Structure–Activity Relationship and Evaluation of Phenethylamine and Tryptamine Derivatives for Affinity towards 5-Hydroxytryptamine Type 2A Receptor

por Wang, Shujie, Zhu, Anlin, Paudel, Suresh, Jang, Choon-Gon, Lee, Yong Sup, Kim, Kyeong-Man
Publicado 2023

Design, Rational Repurposing, Synthesis, In Vitro Evaluation, Homology Modeling and In Silico Study of Sulfuretin Analogs as Potential Antileishmanial Hit Compounds

por Hassan, Ahmed H.E., Phan, Trong-Nhat, Choi, Yeonwoo, Moon, Suyeon, No, Joo Hwan, Lee, Yong Sup
Publicado 2022

Potential Functional Role of Phenethylamine Derivatives in Inhibiting Dopamine Reuptake: Structure–Activity Relationship

por Kundu, Dooti, Zhu, Anlin, Kim, Eunae, Paudel, Suresh, Jang, Choon-Gon, Lee, Yong Sup, Kim, Kyeong-Man
Publicado 2023

(1)H-NMR and (13)C-NMR dataset for some oxidative metabolites of CRA13 and their analogs

por Hassan, Ahmed H.E., Cho, Min Chang, Kim, Hye In, Yang, Ji Seul, Park, Kyung Tae, Lee, Yong Sup
Publicado 2018

The Natural Polypeptides as Significant Elastase Inhibitors

por Ahmad, Shabir, Saleem, Muhammad, Riaz, Naheed, Lee, Yong Sup, Diri, Reem, Noor, Ahmad, Almasri, Diena, Bagalagel, Alaa, Elsebai, Mahmoud Fahmi
Publicado 2020

Chemical transformation of cannabidiol into psychotropic cannabinoids under acidic reaction conditions: Identification of transformed products by GC–MS

por Jeong, Minsun, Lee, Sangin, Seo, Chaeyoung, Kwon, Eunjeong, Rho, Soohyang, Cho, Mansoo, Kim, Moon Yeon, Lee, Wonwoong, Lee, Yong Sup, Hong, Jongki
Publicado 2023

Pyrrolidine-based 3-deoxysphingosylphosphorylcholine analogs as possible candidates against neglected tropical diseases (NTDs): identification of hit compounds towards development...

por Hassan, Ahmed H. E., Phan, Trong-Nhat, Yoon, Seolmin, Lee, Cheol Jung, Jeon, Hye Rim, Kim, Seung-Hwan, No, Joo Hwan, Lee, Yong Sup
Publicado 2021

Design, Synthesis, and Repurposing of Rosmarinic Acid-β-Amino-α-Ketoamide Hybrids as Antileishmanial Agents

por Hassan, Ahmed H.E., Bayoumi, Waleed A., El-Sayed, Selwan M., Phan, Trong-Nhat, Oh, Taegeun, Ham, Gyeongpyo, Mahmoud, Kazem, No, Joo Hwan, Lee, Yong Sup
Publicado 2023

Comparative Metabolite Profiling of Wild and Cultivated Justicia procumbens L. Based on (1)H-NMR Spectroscopy and HPLC-DAD Analysis

por Lee, Hyunyong, Jeon, Jihyun, Yoon, Joobyoung, Kim, Seung-Hwan, Choi, Hyun Sik, Kang, Jong Seung, Lee, Yong Sup, Lee, Mase, Kim, Young Ho, Chang, Hwan Bong
Publicado 2020

Costunolide Triggers Apoptosis in Human Leukemia U937 Cells by Depleting Intracellular Thiols

por Choi, Jung‐Hye, Ha, Joohun, Park, Jae‐Hoon, Lee, Jae Yeol, Lee, Yong Sup, Park, Hee‐Juhn, Choi, Jong‐Won, Masuda, Yutaka, Nakaya, Kazuyasu, Lee, Kyung‐Tae
Publicado 2002

QSAR Model for Predicting the Cannabinoid Receptor 1 Binding Affinity and Dependence Potential of Synthetic Cannabinoids

por Lee, Wonyoung, Park, So-Jung, Hwang, Ji-Young, Hur, Kwang-Hyun, Lee, Yong Sup, Kim, Jongmin, Zhao, Xiaodi, Park, Aekyung, Min, Kyung Hoon, Jang, Choon-Gon, Park, Hyun-Ju
Publicado 2020

Design, synthesis, and study of novel phenethyl-based antitumor phospholipids downregulating p38 mitogen-activated protein kinase

por Hassan, Ahmed H. E., Oh, Yeon Il, Lee, Chae Hyeon, Kim, Yeon Ju, Cho, Soo Bin, Alam, Md. Maqusood, Park, Sang-Eun, Chung, Kyung-Sook, Lee, Kyung-Tae, Lee, Yong Sup
Publicado 2023

Deletion of Cryab increases the vulnerability of mice to the addiction-like effects of the cannabinoid JWH-018 via upregulation of striatal NF-κB expression

por Sayson, Leandro Val, Ortiz, Darlene Mae, Lee, Hyun Jun, Kim, Mikyung, Custodio, Raly James Perez, Yun, Jaesuk, Lee, Chae Hyeon, Lee, Yong Sup, Cha, Hye Jin, Cheong, Jae Hoon, Kim, Hee Jin
Publicado 2023

Abuse Potential of Synthetic Cannabinoids: AM-1248, CB-13, and PB-22

por Hur, Kwang-Hyun, Ma, Shi-Xun, Lee, Bo-Ram, Ko, Yong-Hyun, Seo, Jee-Yeon, Ryu, Hye Won, Kim, Hye Jin, Yoon, Seolmin, Lee, Yong-Sup, Lee, Seok-Yong, Jang, Choon-Gon
Publicado 2021

The Anti-Proliferative Activity of the Hybrid TMS-TMF-4f Compound Against Human Cervical Cancer Involves Apoptosis Mediated by STAT3 Inactivation

por Hong, Joo Young, Chung, Kyung-Sook, Shin, Ji-Sun, Lee, Jeong-Hun, Gil, Hyo-Sun, Lee, Hwi-Ho, Choi, Eunwoo, Choi, Jung-Hye, Hassan, Ahmed H.E., Lee, Yong Sup, Lee, Kyung-Tae
Publicado 2019

4-F-PCP, a Novel PCP Analog Ameliorates the Depressive-Like Behavior of Chronic Social Defeat Stress Mice via NMDA Receptor Antagonism

por Ortiz, Darlene Mae D., Kim, Mikyung, Lee, Hyun Jun, Botanas, Chrislean Jun, Custodio, Raly James Perez, Sayson, Leandro Val, Campomayor, Nicole Bon, Lee, Chaeyeon, Lee, Yong Sup, Cheong, Jae Hoon, Kim, Hee Jin
Publicado 2023

Rational repurposing, synthesis, in vitro and in silico studies of chromone-peptidyl hybrids as potential agents against Leishmania donovani

por Hassan, Ahmed H. E., Bayoumi, Waleed A., El-Sayed, Selwan M., Phan, Trong-Nhat, Kim, Yeon Ju, Lee, Chae Hyeon, Cho, Soo Bin, Oh, Taegeun, Ham, Gyeongpyo, Mahmoud, Kazem, No, Joo Hwan, Lee, Yong Sup
Publicado 2023

Positional scanning of natural product hispidol’s ring-B: discovery of highly selective human monoamine oxidase-B inhibitor analogues downregulating neuroinflammation for managemen...

por Hassan, Ahmed H. E., Kim, Hyeon Jeong, Gee, Min Sung, Park, Jong-Hyun, Jeon, Hye Rim, Lee, Cheol Jung, Choi, Yeonwoo, Moon, Suyeon, Lee, Danbi, Lee, Jong Kil, Park, Ki Duk, Lee, Yong Sup
Publicado 2022

Repurposing Synthetic Congeners of a Natural Product Aurone Unveils a Lead Antitumor Agent Inhibiting Folded P-Loop Conformation of MET Receptor Tyrosine Kinase

por Hassan, Ahmed H. E., Wang, Cai Yi, Lee, Cheol Jung, Jeon, Hye Rim, Choi, Yeonwoo, Moon, Suyeon, Lee, Chae Hyeon, Kim, Yeon Ju, Cho, Soo Bin, Mahmoud, Kazem, El-Sayed, Selwan M., Lee, Sang Kook, Lee, Yong Sup
Publicado 2023

Mosloflavone-Resveratrol Hybrid TMS-HDMF-5z Exhibits Potent In Vitro and In Vivo Anti-Inflammatory Effects Through NF-κB, AP-1, and JAK/STAT Inactivation

por Kim, Seo-Yeon, Hassan, Ahmed H.E., Chung, Kyung-Sook, Kim, Su-Yeon, Han, Hee-Soo, Lee, Hwi-Ho, Jung, Seang-Hwan, Lee, Kwang-Young, Shin, Ji-Sun, Jang, Eungyeong, Yoon, Seolmin, Lee, Yong Sup, Lee, Kyung-Tae
Publicado 2022