GSK6853, a Chemical Probe for Inhibition of the BRPF1 Bromodomain

por Bamborough, Paul, Barnett, Heather A., Becher, Isabelle, Bird, Mark J., Chung, Chun-wa, Craggs, Peter D., Demont, Emmanuel H., Diallo, Hawa, Fallon, David J., Gordon, Laurie J., Grandi, Paola, Hobbs, Clare I., Hooper-Greenhill, Edward, Jones, Emma J., Law, Robert P., Le Gall, Armelle, Lugo, David, Michon, Anne-Marie, Mitchell, Darren J., Prinjha, Rab K., Sheppard, Robert J., Watson, Allan J. B., Watson, Robert J.
Publicado 2016

Modulation of macrophage inflammatory function through selective inhibition of the epigenetic reader protein SP140

por Ghiboub, Mohammed, Koster, Jan, Craggs, Peter D., Li Yim, Andrew Y. F., Shillings, Anthony, Hutchinson, Sue, Bingham, Ryan P., Gatfield, Kelly, Hageman, Ishtu L., Yao, Gang, O’Keefe, Heather P., Coffin, Aaron, Patel, Amish, Sloan, Lisa A., Mitchell, Darren J., Hayhow, Thomas G., Lunven, Laurent, Watson, Robert J., Blunt, Christopher E., Harrison, Lee A., Bruton, Gordon, Kumar, Umesh, Hamer, Natalie, Spaull, John R., Zwijnenburg, Danny A., Welting, Olaf, Hakvoort, Theodorus B. M., te Velde, Anje A., van Limbergen, Johan, Henneman, Peter, Prinjha, Rab K., de Winther, Menno P. J., Harker, Nicola R., Tough, David F., de Jonge, Wouter J.
Publicado 2022