FKBP Ligands—Where We Are and Where to Go?

por Kolos, Jürgen M., Voll, Andreas M., Bauder, Michael, Hausch, Felix
Publicado 2018

FKBP51 and FKBP12.6—Novel and tight interactors of Glomulin

por Hähle, Andreas, Geiger, Thomas M., Merz, Stephanie, Meyners, Christian, Tianqi, Mao, Kolos, Jürgen, Hausch, Felix
Publicado 2019

Development of NanoBRET‐Binding Assays for FKBP‐Ligand Profiling in Living Cells

por Gnatzy, Monika T., Geiger, Thomas M., Kuehn, Angela, Gutfreund, Niklas, Walz, Michael, Kolos, Jürgen M., Hausch, Felix
Publicado 2021

Deconstructing Protein Binding of Sulfonamides and Sulfonamide Analogues

por Purder, Patrick L., Meyners, Christian, Sugiarto, Wisely Oki, Kolos, Jürgen, Löhr, Frank, Gebel, Jakob, Nehls, Thomas, Dötsch, Volker, Lermyte, Frederik, Hausch, Felix
Publicado 2023

FKBP12 is a major regulator of ALK2 activity in multiple myeloma cells

por Quist-Løkken, Ingrid, Andersson-Rusch, Clara, Kastnes, Martin Haugrud, Kolos, Jürgen Markus, Jatzlau, Jerome, Hella, Hanne, Olsen, Oddrun Elise, Sundan, Anders, Knaus, Petra, Hausch, Felix, Holien, Toril
Publicado 2023

Macrocyclic FKBP51 Ligands Define a Transient Binding Mode with Enhanced Selectivity

por Voll, Andreas M., Meyners, Christian, Taubert, Martha C., Bajaj, Thomas, Heymann, Tim, Merz, Stephanie, Charalampidou, Anna, Kolos, Jürgen, Purder, Patrick L., Geiger, Thomas M., Wessig, Pablo, Gassen, Nils C., Bracher, Andreas, Hausch, Felix
Publicado 2021

Picomolar FKBP inhibitors enabled by a single water-displacing methyl group in bicyclic [4.3.1] aza-amides

por Kolos, Jürgen M., Pomplun, Sebastian, Jung, Sascha, Rieß, Benedikt, Purder, Patrick L., Voll, Andreas M., Merz, Stephanie, Gnatzy, Monika, Geiger, Thomas M., Quist-Løkken, Ingrid, Jatzlau, Jerome, Knaus, Petra, Holien, Toril, Bracher, Andreas, Meyners, Christian, Czodrowski, Paul, Krewald, Vera, Hausch, Felix
Publicado 2021