E3 Ligases Meet Their Match: Fragment-Based Approaches to Discover New E3 Ligands and to Unravel E3 Biology

por Michaelides, Iacovos N., Collie, Gavin W.
Publicado 2023

Correction to “E3 Ligases Meet Their Match: Fragment-Based Approaches to Discover New E3 Ligands and to Unravel E3 Biology”

por Michaelides, Iacovos N., Collie, Gavin W.
Publicado 2023

Selective targeting of non-centrosomal AURKA functions through use of a targeted protein degradation tool

por Wang, Richard, Ascanelli, Camilla, Abdelbaki, Ahmed, Fung, Alex, Rasmusson, Tim, Michaelides, Iacovos, Roberts, Karen, Lindon, Catherine
Publicado 2021

Structural Basis for Targeting the Folded P-Loop Conformation of c-MET

por Collie, Gavin W., Michaelides, Iacovos N., Embrey, Kevin, Stubbs, Christopher J., Börjesson, Ulf, Dale, Ian L., Snijder, Arjan, Barlind, Louise, Song, Kun, Khurana, Puneet, Phillips, Christopher, Storer, R. Ian
Publicado 2020

Discovery and Optimization of the First ATP Competitive Type-III c-MET Inhibitor

por Michaelides, Iacovos N., Collie, Gavin W., Börjesson, Ulf, Vasalou, Christina, Alkhatib, Omar, Barlind, Louise, Cheung, Tony, Dale, Ian L., Embrey, Kevin J., Hennessy, Edward J., Khurana, Puneet, Koh, Cheryl M., Lamb, Michelle L., Liu, Jianming, Moss, Thomas A., O’Neill, Daniel J., Phillips, Christopher, Shaw, Joseph, Snijder, Arjan, Storer, R. Ian, Stubbs, Christopher J., Han, Fujin, Li, Chengzhi, Qiao, Jingchuan, Sun, Dong-Qing, Wang, Jingwen, Wang, Peng, Yang, Wenzhen
Publicado 2023