Stereoselective synthesis of carbocyclic analogues of the nucleoside Q precursor (PreQ(0))

por Llona-Minguez, Sabin, Mackay, Simon P
Publicado 2014

Flavanoids induce expression of the suppressor of cytokine signalling 3 (SOCS3) gene and suppress IL-6-activated signal transducer and activator of transcription 3 (STAT3) activati...

por Wiejak, Jolanta, Dunlop, Julia, Mackay, Simon P., Yarwood, Stephen J.
Publicado 2013

Structure–Activity Relationships and Molecular Modeling of Sphingosine Kinase Inhibitors

por Baek, Dong Jae, MacRitchie, Neil, Anthony, Nahoum G., Mackay, Simon P., Pyne, Susan, Pyne, Nigel J., Bittman, Robert
Publicado 2013

Triphenylbutanamines: Kinesin Spindle Protein Inhibitors with in Vivo Antitumor Activity†

por Wang, Fang, Good, James A. D., Rath, Oliver, Kaan, Hung Yi Kristal, Sutcliffe, Oliver B., Mackay, Simon P., Kozielski, Frank
Publicado 2012

Targeting the Non-Canonical NF-κB Pathway in Chronic Lymphocytic Leukemia and Multiple Myeloma

por Burley, Thomas A., Kennedy, Emma, Broad, Georgia, Boyd, Melanie, Li, David, Woo, Timothy, West, Christopher, Ladikou, Eleni E., Ashworth, Iona, Fegan, Christopher, Johnston, Rosalynd, Mitchell, Simon, Mackay, Simon P., Pepper, Andrea G. S., Pepper, Chris
Publicado 2022

Identification of 2-Aminothiazole-4-Carboxylate Derivatives Active against Mycobacterium tuberculosis H(37)R(v) and the β-Ketoacyl-ACP Synthase mtFabH

por Al-Balas, Qosay, Anthony, Nahoum G., Al-Jaidi, Bilal, Alnimr, Amani, Abbott, Grainne, Brown, Alistair K., Taylor, Rebecca C., Besra, Gurdyal S., McHugh, Timothy D., Gillespie, Stephen H., Johnston, Blair F., Mackay, Simon P., Coxon, Geoffrey D.
Publicado 2009

Inhibitory Kappa B Kinase α (IKKα) Inhibitors That Recapitulate Their Selectivity in Cells against Isoform-Related Biomarkers

por Anthony, Nahoum G., Baiget, Jessica, Berretta, Giacomo, Boyd, Marie, Breen, David, Edwards, Joanne, Gamble, Carly, Gray, Alexander I., Harvey, Alan L., Hatziieremia, Sophia, Ho, Ka Ho, Huggan, Judith K., Lang, Stuart, Llona-Minguez, Sabin, Luo, Jia Lin, McIntosh, Kathryn, Paul, Andrew, Plevin, Robin J., Robertson, Murray N., Scott, Rebecca, Suckling, Colin J., Sutcliffe, Oliver B., Young, Louise C., Mackay, Simon P.
Publicado 2017