(2R)-Ethyl 2-(5-bromo-2,3-dioxoindolin-1-yl)propanoate

por Kurkin, Alexander V., Bernovskaya, Anna A., Yurovskaya, Marina A., Rybakov, Victor B.
Publicado 2008

3-Hy­droxy-2,2-bis­(1H-pyrazol-1-yl)­cyclo­penta­none

por Rybakov, Victor B., Utkina, Anastasia A., Kurkin, Alexander V., Yurovskaya, Marina A.
Publicado 2012

(1R,3R,3aS,8aR)-4-Oxo-3-phenyl-1-[(1R)-1-phenyl­eth­yl]deca­hydro­cyclo­hepta­[b]pyrrol-1-ium bromide

por Rybakov, Victor B., Belov, Dmitry S., Lukyanenko, Evgeny R., Kurkin, Alexander V., Yurovskaya, Marina A.
Publicado 2012

Comparative Pharmacokinetics of a Dual Inhibitor of HIV-1, NBD-14189, in Rats and Dogs with a Proof-of-Concept Evaluation of Antiviral Potency in SCID-hu Mouse Model

por Stoddart, Cheryl A., Curreli, Francesca, Horrigan, Stephen, Altieri, Andrea, Kurkin, Alexander V., Debnath, Asim K.
Publicado 2022

Stress promotes RNA G-quadruplex folding in human cells

por Kharel, Prakash, Fay, Marta, Manasova, Ekaterina V., Anderson, Paul J., Kurkin, Alexander V., Guo, Junjie U., Ivanov, Pavel
Publicado 2023

Antiviral Activity and Crystal Structures of HIV-1 gp120 Antagonists

por Curreli, Francesca, Kwon, Young D., Nicolau, Isabella, Burgos, Giancarla, Altieri, Andrea, Kurkin, Alexander V., Verardi, Raffaello, Kwong, Peter D., Debnath, Asim K.
Publicado 2022

Discovery of Highly Potent Fusion Inhibitors with Potential Pan-Coronavirus Activity That Effectively Inhibit Major COVID-19 Variants of Concern (VOCs) in Pseudovirus-Based Assays

por Curreli, Francesca, Ahmed, Shahad, Victor, Sofia M. B., Drelich, Aleksandra, Panda, Siva S., Altieri, Andrea, Kurkin, Alexander V., Tseng, Chien-Te K., Hillyer, Christopher D., Debnath, Asim K.
Publicado 2021

In Vitro and In Vivo Pharmacological Characterization of a Novel TRPM8 Inhibitor Chemotype Identified by Small-Scale Preclinical Screening

por Iraci, Nunzio, Ostacolo, Carmine, Medina-Peris, Alicia, Ciaglia, Tania, Novoselov, Anton M., Altieri, Andrea, Cabañero, David, Fernandez-Carvajal, Asia, Campiglia, Pietro, Gomez-Monterrey, Isabel, Bertamino, Alessia, Kurkin, Alexander V.
Publicado 2022

The Antioxidant Cofactor Alpha-Lipoic Acid May Control Endogenous Formaldehyde Metabolism in Mammals

por Shindyapina, Anastasia V., Komarova, Tatiana V., Sheshukova, Ekaterina V., Ershova, Natalia M., Tashlitsky, Vadim N., Kurkin, Alexander V., Yusupov, Ildar R., Mkrtchyan, Garik V., Shagidulin, Murat Y., Dorokhov, Yuri L.
Publicado 2017

Structure-Based Identification and Biological Characterization of New NAPRT Inhibitors

por Franco, Jorge, Piacente, Francesco, Walter, Melanie, Fratta, Simone, Ghanem, Moustafa, Benzi, Andrea, Caffa, Irene, Kurkin, Alexander V., Altieri, Andrea, Herr, Patrick, Martínez-Bailén, Macarena, Robina, Inmaculada, Bruzzone, Santina, Nencioni, Alessio, Del Rio, Alberto
Publicado 2022