Amide-to-Ester Substitution as a Strategy for Optimizing PROTAC Permeability and Cellular Activity

por Klein, Victoria G., Bond, Adam G., Craigon, Conner, Lokey, R. Scott, Ciulli, Alessio
Publicado 2021

Understanding and Improving the Membrane Permeability of VH032-Based PROTACs

por Klein, Victoria G., Townsend, Chad E., Testa, Andrea, Zengerle, Michael, Maniaci, Chiara, Hughes, Scott J., Chan, Kwok-Ho, Ciulli, Alessio, Lokey, R. Scott
Publicado 2020