Amide-to-ester substitution as a stable alternative to N-methylation for increasing membrane permeability in cyclic peptides

por Hosono, Yuki, Uchida, Satoshi, Shinkai, Moe, Townsend, Chad E., Kelly, Colin N., Naylor, Matthew R., Lee, Hsiau-Wei, Kanamitsu, Kayoko, Ishii, Mayumi, Ueki, Ryosuke, Ueda, Takumi, Takeuchi, Koh, Sugita, Masatake, Akiyama, Yutaka, Lokey, Scott R., Morimoto, Jumpei, Sando, Shinsuke
Publicado 2023