Benzoylphenyl thiocyanates are new, effective inhibitors of the mycobacterial resuscitation promoting factor B protein

por Demina, Galina R., Nikitushkin, Vadim D., Shleeva, Margarita O., Riabova, Olga B., Lepioshkin, Alexander Yu., Makarov, Vadim A., Kaprelyants, Arseny S.
Publicado 2017

Pyrrolo[2,3-e]indazole as a novel chemotype for both influenza A virus and pneumococcal neuraminidase inhibitors

por Egorova, Anna, Richter, Martina, Khrenova, Maria, Dietrich, Elisabeth, Tsedilin, Andrey, Kazakova, Elena, Lepioshkin, Alexander, Jahn, Birgit, Chernyshev, Vladimir, Schmidtke, Michaela, Makarov, Vadim
Publicado 2023

Synthesis and Evaluation of 9-Aminoacridines with SARS-CoV-2 Antiviral Activity

por Jones, Thane, Monakhova, Natalia, Guivel-Benhassine, Florence, Lepioshkin, Alexander, Bruel, Timothée, Lane, Thomas R., Schwartz, Olivier, Puhl, Ana C., Makarov, Vadim, Ekins, Sean
Publicado 2023

A New Benzothiazolthiazolidine Derivative, 11726172, Is Active In Vitro, In Vivo, and against Nonreplicating Cells of Mycobacterium tuberculosis

por Salina, Elena G., Postiglione, Umberto, Chiarelli, Laurent R., Recchia, Deborah, Záhorszká, Monika, Lepioshkin, Alexander, Monakhova, Natalia, Pál, Adrian, Porta, Alessio, Zanoni, Giuseppe, Korduláková, Jana, Kazakova, Elena, Sassera, Davide, Pasca, Maria Rosalia, Makarov, Vadim, Degiacomi, Giulia
Publicado 2022

Thiophenecarboxamide Derivatives Activated by EthA Kill Mycobacterium tuberculosis by Inhibiting the CTP Synthetase PyrG

por Mori, Giorgia, Chiarelli, Laurent R., Esposito, Marta, Makarov, Vadim, Bellinzoni, Marco, Hartkoorn, Ruben C., Degiacomi, Giulia, Boldrin, Francesca, Ekins, Sean, de Jesus Lopes Ribeiro, Ana Luisa, Marino, Leonardo B., Centárová, Ivana, Svetlíková, Zuzana, Blaško, Jaroslav, Kazakova, Elena, Lepioshkin, Alexander, Barilone, Nathalie, Zanoni, Giuseppe, Porta, Alessio, Fondi, Marco, Fani, Renato, Baulard, Alain R., Mikušová, Katarína, Alzari, Pedro M., Manganelli, Riccardo, de Carvalho, Luiz Pedro S., Riccardi, Giovanna, Cole, Stewart T., Pasca, Maria Rosalia
Publicado 2015