Identification of Novel Potential Inhibitors of Pteridine Reductase 1 in Trypanosoma brucei via Computational Structure-Based Approaches and in Vitro Inhibition Assays

por Kimuda, Magambo Phillip, Laming, Dustin, Hoppe, Heinrich C., Tastan Bishop, Özlem
Publicado 2019

Anti-Trypanosomal and Antimalarial Properties of Tetralone Derivatives and Structurally Related Benzocycloalkanones

por Beteck, Richard M., Legoabe, Lesetja J., Isaacs, Michelle, Khanye, Setshaba D., Laming, Dustin, Hoppe, Heinrich C.
Publicado 2019

New Quinolone-Based Thiosemicarbazones Showing Activity Against Plasmodium falciparum and Mycobacterium tuberculosis

por Beteck, Richard M., Seldon, Ronnett, Jordaan, Audrey, Warner, Digby F., Hoppe, Heinrich C., Laming, Dustin, Khanye, Setshaba D.
Publicado 2019

Easy-To-Access Quinolone Derivatives Exhibiting Antibacterial and Anti-Parasitic Activities

por Beteck, Richard M., Jordaan, Audrey, Seldon, Ronnett, Laming, Dustin, Hoppe, Heinrich C., Warner, Digby F., Khanye, Setshaba D.
Publicado 2021

Detection of the in vitro modulation of Plasmodium falciparum Arf1 by Sec7 and ArfGAP domains using a colorimetric plate-based assay

por Swart, Tarryn, Khan, Farrah D., Ntlantsana, Apelele, Laming, Dustin, Veale, Clinton G. L., Przyborski, Jude M., Edkins, Adrienne L., Hoppe, Heinrich C.
Publicado 2020

Coumarin-Annulated Ferrocenyl 1,3-Oxazine Derivatives Possessing In Vitro Antimalarial and Antitrypanosomal Potency

por Mbaba, Mziyanda, Dingle, Laura M. K., Zulu, Ayanda I., Laming, Dustin, Swart, Tarryn, de la Mare, Jo-Anne, Hoppe, Heinrich C., Edkins, Adrienne L., Khanye, Setshaba D.
Publicado 2021

Cinnamoyl-Oxaborole Amides: Synthesis and Their in Vitro Biological Activity

por Gumbo, Maureen, Beteck, Richard M., Mandizvo, Tawanda, Seldon, Ronnett, Warner, Digby F., Hoppe, Heinrich C., Isaacs, Michelle, Laming, Dustin, Tam, Christina C., Cheng, Luisa W., Liu, Nicole, Land, Kirkwood M., Khanye, Setshaba D.
Publicado 2018