Optimization of Covalent MKK7 Inhibitors via Crude Nanomole-Scale Libraries

por Gehrtz, Paul, Marom, Shir, Bührmann, Mike, Hardick, Julia, Kleinbölting, Silke, Shraga, Amit, Dubiella, Christian, Gabizon, Ronen, Wiese, Jan N., Müller, Matthias P., Cohen, Galit, Babaev, Ilana, Shurrush, Khriesto, Avram, Liat, Resnick, Efrat, Barr, Haim, Rauh, Daniel, London, Nir
Publicado 2022

Sulfamate Acetamides as Self-Immolative Electrophiles for Covalent Ligand-Directed Release Chemistry

por Reddi, Rambabu N., Rogel, Adi, Gabizon, Ronen, Rawale, Dattatraya Gautam, Harish, Battu, Marom, Shir, Tivon, Barr, Arbel, Yamit Shorer, Gurwicz, Neta, Oren, Roni, David, Keren, Liu, Jingjing, Duberstein, Shirly, Itkin, Maxim, Malitsky, Sergey, Barr, Haim, Katz, Ben-Zion, Herishanu, Yair, Shachar, Idit, Shulman, Ziv, London, Nir
Publicado 2023