A covalent antagonist for the human adenosine A(2A) receptor

por Yang, Xue, Dong, Guo, Michiels, Thomas J.M., Lenselink, Eelke B., Heitman, Laura, Louvel, Julien, IJzerman, Ad P.
Publicado 2016

Structure–Affinity Relationships and Structure–Kinetic Relationships of 1,2-Diarylimidazol-4-carboxamide Derivatives as Human Cannabinoid 1 Receptor Antagonists

por Xia, Lizi, de Vries, Henk, Lenselink, Eelke B., Louvel, Julien, Waring, Michael J., Cheng, Leifeng, Pahlén, Sara, Petersson, Maria J., Schell, Peter, Olsson, Roine I., Heitman, Laura H., Sheppard, Robert J., IJzerman, Adriaan P.
Publicado 2017

Design and Characterization of an Intracellular Covalent Ligand for CC Chemokine Receptor 2

por Ortiz Zacarías, Natalia V., Chahal, Kirti K., Šimková, Tereza, van der Horst, Cas, Zheng, Yi, Inoue, Asuka, Theunissen, Emy, Mallee, Lloyd, van der Es, Daan, Louvel, Julien, IJzerman, Adriaan P., Handel, Tracy M., Kufareva, Irina, Heitman, Laura H.
Publicado 2021

Predicting Binding Affinities for GPCR Ligands Using Free-Energy Perturbation

por Lenselink, Eelke B., Louvel, Julien, Forti, Anna F., van Veldhoven, Jacobus P. D., de Vries, Henk, Mulder-Krieger, Thea, McRobb, Fiona M., Negri, Ana, Goose, Joseph, Abel, Robert, van Vlijmen, Herman W. T., Wang, Lingle, Harder, Edward, Sherman, Woody, IJzerman, Adriaan P., Beuming, Thijs
Publicado 2016