Substituted N-Benzylpyrazine-2-carboxamides: Synthesis and Biological Evaluation (†)

por Servusová, Barbora, Eibinová, Drahomíra, Doležal, Martin, Kubíček, Vladimír, Paterová, Pavla, Peško, Matúš, Kráľová, Katarína
Publicado 2012

Carbonyl Reduction of Flubendazole in the Human Liver: Strict Stereospecificity, Sex Difference, Low Risk of Drug Interactions

por Kubíček, Vladimír, Skálová, Lenka, Skarka, Adam, Králová, Věra, Holubová, Jana, Štěpánková, Jana, Šubrt, Zdeněk, Szotáková, Barbora
Publicado 2019

Direct Amination of Nitroquinoline Derivatives via Nucleophilic Displacement of Aromatic Hydrogen

por Wantulok, Jakub, Swoboda, Daniel, Nycz, Jacek E., Książek, Maria, Kusz, Joachim, Małecki, Jan Grzegorz, Kubíček, Vladimír
Publicado 2021

Synthesis of Novel Pyrazinamide Derivatives Based on 3-Chloropyrazine-2-carboxamide and Their Antimicrobial Evaluation

por Jandourek, Ondrej, Tauchman, Marek, Paterova, Pavla, Konecna, Klara, Navratilova, Lucie, Kubicek, Vladimir, Holas, Ondrej, Zitko, Jan, Dolezal, Martin
Publicado 2017

N-Substituted 5-Amino-6-methylpyrazine-2,3-dicarbonitriles: Microwave-Assisted Synthesis and Biological Properties

por Jandourek, Ondrej, Dolezal, Martin, Paterova, Pavla, Kubicek, Vladimir, Pesko, Matus, Kunes, Jiri, Coffey, Aidan, Guo, Jiahui, Kralova, Katarina
Publicado 2014

New Potentially Active Pyrazinamide Derivatives Synthesized Under Microwave Conditions

por Jandourek, Ondrej, Dolezal, Martin, Kunes, Jiri, Kubicek, Vladimir, Paterova, Pavla, Pesko, Matus, Buchta, Vladimir, Kralova, Katarina, Zitko, Jan
Publicado 2014

Nerolidol and Farnesol Inhibit Some Cytochrome P450 Activities but Did Not Affect Other Xenobiotic-Metabolizing Enzymes in Rat and Human Hepatic Subcellular Fractions

por Špičáková, Alena, Szotáková, Barbora, Dimunová, Diana, Myslivečková, Zuzana, Kubíček, Vladimír, Ambrož, Martin, Lněničková, Kateřina, Krasulová, Kristýna, Anzenbacher, Pavel, Skálová, Lenka
Publicado 2017

3-Substituted N-Benzylpyrazine-2-carboxamide Derivatives: Synthesis, Antimycobacterial and Antibacterial Evaluation

por Semelková, Lucia, Janďourek, Ondřej, Konečná, Klára, Paterová, Pavla, Navrátilová, Lucie, Trejtnar, František, Kubíček, Vladimír, Kuneš, Jiří, Doležal, Martin, Zitko, Jan
Publicado 2017

Synthesis, Antimycobacterial Activity and In Vitro Cytotoxicity of 5-Chloro-N-phenylpyrazine-2-carboxamides

por Zitko, Jan, Servusová, Barbora, Paterová, Pavla, Mandíková, Jana, Kubíček, Vladimír, Kučera, Radim, Hrabcová, Veronika, Kuneš, Jiří, Soukup, Ondřej, Doležal, Martin
Publicado 2013

Derivatives of 3-Aminopyrazine-2-carboxamides: Synthesis, Antimicrobial Evaluation, and in Vitro Cytotoxicity

por Bouz, Ghada, Semelková, Lucia, Janďourek, Ondřej, Konečná, Klára, Paterová, Pavla, Navrátilová, Lucie, Kubíček, Vladimír, Kuneš, Jiří, Doležal, Martin, Zitko, Jan
Publicado 2019

Design, Synthesis and Antimicrobial Evaluation of New N-(1-Hydroxy-1,3-dihydrobenzo[c][1,2]oxaborol-6-yl)(hetero)aryl-2-carboxamides as Potential Inhibitors of Mycobacterial Leucyl...

por Šlechta, Petr, Needle, Adam Anthony, Jand’ourek, Ondřej, Paterová, Pavla, Konečná, Klára, Bárta, Pavel, Kuneš, Jiří, Kubíček, Vladimír, Doležal, Martin, Kučerová-Chlupáčová, Marta
Publicado 2023

Synthesis and Biological Evaluation of N-Alkyl-3-(alkylamino)-pyrazine-2-carboxamides

por Semelkova, Lucia, Konecna, Klara, Paterova, Pavla, Kubicek, Vladimir, Kunes, Jiri, Novakova, Lucie, Marek, Jan, Naesens, Lieve, Pesko, Matus, Kralova, Katarina, Dolezal, Martin, Zitko, Jan
Publicado 2015

Substituted N-(Pyrazin-2-yl)benzenesulfonamides; Synthesis, Anti-Infective Evaluation, Cytotoxicity, and In Silico Studies

por Bouz, Ghada, Juhás, Martin, Pausas Otero, Lluis, Paredes de la Red, Cristina, Janďourek, Ondřej, Konečná, Klára, Paterová, Pavla, Kubíček, Vladimír, Janoušek, Jiří, Doležal, Martin, Zitko, Jan
Publicado 2019

N-Pyrazinoyl Substituted Amino Acids as Potential Antimycobacterial Agents—the Synthesis and Biological Evaluation of Enantiomers

por Juhás, Martin, Kučerová, Lucie, Horáček, Ondřej, Janďourek, Ondřej, Kubíček, Vladimír, Konečná, Klára, Kučera, Radim, Bárta, Pavel, Janoušek, Jiří, Paterová, Pavla, Kuneš, Jiří, Doležal, Martin, Zitko, Jan
Publicado 2020