Bioluminescence Resonance Energy Transfer Based G Protein-Activation Assay to Probe Duration of Antagonism at the Histamine H(3) Receptor

por Mocking, Tamara A. M., Buzink, Maurice C. M. L., Leurs, Rob, Vischer, Henry F.
Publicado 2019

MPP(+)-Induced Changes in Cellular Impedance as a Measure for Organic Cation Transporter (SLC22A1-3) Activity and Inhibition

por Mocking, Tamara A. M., Sijben, Hubert J., Vermeulen, Yimé W., IJzerman, Adriaan P., Heitman, Laura H.
Publicado 2022

Optimization of Peptide Linker-Based Fluorescent Ligands for the Histamine H(1) Receptor

por Kok, Zhi Yuan, Stoddart, Leigh A., Mistry, Sarah J., Mocking, Tamara A. M., Vischer, Henry F., Leurs, Rob, Hill, Stephen J., Mistry, Shailesh N., Kellam, Barrie
Publicado 2022

A Photoswitchable Agonist for the Histamine H(3) Receptor, a Prototypic Family A G‐Protein‐Coupled Receptor

por Hauwert, Niels J., Mocking, Tamara A. M., Da Costa Pereira, Daniel, Lion, Ken, Huppelschoten, Yara, Vischer, Henry F., De Esch, Iwan J. P., Wijtmans, Maikel, Leurs, Rob
Publicado 2019

Covalent Inhibition of the Histamine H(3) Receptor

por Wágner, Gábor, Mocking, Tamara A. M., Kooistra, Albert J., Slynko, Inna, Ábrányi-Balogh, Péter, Keserű, György M., Wijtmans, Maikel, Vischer, Henry F., de Esch, Iwan J. P., Leurs, Rob
Publicado 2019

A toolbox of molecular photoswitches to modulate the CXCR3 chemokine receptor with light

por Gómez-Santacana, Xavier, de Munnik, Sabrina M, Mocking, Tamara A M, Hauwert, Niels J, Sun, Shanliang, Vijayachandran, Prashanna, de Esch, Iwan J P, Vischer, Henry F, Wijtmans, Maikel, Leurs, Rob
Publicado 2019

4-(3-Aminoazetidin-1-yl)pyrimidin-2-amines as High-Affinity Non-imidazole Histamine H(3) Receptor Agonists with in Vivo Central Nervous System Activity

por Wágner, Gábor, Mocking, Tamara A. M., Arimont, Marta, Provensi, Gustavo, Rani, Barbara, Silva-Marques, Bruna, Latacz, Gniewomir, Da Costa Pereira, Daniel, Karatzidou, Christina, Vischer, Henry F., Wijtmans, Maikel, Kieć-Kononowicz, Katarzyna, de Esch, Iwan J. P., Leurs, Rob
Publicado 2019

Synthesis and Characterization of a Bidirectional Photoswitchable Antagonist Toolbox for Real-Time GPCR Photopharmacology

por Hauwert, Niels J., Mocking, Tamara A. M., Da Costa Pereira, Daniel, Kooistra, Albert J., Wijnen, Lisa M., Vreeker, Gerda C. M., Verweij, Eléonore W. E., De Boer, Albertus H., Smit, Martine J., De Graaf, Chris, Vischer, Henry F., de Esch, Iwan J. P., Wijtmans, Maikel, Leurs, Rob
Publicado 2018