A 3D-QSAR model for cannabinoid receptor (CB2) ligands derived from aligned pharmacophors

por Günther, Robert, Deuther-Conrad, Winnie, Moldovan, Rareś, Fischer, Steffen, Brust, Peter
Publicado 2013

Synthesis and Preliminary Biological Evaluation of Indol-3-yl-oxoacetamides as Potent Cannabinoid Receptor Type 2 Ligands

por Moldovan, Rareş-Petru, Deuther-Conrad, Winnie, Horti, Andrew G., Brust, Peter
Publicado 2017

One-step radiosynthesis of the MCTs imaging agent [(18)F]FACH by aliphatic (18)F-labelling of a methylsulfonate precursor containing an unprotected carboxylic acid group

por Sadeghzadeh, Masoud, Moldovan, Rareş-Petru, Teodoro, Rodrigo, Brust, Peter, Wenzel, Barbara
Publicado 2019

Development of cannabinoid receptor (CB 2 R) ligands for application in PET studies - where to attach the radiolabel?

por Günther, Robert, Moldovan, Rareş, Lueg, Corinna, Deuther-Conrad, Winnie, Wünsch, Bernhard, Brust, Peter
Publicado 2014

Development of [(18)F]LU14 for PET Imaging of Cannabinoid Receptor Type 2 in the Brain

por Teodoro, Rodrigo, Gündel, Daniel, Deuther-Conrad, Winnie, Ueberham, Lea, Toussaint, Magali, Bormans, Guy, Brust, Peter, Moldovan, Rareş-Petru
Publicado 2021

Synthesis and Biological Evaluation of a Novel (18)F-Labeled Radiotracer for PET Imaging of the Adenosine A(2A) Receptor

por Lai, Thu Hang, Toussaint, Magali, Teodoro, Rodrigo, Dukić-Stefanović, Sladjana, Kranz, Mathias, Deuther-Conrad, Winnie, Moldovan, Rareş-Petru, Brust, Peter
Publicado 2021

Design, Radiosynthesis and Preliminary Biological Evaluation in Mice of a Brain-Penetrant (18)F-Labelled σ(2) Receptor Ligand

por Moldovan, Rareş-Petru, Gündel, Daniel, Teodoro, Rodrigo, Ludwig, Friedrich-Alexander, Fischer, Steffen, Toussaint, Magali, Schepmann, Dirk, Wünsch, Bernhard, Brust, Peter, Deuther-Conrad, Winnie
Publicado 2021

Radiofluorination and biological evaluation of N-aryl-oxadiazolyl-propionamides as potential radioligands for PET imaging of cannabinoid CB(2) receptors

por Teodoro, Rodrigo, Moldovan, Rareş-Petru, Lueg, Corinna, Günther, Robert, Donat, Cornelius K, Ludwig, Friedrich-Alexander, Fischer, Steffen, Deuther-Conrad, Winnie, Wünsch, Bernhard, Brust, Peter
Publicado 2013

Development of Fluorinated Non-Peptidic Ghrelin Receptor Ligands for Potential Use in Molecular Imaging

por Moldovan, Rareş-Petru, Els-Heindl, Sylvia, Worm, Dennis J., Kniess, Torsten, Kluge, Michael, Beck-Sickinger, Annette G., Deuther-Conrad, Winnie, Krügel, Ute, Brust, Peter
Publicado 2017

Synthesis, Structure–Activity Relationships, Radiofluorination, and Biological Evaluation of [(18)F]RM365, a Novel Radioligand for Imaging the Human Cannabinoid Receptor Type 2 (CB...

por Teodoro, Rodrigo, Gündel, Daniel, Deuther-Conrad, Winnie, Kazimir, Aleksandr, Toussaint, Magali, Wenzel, Barbara, Bormans, Guy, Hey-Hawkins, Evamarie, Kopka, Klaus, Brust, Peter, Moldovan, Rareş-Petru
Publicado 2023

Radiofluorination of an Anionic, Azide-Functionalized Teroligomer by Copper-Catalyzed Azide-Alkyne Cycloaddition

por Wenzel, Barbara, Schmid, Maximilian, Teodoro, Rodrigo, Moldovan, Rareş-Petru, Lai, Thu Hang, Mitrach, Franziska, Kopka, Klaus, Fischer, Björn, Schulz-Siegmund, Michaela, Brust, Peter, Hacker, Michael C.
Publicado 2023

Development of (18)F-Labeled Radiotracers for PET Imaging of the Adenosine A(2A) Receptor: Synthesis, Radiolabeling and Preliminary Biological Evaluation

por Lai, Thu Hang, Schröder, Susann, Toussaint, Magali, Dukić-Stefanović, Sladjana, Kranz, Mathias, Ludwig, Friedrich-Alexander, Fischer, Steffen, Steinbach, Jörg, Deuther-Conrad, Winnie, Brust, Peter, Moldovan, Rareş-Petru
Publicado 2021

Preclinical Incorporation Dosimetry of [(18)F]FACH—A Novel (18)F-Labeled MCT1/MCT4 Lactate Transporter Inhibitor for Imaging Cancer Metabolism with PET

por Sattler, Bernhard, Kranz, Mathias, Wenzel, Barbara, Jain, Nalin T., Moldovan, Rareş-Petru, Toussaint, Magali, Deuther-Conrad, Winnie, Ludwig, Friedrich-Alexander, Teodoro, Rodrigo, Sattler, Tatjana, Sadeghzadeh, Masoud, Sabri, Osama, Brust, Peter
Publicado 2020

Preclinical Evaluation of [(18)F]FACH in Healthy Mice and Piglets: An (18)F-Labeled Ligand for Imaging of Monocarboxylate Transporters with PET

por Gündel, Daniel, Sadeghzadeh, Masoud, Deuther-Conrad, Winnie, Wenzel, Barbara, Cumming, Paul, Toussaint, Magali, Ludwig, Friedrich-Alexander, Moldovan, Rareş-Petru, Kranz, Mathias, Teodoro, Rodrigo, Sattler, Bernhard, Sabri, Osama, Brust, Peter
Publicado 2021

Development of a Radiofluorinated Adenosine A(2B) Receptor Antagonist as Potential Ligand for PET Imaging

por Lindemann, Marcel, Moldovan, Rareş-Petru, Hinz, Sonja, Deuther-Conrad, Winnie, Gündel, Daniel, Dukic-Stefanovic, Sladjana, Toussaint, Magali, Teodoro, Rodrigo, Juhl, Cathleen, Steinbach, Jörg, Brust, Peter, Müller, Christa E., Wenzel, Barbara
Publicado 2020

Non-Invasive Assessment of Locally Overexpressed Human Adenosine 2A Receptors in the Heart of Transgenic Mice

por Gündel, Daniel, Lai, Thu Hang, Dukic-Stefanovic, Sladjana, Teodoro, Rodrigo, Deuther-Conrad, Winnie, Toussaint, Magali, Kopka, Klaus, Moldovan, Rareş-Petru, Boknik, Peter, Hofmann, Britt, Gergs, Ulrich, Neumann, Joachim, Brust, Peter
Publicado 2022

Quantitation of the A(2A) Adenosine Receptor Density in the Striatum of Mice and Pigs with [(18)F]FLUDA by Positron Emission Tomography

por Gündel, Daniel, Toussaint, Magali, Lai, Thu Hang, Deuther-Conrad, Winnie, Cumming, Paul, Schröder, Susann, Teodoro, Rodrigo, Moldovan, Rareş-Petru, Pan-Montojo, Francisco, Sattler, Bernhard, Kopka, Klaus, Sabri, Osama, Brust, Peter
Publicado 2022

PET Imaging of the Adenosine A(2A) Receptor in the Rotenone-Based Mouse Model of Parkinson’s Disease with [(18)F]FESCH Synthesized by a Simplified Two-Step One-Pot Radiolabeling St...

por Schröder, Susann, Lai, Thu Hang, Toussaint, Magali, Kranz, Mathias, Chovsepian, Alexandra, Shang, Qi, Dukić-Stefanović, Sladjana, Deuther-Conrad, Winnie, Teodoro, Rodrigo, Wenzel, Barbara, Moldovan, Rareş-Petru, Pan-Montojo, Francisco, Brust, Peter
Publicado 2020

Improved in vivo PET imaging of the adenosine A(2A) receptor in the brain using [(18)F]FLUDA, a deuterated radiotracer with high metabolic stability

por Lai, Thu Hang, Toussaint, Magali, Teodoro, Rodrigo, Dukić-Stefanović, Sladjana, Gündel, Daniel, Ludwig, Friedrich-Alexander, Wenzel, Barbara, Schröder, Susann, Sattler, Bernhard, Moldovan, Rareş-Petru, Falkenburger, Björn H., Sabri, Osama, Deuther-Conrad, Winnie, Brust, Peter
Publicado 2021

Development of Novel Analogs of the Monocarboxylate Transporter Ligand FACH and Biological Validation of One Potential Radiotracer for Positron Emission Tomography (PET) Imaging

por Sadeghzadeh, Masoud, Wenzel, Barbara, Gündel, Daniel, Deuther-Conrad, Winnie, Toussaint, Magali, Moldovan, Rareş-Petru, Fischer, Steffen, Ludwig, Friedrich-Alexander, Teodoro, Rodrigo, Jonnalagadda, Shirisha, Jonnalagadda, Sravan K., Schüürmann, Gerrit, Mereddy, Venkatram R., Drewes, Lester R., Brust, Peter
Publicado 2020