AhR-Mediated, Non-Genomic Modulation of IDO1 Function

por Pallotta, Maria Teresa, Fallarino, Francesca, Matino, Davide, Macchiarulo, Antonio, Orabona, Ciriana
Publicado 2014

One Key and Multiple Locks: Substrate Binding in Structures of Tryptophan Dioxygenases and Hydroxylases

por Mammoli, Andrea, Riccio, Alessandra, Bianconi, Elisa, Coletti, Alice, Camaioni, Emidio, Macchiarulo, Antonio
Publicado 2021

Enantioselective HPLC Analysis to Assist the Chemical Exploration of Chiral Imidazolines

por Cerra, Bruno, Macchiarulo, Antonio, Carotti, Andrea, Camaioni, Emidio, Varfaj, Ina, Sardella, Roccaldo, Gioiello, Antimo
Publicado 2020

PROTACs bearing piperazine-containing linkers: what effect on their protonation state?

por Desantis, Jenny, Mammoli, Andrea, Eleuteri, Michela, Coletti, Alice, Croci, Federico, Macchiarulo, Antonio, Goracci, Laura
Publicado 2022

Docking Studies and Molecular Dynamic Simulations Reveal Different Features of IDO1 Structure

por Greco, Francesco Antonio, Bournique, Answald, Coletti, Alice, Custodi, Chiara, Dolciami, Daniela, Carotti, Andrea, Macchiarulo, Antonio
Publicado 2016

Synthesis and Quantitative Structure-Property Relationships of Side Chain-Modified Hyodeoxycholic Acid Derivatives

por Sabbatini, Paola, Filipponi, Paolo, Sardella, Roccaldo, Natalini, Benedetto, Nuti, Roberto, Macchiarulo, Antonio, Pellicciari, Roberto, Gioiello, Antimo
Publicado 2013

Environmentally Sustainable Achiral and Chiral Chromatographic Analysis of Amino Acids in Food Supplements

por Varfaj, Ina, Carotti, Andrea, Mangiapelo, Luciano, Cossignani, Lina, Taticchi, Agnese, Macchiarulo, Antonio, Ianni, Federica, Sardella, Roccaldo
Publicado 2022

Identification by Virtual Screening and In Vitro Testing of Human DOPA Decarboxylase Inhibitors

por Daidone, Frederick, Montioli, Riccardo, Paiardini, Alessandro, Cellini, Barbara, Macchiarulo, Antonio, Giardina, Giorgio, Bossa, Francesco, Borri Voltattorni, Carla
Publicado 2012

Indoleamine 2,3‐dioxygenase 1 (IDO1): an up‐to‐date overview of an eclectic immunoregulatory enzyme

por Pallotta, Maria Teresa, Rossini, Sofia, Suvieri, Chiara, Coletti, Alice, Orabona, Ciriana, Macchiarulo, Antonio, Volpi, Claudia, Grohmann, Ursula
Publicado 2021

Glucocorticoid-induced leucine zipper (GILZ)/NF-κB interaction: role of GILZ homo-dimerization and C-terminal domain

por Marco, Barbara Di, Massetti, Michela, Bruscoli, Stefano, Macchiarulo, Antonio, Virgilio, Rosa Di, Velardi, Enrico, Donato, Valerio, Migliorati, Graziella, Riccardi, Carlo
Publicado 2007

Turning a Tumor Microenvironment Pitfall into Opportunity: Discovery of Benzamidoxime as PD-L1 Ligand with pH-Dependent Potency

por Bianconi, Elisa, Riccio, Alessandra, Ruta, Luana, Bigiotti, Carlo, Carotti, Andrea, Moretti, Sonia, Cerra, Bruno, Gioiello, Antimo, Ferlin, Simone, Puxeddu, Efisio, Macchiarulo, Antonio
Publicado 2023

A back-door insight into the modulation of Src kinase activity by the polyamine spermidine

por Rossini, Sofia, Gargaro, Marco, Scalisi, Giulia, Bianconi, Elisa, Ambrosino, Sara, Panfili, Eleonora, Volpi, Claudia, Orabona, Ciriana, Macchiarulo, Antonio, Fallarino, Francesca, Mondanelli, Giada
Publicado 2023

Advances in indoleamine 2,3-dioxygenase 1 medicinal chemistry

por Coletti, Alice, Greco, Francesco Antonio, Dolciami, Daniela, Camaioni, Emidio, Sardella, Roccaldo, Pallotta, Maria Teresa, Volpi, Claudia, Orabona, Ciriana, Grohmann, Ursula, Macchiarulo, Antonio
Publicado 2017

The hope and hype of ellagic acid and urolithins as ligands of SARS-CoV-2 Nsp5 and inhibitors of viral replication

por Bianconi, Elisa, Gidari, Anna, Souma, Maria, Sabbatini, Samuele, Grifagni, Deborah, Bigiotti, Carlo, Schiaroli, Elisabetta, Comez, Lucia, Paciaroni, Alessandro, Cantini, Francesca, Francisci, Daniela, Macchiarulo, Antonio
Publicado 2023

Protective Effects of Commiphora erythraea Resin Constituents Against Cellular Oxidative Damage

por Marcotullio, Maria Carla, Messina, Federica, Curini, Massimo, Macchiarulo, Antonio, Cellanetti, Marco, Ricci, Donata, Giamperi, Laura, Bucchini, Anahi, Minelli, Alba, Mierla, Anna Lisa, Bellezza, Ilaria
Publicado 2011

The Combination of Molnupiravir with Nirmatrelvir or GC376 Has a Synergic Role in the Inhibition of SARS-CoV-2 Replication In Vitro

por Gidari, Anna, Sabbatini, Samuele, Schiaroli, Elisabetta, Bastianelli, Sabrina, Pierucci, Sara, Busti, Chiara, Comez, Lucia, Libera, Valeria, Macchiarulo, Antonio, Paciaroni, Alessandro, Vicenti, Ilaria, Zazzi, Maurizio, Francisci, Daniela
Publicado 2022

Critical Assessment of a Structure-Based Screening Campaign for IDO1 Inhibitors: Tips and Pitfalls

por Mammoli, Andrea, Bianconi, Elisa, Ruta, Luana, Riccio, Alessandra, Bigiotti, Carlo, Souma, Maria, Carotti, Andrea, Rossini, Sofia, Suvieri, Chiara, Pallotta, Maria Teresa, Grohmann, Ursula, Camaioni, Emidio, Macchiarulo, Antonio
Publicado 2022

Very-long-chain fatty acid sphingomyelin in nuclear lipid microdomains of hepatocytes and hepatoma cells: can the exchange from C24:0 to C16:0 affect signal proteins and vitamin D...

por Lazzarini, Andrea, Macchiarulo, Antonio, Floridi, Alessandro, Coletti, Alice, Cataldi, Samuela, Codini, Michela, Lazzarini, Remo, Bartoccini, Elisa, Cascianelli, Giacomo, Ambesi-Impiombato, Francesco Saverio, Beccari, Tommaso, Curcio, Francesco, Albi, Elisabetta
Publicado 2015

Distinct roles of immunoreceptor tyrosine‐based motifs in immunosuppressive indoleamine 2,3‐dioxygenase 1

por Albini, Elisa, Rosini, Verdiana, Gargaro, Marco, Mondanelli, Giada, Belladonna, Maria L., Pallotta, Maria Teresa, Volpi, Claudia, Fallarino, Francesca, Macchiarulo, Antonio, Antognelli, Cinzia, Bianchi, Roberta, Vacca, Carmine, Puccetti, Paolo, Grohmann, Ursula, Orabona, Ciriana
Publicado 2016

Biological Evaluation of New Thienopyridinium and Thienopyrimidinium Derivatives as Human Choline Kinase Inhibitors

por Luque-Navarro, Pilar María, Mariotto, Elena, Ballarotto, Marco, Rubbini, Gianluca, Aguilar-Troyano, Francisco José, Fasiolo, Alberto, Torretta, Archimede, Parisini, Emilio, Macchiarulo, Antonio, Laso, Alejandro, Marco, Carmen, Viola, Giampietro, Carrasco-Jimenez, María Paz, López-Cara, Luisa Carlota
Publicado 2022