Anastasia N., Maslennikova, Daria D., Konstantinova, Valeria V., Kanov, Evgeny V., Gainetdinov, Raul R.
Publicado 2023

Novel 1-Amidino-4-Phenylpiperazines as Potent Agonists at Human TAAR1 Receptor: Rational Design, Synthesis, Biological Evaluation and Molecular Docking Studies

por Francesconi, Valeria, Cichero, Elena, Kanov, Evgeny V., Laurini, Erik, Pricl, Sabrina, Gainetdinov, Raul R., Tonelli, Michele
Publicado 2020

Discovery of Guanfacine as a Novel TAAR1 Agonist: A Combination Strategy through Molecular Modeling Studies and Biological Assays

por Cichero, Elena, Francesconi, Valeria, Casini, Beatrice, Casale, Monica, Kanov, Evgeny, Gerasimov, Andrey S., Sukhanov, Ilya, Savchenko, Artem, Espinoza, Stefano, Gainetdinov, Raul R., Tonelli, Michele
Publicado 2023

Discovery and In Vivo Efficacy of Trace Amine-Associated Receptor 1 (TAAR1) Agonist 4-(2-Aminoethyl)-N-(3,5-dimethylphenyl)piperidine-1-carboxamide Hydrochloride (AP163) for the Tr...

por Krasavin, Mikhail, Peshkov, Anatoly A., Lukin, Alexey, Komarova, Kristina, Vinogradova, Lyubov, Smirnova, Daria, Kanov, Evgeny V., Kuvarzin, Savelii R., Murtazina, Ramilya Z., Efimova, Evgeniya V., Gureev, Maxim, Onokhin, Kirill, Zakharov, Konstantin, Gainetdinov, Raul R.
Publicado 2022