(2R)-Ethyl 2-(5-bromo-2,3-dioxoindolin-1-yl)propanoate

por Kurkin, Alexander V., Bernovskaya, Anna A., Yurovskaya, Marina A., Rybakov, Victor B.
Publicado 2008

3-Hy­droxy-2,2-bis­(1H-pyrazol-1-yl)­cyclo­penta­none

por Rybakov, Victor B., Utkina, Anastasia A., Kurkin, Alexander V., Yurovskaya, Marina A.
Publicado 2012

(1R,3R,3aS,8aR)-4-Oxo-3-phenyl-1-[(1R)-1-phenyl­eth­yl]deca­hydro­cyclo­hepta­[b]pyrrol-1-ium bromide

por Rybakov, Victor B., Belov, Dmitry S., Lukyanenko, Evgeny R., Kurkin, Alexander V., Yurovskaya, Marina A.
Publicado 2012

Comparative Pharmacokinetics of a Dual Inhibitor of HIV-1, NBD-14189, in Rats and Dogs with a Proof-of-Concept Evaluation of Antiviral Potency in SCID-hu Mouse Model

por Stoddart, Cheryl A., Curreli, Francesca, Horrigan, Stephen, Altieri, Andrea, Kurkin, Alexander V., Debnath, Asim K.
Publicado 2022

Stress promotes RNA G-quadruplex folding in human cells

por Kharel, Prakash, Fay, Marta, Manasova, Ekaterina V., Anderson, Paul J., Kurkin, Alexander V., Guo, Junjie U., Ivanov, Pavel
Publicado 2023

ZB-16, a Novel GPR119 Agonist, Relieves the Severity of Streptozotocin–Nicotinamide-Induced Diabetes in Rats

por Tyurenkov, Ivan N., Kurkin, Denis V., Bakulin, Dmitry A., Volotova, Elena V., Chafeev, Mikhail A., Smirnov, Alexey V., Morkovin, Evgeny I.
Publicado 2017

Chemistry and Hypoglycemic Activity of GPR119 Agonist ZB-16

por Tyurenkov, Ivan N., Kurkin, Denis V., Bakulin, Dmitry A., Volotova, Elena V., Morkovin, Evgeny I., Chafeev, Mikhail A., Karapetian, Ruben N.
Publicado 2018

PROTAC: targeted drug strategy. Principles and limitations

por Koroleva, O. A., Dutikova, Yu. V., Trubnikov, A. V., Zenov, F. A., Manasova, E. V., Shtil, A. A., Kurkin, A. V.
Publicado 2022

Antiviral Activity and Crystal Structures of HIV-1 gp120 Antagonists

por Curreli, Francesca, Kwon, Young D., Nicolau, Isabella, Burgos, Giancarla, Altieri, Andrea, Kurkin, Alexander V., Verardi, Raffaello, Kwong, Peter D., Debnath, Asim K.
Publicado 2022

Evaluation of the Efficiency of Oxygen–Helium Therapy for Patients with Covid-19-Associated Pneumonia

por Manuilov, V. M., Suvorov, A. V., Kurkin, S. V., Olenev, Yu. O., Pavlov, N. B., Logunov, A. T., Anikeev, D. A., Orlov, O. I.
Publicado 2023

Discovery of Highly Potent Fusion Inhibitors with Potential Pan-Coronavirus Activity That Effectively Inhibit Major COVID-19 Variants of Concern (VOCs) in Pseudovirus-Based Assays

por Curreli, Francesca, Ahmed, Shahad, Victor, Sofia M. B., Drelich, Aleksandra, Panda, Siva S., Altieri, Andrea, Kurkin, Alexander V., Tseng, Chien-Te K., Hillyer, Christopher D., Debnath, Asim K.
Publicado 2021

In Vitro and In Vivo Pharmacological Characterization of a Novel TRPM8 Inhibitor Chemotype Identified by Small-Scale Preclinical Screening

por Iraci, Nunzio, Ostacolo, Carmine, Medina-Peris, Alicia, Ciaglia, Tania, Novoselov, Anton M., Altieri, Andrea, Cabañero, David, Fernandez-Carvajal, Asia, Campiglia, Pietro, Gomez-Monterrey, Isabel, Bertamino, Alessia, Kurkin, Alexander V.
Publicado 2022

The Antioxidant Cofactor Alpha-Lipoic Acid May Control Endogenous Formaldehyde Metabolism in Mammals

por Shindyapina, Anastasia V., Komarova, Tatiana V., Sheshukova, Ekaterina V., Ershova, Natalia M., Tashlitsky, Vadim N., Kurkin, Alexander V., Yusupov, Ildar R., Mkrtchyan, Garik V., Shagidulin, Murat Y., Dorokhov, Yuri L.
Publicado 2017

Synthesis, structure, and biological activity of 4-hetaryl-2-pyrrolidones containing a pyrazole ring

por Gorodnicheva, Natal’ya V., Vasil’eva, Olga S., Ostroglyadov, Evgeny S., Baichurin, Ruslan I., Litvinov, Igor A., Tyurenkov, Ivan N., Kovalev, Nikolay S., Bakulin, Dmitry A., Kurkin, Denis V., Baichurina, Larisa V., Makarenko, Sergey V.
Publicado 2022

Structure-Based Identification and Biological Characterization of New NAPRT Inhibitors

por Franco, Jorge, Piacente, Francesco, Walter, Melanie, Fratta, Simone, Ghanem, Moustafa, Benzi, Andrea, Caffa, Irene, Kurkin, Alexander V., Altieri, Andrea, Herr, Patrick, Martínez-Bailén, Macarena, Robina, Inmaculada, Bruzzone, Santina, Nencioni, Alessio, Del Rio, Alberto
Publicado 2022

Neuroprotective action of Cortexin, Cerebrolysin and Actovegin in acute or chronic brain ischemia in rats

por Kurkin, Denis V., Bakulin, Dmitry A., Morkovin, Evgeny I., Kalatanova, Anna V., Makarenko, Igor E., Dorotenko, Artem R., Kovalev, Nikolay S., Dubrovina, Marina A., Verkholyak, Dmitry V., Abrosimova, Elizaveta E., Smirnov, Alexey V., Shmidt, Maksim V., Tyurenkov, Ivan N.
Publicado 2021