Effect of Selected Silyl Groups on the Anticancer Activity of 3,4-Dibromo-5-Hydroxy-Furan-2(5H)-One Derivatives

por Kitel, Radoslaw, Byczek-Wyrostek, Anna, Hopko, Katarzyna, Kasprzycka, Anna, Walczak, Krzysztof
Publicado 2021

Synthesis and Cytotoxicity of 2,3-Enopyranosyl C-Linked Conjugates of Genistein

por Szeja, Wieslaw, Grynkiewicz, Grzegorz, Bieg, Tadeusz, Swierk, Piotr, Byczek, Anna, Papaj, Katarzyna, Kitel, Radosław, Rusin, Aleksandra
Publicado 2014

Computer- and NMR-Aided Design of Small-Molecule Inhibitors of the Hub1 Protein

por Reyes Romero, Atilio, Kubica, Katarzyna, Kitel, Radoslaw, Rodríguez, Ismael, Magiera-Mularz, Katarzyna, Dömling, Alexander, Holak, Tad A., Surmiak, Ewa
Publicado 2022

PD-L1 Inhibitors: Different Classes, Activities, and Mechanisms of Action

por Surmiak, Ewa, Magiera-Mularz, Katarzyna, Musielak, Bogdan, Muszak, Damian, Kocik-Krol, Justyna, Kitel, Radoslaw, Plewka, Jacek, Holak, Tad A., Skalniak, Lukasz
Publicado 2021

Hexokinase 2 Inhibition and Biological Effects of BNBZ and Its Derivatives: The Influence of the Number and Arrangement of Hydroxyl Groups

por Juszczak, Karolina, Kubicka, Anna, Kitel, Radosław, Dzido, Grzegorz, Łabieniec-Watała, Magdalena, Zawadzki, Serafin, Marczak, Agnieszka, Walczak, Krzysztof, Matczak, Karolina, Tomczyk, Mateusz D.
Publicado 2022

Analysis tools for single-monomer measurements of self-assembly processes

por Hoyer, Maria, Crevenna, Alvaro H., Kitel, Radoslaw, Willems, Kherim, Czub, Miroslawa, Dubin, Grzegorz, Van Dorpe, Pol, Holak, Tad A., Lamb, Don C.
Publicado 2022

Exploring the Surface of the Ectodomain of the PD-L1 Immune Checkpoint with Small-Molecule Fragments

por Kitel, Radoslaw, Rodríguez, Ismael, del Corte, Xabier, Atmaj, Jack, Żarnik, Magdalena, Surmiak, Ewa, Muszak, Damian, Magiera-Mularz, Katarzyna, Popowicz, Grzegorz M., Holak, Tad A., Musielak, Bogdan
Publicado 2022

Structural Determinants of Substrate Specificity of SplF Protease from Staphylococcus aureus

por Stach, Natalia, Karim, Abdulkarim, Golik, Przemyslaw, Kitel, Radoslaw, Pustelny, Katarzyna, Gruba, Natalia, Groborz, Katarzyna, Jankowska, Urszula, Kedracka-Krok, Sylwia, Wladyka, Benedykt, Drag, Marcin, Lesner, Adam, Dubin, Grzegorz
Publicado 2021

Design, Synthesis, and Biological Evaluation of Imidazopyridines as PD-1/PD-L1 Antagonists

por Butera, Roberto, Ważyńska, Marta, Magiera-Mularz, Katarzyna, Plewka, Jacek, Musielak, Bogdan, Surmiak, Ewa, Sala, Dominik, Kitel, Radoslaw, de Bruyn, Marco, Nijman, Hans W., Elsinga, Philip H., Holak, Tad A., Dömling, Alexander
Publicado 2021

Terphenyl-Based Small-Molecule Inhibitors of Programmed Cell Death-1/Programmed Death-Ligand 1 Protein–Protein Interaction

por Muszak, Damian, Surmiak, Ewa, Plewka, Jacek, Magiera-Mularz, Katarzyna, Kocik-Krol, Justyna, Musielak, Bogdan, Sala, Dominik, Kitel, Radoslaw, Stec, Malgorzata, Weglarczyk, Kazimierz, Siedlar, Maciej, Dömling, Alexander, Skalniak, Lukasz, Holak, Tad A.
Publicado 2021