METTL3 from Target Validation to the First Small-Molecule Inhibitors: A Medicinal Chemistry Journey

por Fiorentino, Francesco, Menna, Martina, Rotili, Dante, Valente, Sergio, Mai, Antonello
Publicado 2023

Anti-influenza A virus activity and structure–activity relationship of a series of nitrobenzoxadiazole derivatives

por Fiorentino, Francesco, De Angelis, Marta, Menna, Martina, Rovere, Annarita, Caccuri, Anna Maria, D’Acunzo, Francesca, Palamara, Anna Teresa, Nencioni, Lucia, Rotili, Dante, Mai, Antonello
Publicado 2021

Systematic Design of Adenosine Analogs as Inhibitors of a Clostridioides difficile-Specific DNA Adenine Methyltransferase Required for Normal Sporulation and Persistence

por Zhou, Jujun, Horton, John R., Menna, Martina, Fiorentino, Francesco, Ren, Ren, Yu, Dan, Hajian, Taraneh, Vedadi, Masoud, Mazzoccanti, Giulia, Ciogli, Alessia, Weinhold, Elmar, Hüben, Michael, Blumenthal, Robert M., Zhang, Xing, Mai, Antonello, Rotili, Dante, Cheng, Xiaodong
Publicado 2022

First-in-Class Selective Inhibitors of the Lysine Acetyltransferase KAT8

por Fiorentino, Francesco, Sementilli, Sara, Menna, Martina, Turrisi, Federica, Tomassi, Stefano, Pellegrini, Francesca Romana, Iuzzolino, Angela, D’Acunzo, Francesca, Feoli, Alessandra, Wapenaar, Hannah, Taraglio, Sophie, Fraschetti, Caterina, Del Bufalo, Donatella, Sbardella, Gianluca, Dekker, Frank J., Paiardini, Alessandro, Trisciuoglio, Daniela, Mai, Antonello, Rotili, Dante
Publicado 2023