SAT022 A Mechanism Of Resistance To Novel Inhibitors Of The N-Terminal Domain Of Androgen Receptor

por Setiawan, Josie, Mawji, Nasrin R, Tien, Amy H, Andersen, Raymond J, Sadar, Marianne D
Publicado 2023

Pin1 inhibition improves the efficacy of ralaniten compounds that bind to the N-terminal domain of androgen receptor

por Leung, Jacky K., Imamura, Yusuke, Kato, Minoru, Wang, Jun, Mawji, Nasrin R., Sadar, Marianne D.
Publicado 2021

Differential Gene Expression Profiles between N-Terminal Domain and Ligand-Binding Domain Inhibitors of Androgen Receptor Reveal Ralaniten Induction of Metallothionein by a Mechani...

por Obst, Jon K., Mawji, Nasrin R., Teskey, Simon J. L., Wang, Jun, Sadar, Marianne D.
Publicado 2022

Inhibition of androgen receptor by decoy molecules delays progression to castration-recurrent prostate cancer

por Myung, Jae-Kyung, Wang, Gang, Chiu, Helen H. L., Wang, Jun, Mawji, Nasrin R., Sadar, Marianne D.
Publicado 2017

Characterization of Niphatenones that Inhibit Androgen Receptor N-Terminal Domain

por Banuelos, Carmen A., Lal, Aaron, Tien, Amy H., Shah, Neel, Yang, Yu Chi, Mawji, Nasrin R., Meimetis, Labros G., Park, Jacob, Kunzhong, Jian, Andersen, Raymond J., Sadar, Marianne D.
Publicado 2014

Ralaniten Sensitizes Enzalutamide-Resistant Prostate Cancer to Ionizing Radiation in Prostate Cancer Cells that Express Androgen Receptor Splice Variants

por Banuelos, Carmen A., Ito, Yusuke, Obst, Jon K., Mawji, Nasrin R., Wang, Jun, Hirayama, Yukiyoshi, Leung, Jacky K., Tam, Teresa, Tien, Amy H., Andersen, Raymond J., Sadar, Marianne D.
Publicado 2020

Sintokamide A Is a Novel Antagonist of Androgen Receptor That Uniquely Binds Activation Function-1 in Its Amino-terminal Domain

por Banuelos, Carmen A., Tavakoli, Iran, Tien, Amy H., Caley, Daniel P., Mawji, Nasrin R., Li, Zhenzhen, Wang, Jun, Yang, Yu Chi, Imamura, Yusuke, Yan, Luping, Wen, Jian Guo, Andersen, Raymond J., Sadar, Marianne D.
Publicado 2016