Polymyxins and quinazolines are LSD1/KDM1A inhibitors with unusual structural features

por Speranzini, Valentina, Rotili, Dante, Ciossani, Giuseppe, Pilotto, Simona, Marrocco, Biagina, Forgione, Mariantonietta, Lucidi, Alessia, Forneris, Federico, Mehdipour, Parinaz, Velankar, Sameer, Mai, Antonello, Mattevi, Andrea
Publicado 2016

Properly Substituted Analogues of BIX-01294 Lose Inhibition of G9a Histone Methyltransferase and Gain Selective Anti-DNA Methyltransferase 3A Activity

por Rotili, Dante, Tarantino, Domenico, Marrocco, Biagina, Gros, Christina, Masson, Véronique, Poughon, Valérie, Ausseil, Fréderic, Chang, Yanqi, Labella, Donatella, Cosconati, Sandro, Di Maro, Salvatore, Novellino, Ettore, Schnekenburger, Michael, Grandjenette, Cindy, Bouvy, Celine, Diederich, Marc, Cheng, Xiaodong, Arimondo, Paola B., Mai, Antonello
Publicado 2014

The histone methyltransferase EZH2 as a druggable target in SHH medulloblastoma cancer stem cells

por Miele, Evelina, Valente, Sergio, Alfano, Vincenzo, Silvano, Marianna, Mellini, Paolo, Borovika, Diana, Marrocco, Biagina, Po, Agnese, Besharat, Zein Mersini, Catanzaro, Giuseppina, Battaglia, Giuseppe, Abballe, Luana, Zwergel, Clemens, Stazi, Giulia, Milite, Ciro, Castellano, Sabrina, Tafani, Marco, Trapencieris, Peteris, Mai, Antonello, Ferretti, Elisabetta
Publicado 2017