Synthesis and Evaluation of 9-Aminoacridines with SARS-CoV-2 Antiviral Activity

por Jones, Thane, Monakhova, Natalia, Guivel-Benhassine, Florence, Lepioshkin, Alexander, Bruel, Timothée, Lane, Thomas R., Schwartz, Olivier, Puhl, Ana C., Makarov, Vadim, Ekins, Sean
Publicado 2023

Chemical, Metabolic, and Cellular Characterization of a FtsZ Inhibitor Effective Against Burkholderia cenocepacia

por Chiarelli, Laurent R., Scoffone, Viola Camilla, Trespidi, Gabriele, Barbieri, Giulia, Riabova, Olga, Monakhova, Natalia, Porta, Alessio, Manina, Giulia, Riccardi, Giovanna, Makarov, Vadim, Buroni, Silvia
Publicado 2020

New 2-Ethylthio-4-methylaminoquinazoline derivatives inhibiting two subunits of cytochrome bc1 in Mycobacterium tuberculosis

por Lupien, Andréanne, Foo, Caroline Shi-Yan, Savina, Svetlana, Vocat, Anthony, Piton, Jérémie, Monakhova, Natalia, Benjak, Andrej, Lamprecht, Dirk A., Steyn, Adrie J. C., Pethe, Kevin, Makarov, Vadim A., Cole, Stewart T.
Publicado 2020

A New Benzothiazolthiazolidine Derivative, 11726172, Is Active In Vitro, In Vivo, and against Nonreplicating Cells of Mycobacterium tuberculosis

por Salina, Elena G., Postiglione, Umberto, Chiarelli, Laurent R., Recchia, Deborah, Záhorszká, Monika, Lepioshkin, Alexander, Monakhova, Natalia, Pál, Adrian, Porta, Alessio, Zanoni, Giuseppe, Korduláková, Jana, Kazakova, Elena, Sassera, Davide, Pasca, Maria Rosalia, Makarov, Vadim, Degiacomi, Giulia
Publicado 2022

Competitive Fitness of Essential Gene Knockdowns Reveals a Broad-Spectrum Antibacterial Inhibitor of the Cell Division Protein FtsZ

por Hogan, Andrew M., Scoffone, Viola C., Makarov, Vadim, Gislason, April S., Tesfu, Haben, Stietz, Maria S., Brassinga, Ann Karen C., Domaratzki, Michael, Li, Xuan, Azzalin, Alberto, Biggiogera, Marco, Riabova, Olga, Monakhova, Natalia, Chiarelli, Laurent R., Riccardi, Giovanna, Buroni, Silvia, Cardona, Silvia T.
Publicado 2018